Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50056378 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.160 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088696 (3-Amino-6-ethyl-2-{3-[4-(2-methoxy-phenyl)-piperaz...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088686 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50056384 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 0.650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088693 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088690 (3-Amino-5,6-dimethyl-2-{3-[4-(2-nitro-phenyl)-pipe...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50056384 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088695 (2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyls...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088692 (3-Amino-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-p...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50056362 (3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088688 (3-Amino-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-pro...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50056378 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088689 (1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088686 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 7.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088691 (3-Amino-6-ethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088687 (3-Amino-6-ethyl-2-{3-[4-(2-nitro-phenyl)-piperazin...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088695 (2-{3-[4-(2-Methoxy-phenyl)-piperazin-1-yl]-propyls...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088693 (3-Amino-2-{3-[4-(2-methoxy-phenyl)-piperazin-1-yl]...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088696 (3-Amino-6-ethyl-2-{3-[4-(2-methoxy-phenyl)-piperaz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 22 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088689 (1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 32 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088692 (3-Amino-2-{3-[4-(2-nitro-phenyl)-piperazin-1-yl]-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088690 (3-Amino-5,6-dimethyl-2-{3-[4-(2-nitro-phenyl)-pipe...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 123 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
5-hydroxytryptamine receptor 1A (Rattus norvegicus (rat)) | BDBM50088694 (1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 135 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptor of rat hippocampus membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088687 (3-Amino-6-ethyl-2-{3-[4-(2-nitro-phenyl)-piperazin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 195 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088688 (3-Amino-2-[3-(4-pyrimidin-2-yl-piperazin-1-yl)-pro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 366 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50056362 (3-Amino-5,6-dimethyl-2-[3-(4-pyrimidin-2-yl-pipera...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 434 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088694 (1-{3-[5-(2-Ethoxy-phenyl)-[1,3,4]thiadiazol-2-ylsu...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 437 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Alpha-1A/Alpha-1B/Alpha-1D adrenergic receptor (Rattus norvegicus (rat)-Rattus norvegicus (Rat)) | BDBM50088691 (3-Amino-6-ethyl-2-[3-(4-pyrimidin-2-yl-piperazin-1...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Università di Catania Curated by ChEMBL | Assay Description Displacement of [3H]prazosin from Alpha-1 adrenergic receptor of rat cortex membranes | Bioorg Med Chem Lett 10: 1089-92 (2000) BindingDB Entry DOI: 10.7270/Q25D8R2B | |||||||||||
More data for this Ligand-Target Pair |