Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097485 (CHEMBL3585872) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097489 (CHEMBL3585870) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097491 (CHEMBL3585876) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 470 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097486 (CHEMBL3585873) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.12E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097488 (CHEMBL3585869) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.49E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097484 (CHEMBL3585871) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.54E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097490 (CHEMBL3585875) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.63E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-specific 3',5'-cyclic phosphodiesterase 4D (Homo sapiens (Human)) | BDBM50097487 (CHEMBL3585874) | PDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.84E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Genoa Curated by ChEMBL | Assay Description Inhibition of human recombinant PDE4D3 expressed in baculoviral system using cAMP as substrate by fluorescence polarization assay | Bioorg Med Chem 23: 3426-35 (2015) Article DOI: 10.1016/j.bmc.2015.04.027 BindingDB Entry DOI: 10.7270/Q2NC62ZZ | |||||||||||
More data for this Ligand-Target Pair |