Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Translocator protein (Rattus norvegicus (rat)) | BDBM50430877 (CHEMBL2336480) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.180 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430878 (CHEMBL2336474) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50243007 (2-(2-(4-(2-Fluoroethoxy)phenyl)-5,7-dimethylpyrazo...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | 9.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50327238 (2-[2-(4'-Methoxyphenyl)-5,7-dimethylpyrazolo[1,5-a...) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430876 (CHEMBL2336473) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430887 (CHEMBL2336479) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 68 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430886 (CHEMBL2336476) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430885 (CHEMBL2336482) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 94 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430884 (CHEMBL2336483) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 157 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430883 (CHEMBL2336484) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 201 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430882 (CHEMBL2336478) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 252 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430881 (CHEMBL2336477) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 277 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430879 (CHEMBL2336475) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50430880 (CHEMBL2336481) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Institute of Imaging Science (VUIIS) Curated by ChEMBL | Assay Description Displacement of [3H]-PK 11195 from TSPO in rat C6 cell lysates after 2 hrs by scintillation counting analysis | J Med Chem 56: 3429-33 (2013) Article DOI: 10.1021/jm4001874 BindingDB Entry DOI: 10.7270/Q2Z3211Z | |||||||||||
More data for this Ligand-Target Pair |