Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM50150818 (CHEMBL3774575) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | PDB Article PubMed | n/a | n/a | 7.60 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Texas MD Anderson Cancer Center Curated by ChEMBL | Assay Description Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ... | J Med Chem 59: 1440-54 (2016) Article DOI: 10.1021/acs.jmedchem.5b00405 BindingDB Entry DOI: 10.7270/Q26975F4 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM50150821 (CHEMBL3775251) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Texas MD Anderson Cancer Center Curated by ChEMBL | Assay Description Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ... | J Med Chem 59: 1440-54 (2016) Article DOI: 10.1021/acs.jmedchem.5b00405 BindingDB Entry DOI: 10.7270/Q26975F4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM50150820 (CHEMBL3774933) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.30 | n/a | n/a | n/a | n/a | n/a | n/a |
The University of Texas MD Anderson Cancer Center Curated by ChEMBL | Assay Description Inhibition of human N-terminal His-tagged KDM4A (1 to 359 residues) expressed in Escherichia coli using biotin-H3K9me3 as substrate preincubated for ... | J Med Chem 59: 1440-54 (2016) Article DOI: 10.1021/acs.jmedchem.5b00405 BindingDB Entry DOI: 10.7270/Q26975F4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329912 ((s.e.)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329913 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(6-phenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329914 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-({2-[3-(1-met...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329915 ((rac)-{(1R,2R,3S,4R)-4-[(2-{3-[2-chloro-1-(hydroxy...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449269 (US10702504, Compound I-A6) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449285 (US10702504, Compound I-A10) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449294 (US10702504, Compound I-A11) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449296 (US10702504, Compound I-A12) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449304 (US10702504, Compound I-B2) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM449307 (US10702504, Compound I-B4) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM50150808 (CHEMBL3774507 | US10702504, Compound C) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Similars | PDB US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Transcription intermediary factor 1-alpha (Homo sapiens (Human)) | BDBM50150812 (CHEMBL3775853 | US10702504, Compound D) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Similars | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
DANA-FARBER CANCER INSTITUTE, INC. US Patent | Assay Description The alpha assay was used to assess the binding of the compounds of the application to TRIM24 at various concentrations. All compounds were added at c... | US Patent US10702504 (2020) BindingDB Entry DOI: 10.7270/Q22B921C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329847 ((rac)-[(1R,2R,3S,4R)-4-{[2-(6-chloro-1H-indol-3-yl...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329848 ((rac)-((1R,2R,3S,4R)-4-((2-(Dibenzo[b,d]thiophen-4...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329849 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chloro-2-(trifluorome...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329850 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(1,1,1-...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329853 ((rac)-((1R,2R,3S,4R)-4-((2-(Benzo[b]thiophen-4-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329854 ((rac)-[(1R,2R,3S,4R)-4-{[2-(9H-carbazol-2-yl)pyraz...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM347108 (US10202389, Compound I-063 | US10202389, Example 9...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329857 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329858 ((rac)-((1R,2R,3S,4R)-2,3-Dihydroxy-4-((2-(2-methox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329859 ((rac)-[(1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(2-phenyl...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329862 ((rac)-((1R,2R,3S,4R)-4-(2-(4-fluoro-2-methoxypheny...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329863 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzo[b]thiophe...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329864 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(2-methoyp...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329867 ((rac)-((1R,2R,3S,4R)-4-(2-(1H-indol-4-yl)pyrazolo[...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329868 ((rac)-((1R,2R,3S,4R)-4-(2-(3-(cyclopropylmethylthi...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329869 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(piperi...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329870 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-morphol...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329873 ((rac)-((1R,2R,3S,4R)-4-(2-(5-fluorobenzo[b]thiophe...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329874 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-meth...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329875 ((rac)-[(1R,2R,3S,4R)-4-{[2-(3-ethynylphenyl)pyrazo...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329876 ((rac)-((1R,2R,3S,4R)-4-(2-(3-(2-ethoxypropan-2-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329877 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(9-oxo-9H-...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329878 ((rac)-((1R,2R,3S,4R)-4-(2-(benzofuran-2-yl)pyrazol...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329879 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-oxop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329882 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(2-prop...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329883 ((rac)-((1R,2R,3S,4R)-4-(2-(6-chlorobenzo[b]thiophe...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329884 ((rac)-((1R,2R,3S,4R)-4-(2-(5-chlorobenzofuran-3-yl...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329885 ((rac)-((1R,2R,3S,4R)-4-(2-(dibenzo[b,d]furan-3-yl)...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329886 ((rac)-((1R,2R,3S,4R)-4-(2-(5-ethylbenzo[b]thiophen...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329888 ((rac)-methyl rel-5-[7-({(1R,2S,3R,4R)-2,3-dihydrox...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329889 ((rac)-((1R,2R,3S,4R)-4-(2-(5-fluoronaphthalen-1-yl...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329794 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-{[2-(1-naphth...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM354140 (US9796725, Compound I-099 | US9796725, Example 11) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329892 ((s.e.)-((1R,2R,3S,4R)-4-(2-(4-fluoronaphthalen-1-y...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
SUMO-activating enzyme subunit 2 (Homo sapiens (Human)) | BDBM329836 ((rac)-((1R,2R,3S,4R)-2,3-dihydroxy-4-(2-(3-(triflu...) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | US Patent | n/a | n/a | <10 | n/a | n/a | n/a | n/a | n/a | n/a |
Millennium Pharmaceuticals, Inc. US Patent | Assay Description he UAE enzymatic reaction totals 50 μL and contains 50 mmol HEPES (pH 7.5), 0.05% BSA, 2.5 mM MgCl2, 0.1 uM ATP, 8 nM GST-Ubc-2, 35 nM flag-ubiq... | US Patent US9796725 (2017) BindingDB Entry DOI: 10.7270/Q23T9KC6 | |||||||||||
More data for this Ligand-Target Pair |
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