Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Solute carrier family 22 member 1 (Mus musculus) | BDBM18512 (5-(4-chlorophenyl)-6-ethylpyrimidine-2,4-diamine |...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
RIKEN Center for Life Science Technologies Curated by ChEMBL | Assay Description Inhibition of mouse Oct1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analys... | Bioorg Med Chem 21: 7584-90 (2013) Article DOI: 10.1016/j.bmc.2013.10.041 BindingDB Entry DOI: 10.7270/Q2CN75C7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 1 (Mus musculus) | BDBM50416487 (CHEMBL1236196 | TETRABUTYLAMMONIUM) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank PC cid PC sid PDB UniChem Similars | PubMed | 7.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytes | J Pharmacol Exp Ther 292: 1146-52 (2000) BindingDB Entry DOI: 10.7270/Q2XS5WPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 1 (Mus musculus) | BDBM50420179 (CHEMBL2074857) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | PubMed | 1.98E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytes | J Pharmacol Exp Ther 292: 1146-52 (2000) BindingDB Entry DOI: 10.7270/Q2XS5WPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 1 (Mus musculus) | BDBM50149890 (CHEMBL9324 | tetraethylammonium) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid UniChem Patents Similars | PubMed | 1.28E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytes | J Pharmacol Exp Ther 292: 1146-52 (2000) BindingDB Entry DOI: 10.7270/Q2XS5WPJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Solute carrier family 22 member 1 (Mus musculus) | BDBM50079455 (CHEMBL46486 | tetramethylammonium) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 2.04E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of California Curated by ChEMBL | Assay Description TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytes | J Pharmacol Exp Ther 292: 1146-52 (2000) BindingDB Entry DOI: 10.7270/Q2XS5WPJ | |||||||||||
More data for this Ligand-Target Pair |