Compile Data Set for Download or QSAR

Found 835 hits Enz. Inhib. hit(s) with Target = 'Voltage-gated potassium channel subunit Kv1.5'   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50067880 (4-methoxy-7H-furo[3,2-g][1]benzopyran-7-one | 4-me...) Show SMILES COc1c2ccoc2cc2oc(=O)ccc12 Show InChI InChI=1S/C12H8O4/c1-14-12-7-2-3-11(13)16-10(7)6-9-8(12)4-5-15-9/h2-6H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL MCE KEGG PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	n/a	1.77E+5	n/a	n/a	n/a	n/a	n/a
University of Kiel Curated by ChEMBL					Assay Description Blockade of peak K+ currents against Kv1.5 gene				J Med Chem 41: 4542-9 (1998) Article DOI: 10.1021/jm981032o BindingDB Entry DOI: 10.7270/Q2B56HWK
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50067878 (9-Methoxy-furo[3',2':4,5]benzo[1,2-b][1,4]oxazin-3...) Show SMILES COc1c2ccoc2cc2oc(=O)cnc12 Show InChI InChI=1S/C11H7NO4/c1-14-11-6-2-3-15-7(6)4-8-10(11)12-5-9(13)16-8/h2-5H,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	2.70E+5	n/a	n/a	n/a	n/a	n/a
University of Kiel Curated by ChEMBL					Assay Description Blockade of peak K+ currents against Kv1.5 gene				J Med Chem 41: 4542-9 (1998) Article DOI: 10.1021/jm981032o BindingDB Entry DOI: 10.7270/Q2B56HWK
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196834 (US9212187, 10) Show SMILES CCN1c2ccc(CCCN(CCn3ccc4oc(C)cc4c3=O)Cc3ccncc3)cc2N(C)C(=O)C(C)(C)C1=O Show InChI InChI=1S/C33H39N5O4/c1-6-38-27-10-9-24(21-28(27)35(5)31(40)33(3,4)32(38)41)8-7-16-36(22-25-11-14-34-15-12-25)18-19-37-17-13-29-26(30(37)39)20-23(2)42-29/h9-15,17,20-21H,6-8,16,18-19,22H2,1-5H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	620	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196835 (US9212187, 15) Show SMILES Cn1c2ccc(OCCCCCN(CCCc3ccccc3)Cc3cccnc3)cc2ccc1=O Show InChI InChI=1S/C30H35N3O2/c1-32-29-16-15-28(22-27(29)14-17-30(32)34)35-21-7-3-6-19-33(24-26-12-8-18-31-23-26)20-9-13-25-10-4-2-5-11-25/h2,4-5,8,10-12,14-18,22-23H,3,6-7,9,13,19-21,24H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	810	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196836 (US9212187, 16) Show SMILES Cn1c2ccc(OCCCCCN(Cc3cccnc3)Cc3cccnc3)cc2ccc1=O Show InChI InChI=1S/C27H30N4O2/c1-30-26-11-10-25(17-24(26)9-12-27(30)32)33-16-4-2-3-15-31(20-22-7-5-13-28-18-22)21-23-8-6-14-29-19-23/h5-14,17-19H,2-4,15-16,20-21H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	510	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196837 (US9212187, 18) Show SMILES Cn1c2ccc(OCCCCCN(CCCc3ccccc3)c3cccnc3)cc2ccc1=O Show InChI InChI=1S/C29H33N3O2/c1-31-28-16-15-27(22-25(28)14-17-29(31)33)34-21-7-3-6-19-32(26-13-8-18-30-23-26)20-9-12-24-10-4-2-5-11-24/h2,4-5,8,10-11,13-18,22-23H,3,6-7,9,12,19-21H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	600	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196838 (US9212187, 35) Show SMILES O=C1NCCc2cc(OCCCN(CCc3cccnc3)Cc3ccncc3)ccc12 Show InChI InChI=1S/C25H28N4O2/c30-25-24-5-4-23(17-22(24)8-13-28-25)31-16-2-14-29(19-21-6-11-26-12-7-21)15-9-20-3-1-10-27-18-20/h1,3-7,10-12,17-18H,2,8-9,13-16,19H2,(H,28,30)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	940	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196839 (US9212187, 41) Show SMILES Cn1c2ccc(OCCCN(CCc3ccccn3)Cc3ccncc3)cc2ccc1=O Show InChI InChI=1S/C26H28N4O2/c1-29-25-8-7-24(19-22(25)6-9-26(29)31)32-18-4-16-30(20-21-10-14-27-15-11-21)17-12-23-5-2-3-13-28-23/h2-3,5-11,13-15,19H,4,12,16-18,20H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6.30E+3	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196840 (US9212187, 42) Show SMILES CN(CCN(CCCOc1ccc2n(C)c(=O)ccc2c1)Cc1ccncc1)C(=O)c1ccccc1 Show InChI InChI=1S/C29H32N4O3/c1-31(29(35)24-7-4-3-5-8-24)18-19-33(22-23-13-15-30-16-14-23)17-6-20-36-26-10-11-27-25(21-26)9-12-28(34)32(27)2/h3-5,7-16,21H,6,17-20,22H2,1-2H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.70E+3	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196841 (US9212187, 43) Show SMILES CCn1c2ccc(OCCCN(CCc3cccnc3)Cc3ccncc3)cc2ccc1=O Show InChI InChI=1S/C27H30N4O2/c1-2-31-26-8-7-25(19-24(26)6-9-27(31)32)33-18-4-16-30(21-23-10-14-28-15-11-23)17-12-22-5-3-13-29-20-22/h3,5-11,13-15,19-20H,2,4,12,16-18,21H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	320	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196842 (US9212187, 48) Show SMILES Cn1c2ccccc2cc(OCCCN(CCc2cccnc2)Cc2ccncc2)c1=O Show InChI InChI=1S/C26H28N4O2/c1-29-24-8-3-2-7-23(24)18-25(26(29)31)32-17-5-15-30(20-22-9-13-27-14-10-22)16-11-21-6-4-12-28-19-21/h2-4,6-10,12-14,18-19H,5,11,15-17,20H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	300	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196843 (US9212187, 104) Show SMILES Cn1c2ccc(OCCCCCN(CCc3cccnc3)C(=O)c3cccnc3)cc2ccc1=O Show InChI InChI=1S/C28H30N4O3/c1-31-26-11-10-25(19-23(26)9-12-27(31)33)35-18-4-2-3-16-32(17-13-22-7-5-14-29-20-22)28(34)24-8-6-15-30-21-24/h5-12,14-15,19-21H,2-4,13,16-18H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	1.40E+3	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196844 (US9212187, 317) Show SMILES CCN1c2ccc(CN(CCn3ccc4oc(C)cc4c3=O)Cc3cccnc3COC)cc2N(C)C(=O)C(C)(C)C1=O Show InChI InChI=1S/C33H39N5O5/c1-7-38-27-11-10-23(18-28(27)35(5)31(40)33(3,4)32(38)41)19-36(20-24-9-8-13-34-26(24)21-42-6)15-16-37-14-12-29-25(30(37)39)17-22(2)43-29/h8-14,17-18H,7,15-16,19-21H2,1-6H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	630	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196845 (US9212187, 318) Show SMILES CCN1c2ccc(CN(CCn3cc(C)c4occc4c3=O)Cc3cccnc3COC)cc2N(C)C(=O)C(C)(C)C1=O Show InChI InChI=1S/C33H39N5O5/c1-7-38-27-11-10-23(17-28(27)35(5)31(40)33(3,4)32(38)41)19-36(20-24-9-8-13-34-26(24)21-42-6)14-15-37-18-22(2)29-25(30(37)39)12-16-43-29/h8-13,16-18H,7,14-15,19-21H2,1-6H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	2.90E+3	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM196846 (US9212187, 330) Show SMILES CCN1c2ccc(CN(CCc3cccnc3)C(=O)Cc3cn(C)c4ccccc34)cc2N(C)C(=O)C(C)(C)C1=O Show InChI InChI=1S/C33H37N5O3/c1-6-38-28-14-13-24(18-29(28)36(5)31(40)33(2,3)32(38)41)21-37(17-15-23-10-9-16-34-20-23)30(39)19-25-22-35(4)27-12-8-7-11-26(25)27/h7-14,16,18,20,22H,6,15,17,19,21H2,1-5H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	860	n/a	n/a	n/a	n/a	n/a	n/a
OTSUKA PHARMACEUTICAL CO., LTD. US Patent					Assay Description CHO-K1 cell lines stably expressing human Kv1.5 channels were prepared in the following manner.Full-length human Kv1.5 cDNA was cloned from a human h...				US Patent US9212187 (2015) BindingDB Entry DOI: 10.7270/Q2J101ZW
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50146377 (CHEMBL94296 | N-((S)-1-Phenyl-propyl)-2-(toluene-4...) Show SMILES CC[C@H](NC(=O)c1ccccc1NS(=O)(=O)c1ccc(C)cc1)c1ccccc1 Show InChI InChI=1S/C23H24N2O3S/c1-3-21(18-9-5-4-6-10-18)24-23(26)20-11-7-8-12-22(20)25-29(27,28)19-15-13-17(2)14-16-19/h4-16,21,25H,3H2,1-2H3,(H,24,26)/t21-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharma Deutschland GmbH Curated by ChEMBL					Assay Description Inhibitory effect against human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytes				Bioorg Med Chem Lett 14: 2823-7 (2004) Article DOI: 10.1016/j.bmcl.2004.03.057 BindingDB Entry DOI: 10.7270/Q2RR1XPJ
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50146377 (CHEMBL94296 | N-((S)-1-Phenyl-propyl)-2-(toluene-4...) Show SMILES CC[C@H](NC(=O)c1ccccc1NS(=O)(=O)c1ccc(C)cc1)c1ccccc1 Show InChI InChI=1S/C23H24N2O3S/c1-3-21(18-9-5-4-6-10-18)24-23(26)20-11-7-8-12-22(20)25-29(27,28)19-15-13-17(2)14-16-19/h4-16,21,25H,3H2,1-2H3,(H,24,26)/t21-/m0/s1	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	700	n/a	n/a	n/a	n/a	n/a	n/a
Aventis Pharma Deutschland GmbH Curated by ChEMBL					Assay Description Inhibitory effect against human voltage-gated potassium channel subunit Kv1.5 expressed in Xenopus oocytes				Bioorg Med Chem Lett 14: 2823-7 (2004) Article DOI: 10.1016/j.bmcl.2004.03.057 BindingDB Entry DOI: 10.7270/Q2RR1XPJ
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50099574 (2-(3,4-Dimethyl-phenyl)-3-[2-(4-methoxy-phenyl)-et...) Show SMILES COc1ccc(CCN2C(SCC2=O)c2ccc(C)c(C)c2)cc1 Show InChI InChI=1S/C20H23NO2S/c1-14-4-7-17(12-15(14)2)20-21(19(22)13-24-20)11-10-16-5-8-18(23-3)9-6-16/h4-9,12,20H,10-11,13H2,1-3H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	PubMed	n/a	n/a	200	n/a	n/a	n/a	n/a	n/a	n/a
Abbott Laboratories Curated by ChEMBL					Assay Description Inhibition of voltage-gated potassium channel subunit Kv1.5				J Med Chem 44: 1627-53 (2001) BindingDB Entry DOI: 10.7270/Q218376D
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016362 (CHEMBL3262835) Show SMILES Clc1ccccc1OCCN1CCN(CC(=O)Nc2nccs2)CC1 Show InChI InChI=1S/C17H21ClN4O2S/c18-14-3-1-2-4-15(14)24-11-10-21-6-8-22(9-7-21)13-16(23)20-17-19-5-12-25-17/h1-5,12H,6-11,13H2,(H,19,20,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.39E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016363 (CHEMBL3262836) Show SMILES O=C(CN1CCN(CCOc2ccc(cc2)C#N)CC1)Nc1nccs1 Show InChI InChI=1S/C18H21N5O2S/c19-13-15-1-3-16(4-2-15)25-11-10-22-6-8-23(9-7-22)14-17(24)21-18-20-5-12-26-18/h1-5,12H,6-11,14H2,(H,20,21,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	970	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016364 (CHEMBL3262837) Show SMILES Clc1ccc(OCCN2CCN(CC(=O)Nc3nccs3)CC2)cc1 Show InChI InChI=1S/C17H21ClN4O2S/c18-14-1-3-15(4-2-14)24-11-10-21-6-8-22(9-7-21)13-16(23)20-17-19-5-12-25-17/h1-5,12H,6-11,13H2,(H,19,20,23)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.18E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016365 (CHEMBL3262839) Show SMILES O=C(CN1CCN(CCOc2ccc3ccccc3c2)CC1)Nc1nccs1 Show InChI InChI=1S/C21H24N4O2S/c26-20(23-21-22-7-14-28-21)16-25-10-8-24(9-11-25)12-13-27-19-6-5-17-3-1-2-4-18(17)15-19/h1-7,14-15H,8-13,16H2,(H,22,23,26)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.80E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016366 (CHEMBL3262840) Show SMILES O=C(N1CCN(CCOc2ccc(cc2)C#N)CC1)c1cccs1 Show InChI InChI=1S/C18H19N3O2S/c19-14-15-3-5-16(6-4-15)23-12-11-20-7-9-21(10-8-20)18(22)17-2-1-13-24-17/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.02E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016367 (CHEMBL3262841) Show SMILES Fc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C17H19FN2O2S/c18-14-3-5-15(6-4-14)22-12-11-19-7-9-20(10-8-19)17(21)16-2-1-13-23-16/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.27E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016368 (CHEMBL3262842) Show SMILES Brc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C17H19BrN2O2S/c18-14-3-5-15(6-4-14)22-12-11-19-7-9-20(10-8-19)17(21)16-2-1-13-23-16/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.22E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016369 (CHEMBL3262843) Show SMILES Clc1ccccc1OCCN1CCN(CC1)C(=O)c1cccs1 Show InChI InChI=1S/C17H19ClN2O2S/c18-14-4-1-2-5-15(14)22-12-11-19-7-9-20(10-8-19)17(21)16-6-3-13-23-16/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	9.74E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016370 (CHEMBL3262803) Show SMILES Clc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)c(Cl)c1 Show InChI InChI=1S/C17H18Cl2N2O2S/c18-13-3-4-15(14(19)12-13)23-10-9-20-5-7-21(8-6-20)17(22)16-2-1-11-24-16/h1-4,11-12H,5-10H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.48E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016371 (CHEMBL3262802) Show SMILES Clc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C17H19ClN2O2S/c18-14-3-5-15(6-4-14)22-12-11-19-7-9-20(10-8-19)17(21)16-2-1-13-23-16/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	720	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016297 (CHEMBL3262796) Show SMILES FC(F)(F)Oc1ccc(cc1)N1CCN(CC1)C(=O)c1cccs1 Show InChI InChI=1S/C16H15F3N2O2S/c17-16(18,19)23-13-5-3-12(4-6-13)20-7-9-21(10-8-20)15(22)14-2-1-11-24-14/h1-6,11H,7-10H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.84E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016298 (CHEMBL3262797) Show SMILES O=C(N1CCN(CCOc2ccccc2)CC1)c1cccs1 Show InChI InChI=1S/C17H20N2O2S/c20-17(16-7-4-14-22-16)19-10-8-18(9-11-19)12-13-21-15-5-2-1-3-6-15/h1-7,14H,8-13H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.75E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016299 (CHEMBL3262798) Show SMILES Cc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C18H22N2O2S/c1-15-4-6-16(7-5-15)22-13-12-19-8-10-20(11-9-19)18(21)17-3-2-14-23-17/h2-7,14H,8-13H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.52E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016300 (CHEMBL3262799) Show SMILES Cc1ccccc1OCCN1CCN(CC1)C(=O)c1cccs1 Show InChI InChI=1S/C18H22N2O2S/c1-15-5-2-3-6-16(15)22-13-12-19-8-10-20(11-9-19)18(21)17-7-4-14-23-17/h2-7,14H,8-13H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.35E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016301 (CHEMBL3262800) Show SMILES COc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C18H22N2O3S/c1-22-15-4-6-16(7-5-15)23-13-12-19-8-10-20(11-9-19)18(21)17-3-2-14-24-17/h2-7,14H,8-13H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.19E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016302 (CHEMBL3262801) Show SMILES FC(F)(F)Oc1ccc(OCCN2CCN(CC2)C(=O)c2cccs2)cc1 Show InChI InChI=1S/C18H19F3N2O3S/c19-18(20,21)26-15-5-3-14(4-6-15)25-12-11-22-7-9-23(10-8-22)17(24)16-2-1-13-27-16/h1-6,13H,7-12H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.44E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50151864 (CHEMBL184412 | DRONEDARONE | N-(2-butyl-3-(4-(3-(d...) Show SMILES CCCCN(CCCC)CCCOc1ccc(cc1)C(=O)c1c(CCCC)oc2ccc(NS(C)(=O)=O)cc12 Show InChI InChI=1S/C31H44N2O5S/c1-5-8-12-29-30(27-23-25(32-39(4,35)36)15-18-28(27)38-29)31(34)24-13-16-26(17-14-24)37-22-11-21-33(19-9-6-2)20-10-7-3/h13-18,23,32H,5-12,19-22H2,1-4H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL DrugBank MCE PC cid PC sid UniChem Patents	Article PubMed	n/a	n/a	2.37E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016303 (CHEMBL3262804) Show SMILES O=C(N1CCN(CCOc2ccccc2)CC1)c1ccccc1 Show InChI InChI=1S/C19H22N2O2/c22-19(17-7-3-1-4-8-17)21-13-11-20(12-14-21)15-16-23-18-9-5-2-6-10-18/h1-10H,11-16H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.88E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016304 (CHEMBL3262805) Show SMILES Clc1ccc(OCCN2CCN(CC2)C(=O)c2ccccc2)cc1 Show InChI InChI=1S/C19H21ClN2O2/c20-17-6-8-18(9-7-17)24-15-14-21-10-12-22(13-11-21)19(23)16-4-2-1-3-5-16/h1-9H,10-15H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.97E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016305 (CHEMBL3262806) Show SMILES O=C(N1CCN(CCOc2ccc(cc2)C#N)CC1)c1ccccc1 Show InChI InChI=1S/C20H21N3O2/c21-16-17-6-8-19(9-7-17)25-15-14-22-10-12-23(13-11-22)20(24)18-4-2-1-3-5-18/h1-9H,10-15H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.23E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016306 (CHEMBL3262807) Show SMILES Cc1ccc(OCCN2CCN(CC2)C(=O)c2ccccc2)cc1 Show InChI InChI=1S/C20H24N2O2/c1-17-7-9-19(10-8-17)24-16-15-21-11-13-22(14-12-21)20(23)18-5-3-2-4-6-18/h2-10H,11-16H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.53E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016307 (CHEMBL3262808) Show SMILES COc1ccc(cc1)C(=O)N1CCN(CCOc2ccccc2)CC1 Show InChI InChI=1S/C20H24N2O3/c1-24-18-9-7-17(8-10-18)20(23)22-13-11-21(12-14-22)15-16-25-19-5-3-2-4-6-19/h2-10H,11-16H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.61E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016308 (CHEMBL3262809) Show SMILES COc1ccc(cc1)C(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 Show InChI InChI=1S/C20H23ClN2O3/c1-25-18-6-2-16(3-7-18)20(24)23-12-10-22(11-13-23)14-15-26-19-8-4-17(21)5-9-19/h2-9H,10-15H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	5.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016319 (CHEMBL3262810) Show SMILES Cc1ccc(cc1)C(=O)N1CCN(CCOc2ccccc2)CC1 Show InChI InChI=1S/C20H24N2O2/c1-17-7-9-18(10-8-17)20(23)22-13-11-21(12-14-22)15-16-24-19-5-3-2-4-6-19/h2-10H,11-16H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.14E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016320 (CHEMBL3262811) Show SMILES Cc1ccc(cc1)C(=O)N1CCN(CCOc2ccc(Cl)cc2)CC1 Show InChI InChI=1S/C20H23ClN2O2/c1-16-2-4-17(5-3-16)20(24)23-12-10-22(11-13-23)14-15-25-19-8-6-18(21)7-9-19/h2-9H,10-15H2,1H3	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.51E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016321 (CHEMBL3262812) Show SMILES Clc1ccccc1C(=O)N1CCN(CCOc2ccccc2)CC1 Show InChI InChI=1S/C19H21ClN2O2/c20-18-9-5-4-8-17(18)19(23)22-12-10-21(11-13-22)14-15-24-16-6-2-1-3-7-16/h1-9H,10-15H2	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	5.68E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016327 (CHEMBL3262813) Show SMILES O=C(CN1CCN(CCOc2ccccc2)CC1)Nc1ccccc1 Show InChI InChI=1S/C20H25N3O2/c24-20(21-18-7-3-1-4-8-18)17-23-13-11-22(12-14-23)15-16-25-19-9-5-2-6-10-19/h1-10H,11-17H2,(H,21,24)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.86E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016328 (CHEMBL3262814) Show SMILES Cc1ccccc1OCCN1CCN(CC(=O)Nc2ccccc2)CC1 Show InChI InChI=1S/C21H27N3O2/c1-18-7-5-6-10-20(18)26-16-15-23-11-13-24(14-12-23)17-21(25)22-19-8-3-2-4-9-19/h2-10H,11-17H2,1H3,(H,22,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.18E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016329 (CHEMBL3262815) Show SMILES FC(F)(F)Oc1ccc(OCCN2CCN(CC(=O)Nc3ccccc3)CC2)cc1 Show InChI InChI=1S/C21H24F3N3O3/c22-21(23,24)30-19-8-6-18(7-9-19)29-15-14-26-10-12-27(13-11-26)16-20(28)25-17-4-2-1-3-5-17/h1-9H,10-16H2,(H,25,28)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.33E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016330 (CHEMBL3262816) Show SMILES Clc1ccc(OCCN2CCN(CC(=O)Nc3ccccc3)CC2)cc1 Show InChI InChI=1S/C20H24ClN3O2/c21-17-6-8-19(9-7-17)26-15-14-23-10-12-24(13-11-23)16-20(25)22-18-4-2-1-3-5-18/h1-9H,10-16H2,(H,22,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.38E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016331 (CHEMBL3262817) Show SMILES O=C(CN1CCN(CCOc2ccc(cc2)C#N)CC1)Nc1ccccc1 Show InChI InChI=1S/C21H24N4O2/c22-16-18-6-8-20(9-7-18)27-15-14-24-10-12-25(13-11-24)17-21(26)23-19-4-2-1-3-5-19/h1-9H,10-15,17H2,(H,23,26)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	9.10E+3	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair
Potassium voltage-gated channel subfamily A member 5 (Homo sapiens (Human))	BDBM50016332 (CHEMBL3262818) Show SMILES COc1ccc(NC(=O)CN2CCN(CCOc3ccccc3)CC2)cc1 Show InChI InChI=1S/C21H27N3O3/c1-26-19-9-7-18(8-10-19)22-21(25)17-24-13-11-23(12-14-24)15-16-27-20-5-3-2-4-6-20/h2-10H,11-17H2,1H3,(H,22,25)	PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.01E+4	n/a	n/a	n/a	n/a	n/a	n/a
China Pharmaceutical University Curated by ChEMBL					Assay Description Inhibition of human Kv1.5 channel expressed in HEK293 cells by whole cell patch clamp assay				Eur J Med Chem 81: 89-94 (2014) Article DOI: 10.1016/j.ejmech.2014.03.075 BindingDB Entry DOI: 10.7270/Q2VX0J3N
					More data for this Ligand-Target Pair

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