Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92971 (Amphiphile, VI) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92969 (Amphiphile, IV) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92976 (Amphiphile, XI) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92978 (Amphiphile, XIII) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92979 (Amphiphile, XVI) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92980 (Amphiphile, XVII) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92974 (Amphiphile, IX) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90E+4 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92977 (Amphiphile, XII) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.64E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92973 (Amphiphile, VIII) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.91E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92972 (Amphiphile, VII) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.46E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92968 (Amphiphile, III) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.58E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92975 (Amphiphile, X) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.08E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM92970 (Amphiphile, V) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.43E+5 | n/a | n/a | n/a | n/a | 7.5 | 30 |
McMaster University | Assay Description The triton X-100 assay previously described by Bell and co-workers were used to measure enzyme activity. | Biochemistry 31: 9025-30 (1992) Article DOI: 10.1021/bi00152a045 BindingDB Entry DOI: 10.7270/Q2W66JCK | |||||||||||
More data for this Ligand-Target Pair |