Affinity Data by PubMed id=16085416

PubMed code 16085416

Found 45 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50050517 (Boronic acid derivative \| CHEMBL305170 \| N-alkyl G...) Show SMILES CC(C)[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	n/a	n/a	0.300	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171653 (CHEMBL196120 \| N-alkyl Gly-boro-Pro derivative) Show SMILES C[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	0.800	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171648 (CHEMBL372180 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171649 (CHEMBL196933 \| N-alkyl Gly-boro-Pro derivative) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.80	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171645 (2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.20	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171650 (2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171656 (2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	4.10	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171647 (CHEMBL373269 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.60	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171653 (CHEMBL196120 \| N-alkyl Gly-boro-Pro derivative) Show SMILES C[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.30	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171649 (CHEMBL196933 \| N-alkyl Gly-boro-Pro derivative) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.80	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171647 (CHEMBL373269 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171657 (2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50050517 (Boronic acid derivative \| CHEMBL305170 \| N-alkyl G...) Show SMILES CC(C)[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171644 (CHEMBL427012 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171651 (2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	15	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171651 (2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171657 (2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	25	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171656 (2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	27	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171650 (2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	27	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171652 (CHEMBL381444 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	35	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50050517 (Boronic acid derivative \| CHEMBL305170 \| N-alkyl G...) Show SMILES CC(C)[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid PDB UniChem Similars	Article PubMed	n/a	n/a	38	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171645 (2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCCCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	58	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171648 (CHEMBL372180 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	61	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171655 (2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	75	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171644 (CHEMBL427012 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	99	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171644 (CHEMBL427012 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	120	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171658 (2-Cyclopropylamino-1-pyrrolidin-1-yl--2-borandihyd...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CC1 Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	130	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171655 (2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	140	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171649 (CHEMBL196933 \| N-alkyl Gly-boro-Pro derivative) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	150	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171657 (2-(Bicyclo[3.2.1]oct-6-ylamino)-1-((S)-2-dihydroxy...) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	180	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171648 (CHEMBL372180 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	270	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171650 (2-Cyclooctonylamino-1-pyrrolidin-1-yl--2-borandihy...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	290	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171647 (CHEMBL373269 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	420	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171645 (2-Cyclodecylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCCCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	530	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171652 (CHEMBL381444 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	560	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171658 (2-Cyclopropylamino-1-pyrrolidin-1-yl--2-borandihyd...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	570	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171656 (2-Cyclohexylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	650	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171652 (CHEMBL381444 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	770	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171646 (CHEMBL196188 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 2 (Homo sapiens (Human))	BDBM50171646 (CHEMBL196188 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.60E+3	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP7 using Ala-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171651 (2-Cyclopentylamino-1-pyrrolidin-1-yl--2-borandihyd...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	Purchase CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	6.50E+3	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171653 (CHEMBL196120 \| N-alkyl Gly-boro-Pro derivative) Show SMILES C[C@@H](N)C(=O)N1CCC[C@H]1B(O)O Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	7.80E+3	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Dipeptidyl peptidase 4 (Homo sapiens (Human))	BDBM50171654 (CHEMBL434184 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	1.60E+4	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human DPP4 using Gly-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171655 (2-Cyclobutylamino-1-pyrrolidin-1-yl--2-borandihydr...) Show SMILES OB(O)[C@@H]1CCCN1C(=O)CNC1CCC1 Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	Article PubMed	n/a	n/a	2.40E+4	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair
Prolyl endopeptidase FAP (Homo sapiens (Human))	BDBM50171646 (CHEMBL196188 \| N-alkyl Gly-boro-Pro derivative) Show SMILES Show InChI	PDB MMDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	3.70E+4	n/a	n/a	n/a	n/a	n/a	n/a
ActivX Biosciences, Inc. Curated by ChEMBL					Assay Description Inhibitory activity against human FAP using Lys-Pro-AMC in fluorometric assay				Bioorg Med Chem Lett 15: 4239-42 (2005) Article DOI: 10.1016/j.bmcl.2005.06.075 BindingDB Entry DOI: 10.7270/Q2CJ8D2F
ActivX Biosciences, Inc. Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%