Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342692 (4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 277 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342693 (2-methyl-6-(1'-(5-methylpyrimidin-2-yl)-4,4'-bipip...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342702 (6-methyl-2-(2-((1S,2R)-2-(1-(5-methylpyrimidin-2-y...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG by patch clamp technique | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342694 (2-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342695 (4-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.06E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342699 (5-chloro-2-(4-((1R,2S)-2-(2-(5-(methylsulfonyl)pyr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG by patch clamp technique | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342700 (2-(4-((1R,2S)-2-(2-(4-(1H-1,2,3-triazol-1-yl)pheno...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG by patch clamp technique | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342703 (CHEMBL1771104 | rac-4-(3-(2-(3-(1-(5-chloropyrimid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | >3.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Potassium voltage-gated channel subfamily H member 2 (Homo sapiens (Human)) | BDBM50342701 (2-(4-((1R,2S)-2-(2-(5-(1H-1,2,3-triazol-1-yl)pyrid...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 4.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Inhibition of human ERG by patch clamp technique | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342679 (CHEMBL1771080 | tert-butyl 1'-(6-cyanopyrimidin-4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342692 (4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342694 (2-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 30 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342674 (CHEMBL1771075 | tert-butyl 1'-(pyridin-2-yl)-4,4'-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2.50E+3 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342683 (1-(4-(methylsulfonyl)phenyl)-1'-(pyrazin-2-yl)-4,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 239 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342684 (1-(4-(methylsulfonyl)phenyl)-1'-(pyrimidin-2-yl)-4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 887 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342685 (1-(5-methylpyrimidin-2-yl)-1'-(4-(methylsulfonyl)p...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 45 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342686 (1-(5-chloropyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 131 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342699 (5-chloro-2-(4-((1R,2S)-2-(2-(5-(methylsulfonyl)pyr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342673 (CHEMBL1771073 | tert-butyl 1'-(4-carbamoylphenyl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 76 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342676 (CHEMBL1771077 | tert-butyl 1'-(pyrimidin-2-yl)-4,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 526 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342680 (CHEMBL1771081 | tert-butyl 1'-(2-cyano-6-methylpyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342683 (1-(4-(methylsulfonyl)phenyl)-1'-(pyrazin-2-yl)-4,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 201 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342689 (6-(1'-(4-(methylsulfonyl)phenyl)-4,4'-bipiperidin-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 62 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342667 (CHEMBL1771067 | tert-butyl 1'-p-tolyl-4,4'-bipiper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342668 (CHEMBL1771068 | tert-butyl 1'-(4-(methylsulfonyl)p...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 36 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342679 (CHEMBL1771080 | tert-butyl 1'-(6-cyanopyrimidin-4-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 31 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342682 (1-(4-(methylsulfonyl)phenyl)-1'-(pyridin-2-yl)-4,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 682 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342688 (1-(5-methylpyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 73 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342703 (CHEMBL1771104 | rac-4-(3-(2-(3-(1-(5-chloropyrimid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342667 (CHEMBL1771067 | tert-butyl 1'-p-tolyl-4,4'-bipiper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 338 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342668 (CHEMBL1771068 | tert-butyl 1'-(4-(methylsulfonyl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 22 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342669 (CHEMBL1771069 | tert-butyl 1'-(3-(methylsulfonyl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.90E+3 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342681 (CHEMBL1771082 | tert-butyl 1'-(6-cyano-2-methylpyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342688 (1-(5-methylpyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 18 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342699 (5-chloro-2-(4-((1R,2S)-2-(2-(5-(methylsulfonyl)pyr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342675 (CHEMBL1771076 | tert-butyl 1'-(pyrimidin-4-yl)-4,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 379 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342677 (CHEMBL1771078 | tert-butyl 1'-(pyrazin-2-yl)-4,4'-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 142 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342687 (1-(5-fluoropyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 206 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342701 (2-(4-((1R,2S)-2-(2-(5-(1H-1,2,3-triazol-1-yl)pyrid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342670 (CHEMBL1771070 | tert-butyl 1'-(4-(methylsulfinyl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342684 (1-(4-(methylsulfonyl)phenyl)-1'-(pyrimidin-2-yl)-4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 98 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342686 (1-(5-chloropyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 48 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342690 (1-(4-(methylsulfonyl)phenyl)-1'-(5-(trifluoromethy...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342680 (CHEMBL1771081 | tert-butyl 1'-(2-cyano-6-methylpyr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342691 (1-(5-chloropyrimidin-2-yl)-1'-(4-(methylsulfonyl)p...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342692 (4-(1'-(5-chloropyrimidin-2-yl)-4,4'-bipiperidin-1-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342664 (CHEMBL1770918 | tert-butyl 1'-(pyridin-3-yl)-4,4'-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 3.60E+3 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342666 (CHEMBL1771066 | tert-butyl 1'-m-tolyl-4,4'-bipiper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 514 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342678 (CHEMBL1771079 | tert-butyl 1'-(2-cyanopyrimidin-4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342682 (1-(4-(methylsulfonyl)phenyl)-1'-(pyridin-2-yl)-4,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 39 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 38 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 14 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342700 (2-(4-((1R,2S)-2-(2-(4-(1H-1,2,3-triazol-1-yl)pheno...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342695 (4-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342689 (6-(1'-(4-(methylsulfonyl)phenyl)-4,4'-bipiperidin-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 41 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342702 (6-methyl-2-(2-((1S,2R)-2-(1-(5-methylpyrimidin-2-y...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342671 (CHEMBL1771071 | tert-butyl 1'-(4-acetylphenyl)-4,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 25 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342672 (CHEMBL1771072 | tert-butyl 1'-(4-(methylthio)pheny...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 600 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342685 (1-(5-methylpyrimidin-2-yl)-1'-(4-(methylsulfonyl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 57 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342687 (1-(5-fluoropyridin-2-yl)-1'-(4-(methylsulfonyl)phe...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 19 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342693 (2-methyl-6-(1'-(5-methylpyrimidin-2-yl)-4,4'-bipip...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 38 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342701 (2-(4-((1R,2S)-2-(2-(5-(1H-1,2,3-triazol-1-yl)pyrid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342702 (6-methyl-2-(2-((1S,2R)-2-(1-(5-methylpyrimidin-2-y...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342671 (CHEMBL1771071 | tert-butyl 1'-(4-acetylphenyl)-4,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 341 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342672 (CHEMBL1771072 | tert-butyl 1'-(4-(methylthio)pheny...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 513 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342673 (CHEMBL1771073 | tert-butyl 1'-(4-carbamoylphenyl)-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 165 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342676 (CHEMBL1771077 | tert-butyl 1'-(pyrimidin-2-yl)-4,4...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 523 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342678 (CHEMBL1771079 | tert-butyl 1'-(2-cyanopyrimidin-4-...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 11 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342681 (CHEMBL1771082 | tert-butyl 1'-(6-cyano-2-methylpyr...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 2 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342690 (1-(4-(methylsulfonyl)phenyl)-1'-(5-(trifluoromethy...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 8 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342693 (2-methyl-6-(1'-(5-methylpyrimidin-2-yl)-4,4'-bipip...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342694 (2-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 82 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342703 (CHEMBL1771104 | rac-4-(3-(2-(3-(1-(5-chloropyrimid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 36 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342665 (CHEMBL1771064 | tert-butyl 1'-phenyl-4,4'-bipiperi...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342674 (CHEMBL1771075 | tert-butyl 1'-(pyridin-2-yl)-4,4'-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 831 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342675 (CHEMBL1771076 | tert-butyl 1'-(pyrimidin-4-yl)-4,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 116 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342677 (CHEMBL1771078 | tert-butyl 1'-(pyrazin-2-yl)-4,4'-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | n/a | n/a | 103 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342691 (1-(5-chloropyrimidin-2-yl)-1'-(4-(methylsulfonyl)p...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 5 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Homo sapiens (Human)) | BDBM50342700 (2-(4-((1R,2S)-2-(2-(4-(1H-1,2,3-triazol-1-yl)pheno...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 4 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at human GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342670 (CHEMBL1771070 | tert-butyl 1'-(4-(methylsulfinyl)p...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 132 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342695 (4-methyl-6-(1'-(5-methylpyrazin-2-yl)-4,4'-bipiper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 64 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342696 ((rac)-cis-4-((2-(1-(5-chloropyrimidin-2-yl)piperid...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 9 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342697 ((+)-trans-4-(2-(2-(1-(5-chloropyrimidin-2-yl)piper...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 0.400 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucose-dependent insulinotropic receptor (Mus musculus) | BDBM50342698 ((rac)-cis-4-((2-((1-(5-chloropyrimidin-2-yl)piperi...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | n/a | n/a | 36 | n/a | n/a | n/a | n/a |
Merck& Co. Curated by ChEMBL | Assay Description Agonist activity at mouse GPR119 expressed in CHO cells co-expressing Galpha15 assessed as increase of intracellular cAMP accumulation after 60 mins ... | Bioorg Med Chem Lett 21: 2665-9 (2011) Article DOI: 10.1016/j.bmcl.2010.12.086 BindingDB Entry DOI: 10.7270/Q2M61KJV | |||||||||||
More data for this Ligand-Target Pair |