Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014005 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014007 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014009 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 505 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014013 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 603 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014012 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 913 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014004 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014011 (4-Ethyl-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dica...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014008 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.05E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014010 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.09E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50014006 (2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 4.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Platelet-activating factor receptor (Cavia porcellus) | BDBM50318494 (3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...) | MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 7.33E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ALTER, S.A. Curated by ChEMBL | Assay Description Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor | J Med Chem 33: 3205-10 (1991) BindingDB Entry DOI: 10.7270/Q2PV6KZ9 | |||||||||||
More data for this Ligand-Target Pair |