Affinity Data by PubMed id=26134550

PubMed code 26134550

Found 9 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Mu-type opioid receptor (Danio rerio)	BDBM50000092 ((-)-(etorphine) \| (-)-morphine \| (1S,5R,13R,14S)-1...) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	Purchase CHEMBL DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars	PDB Article PubMed	187	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair				3D Structure (crystal)
Mu-type opioid receptor (Danio rerio)	BDBM50116156 (CHEMBL3612241) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	8.24E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116158 (CHEMBL3612242) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	9.52E+3	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116163 (CHEMBL3612243) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	1.27E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116155 (CHEMBL3612240) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	3.20E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116081 (CHEMBL3612238) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	3.53E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116153 (CHEMBL3612239) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	3.70E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116169 (CHEMBL3612245) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	7.58E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair
Mu-type opioid receptor (Danio rerio)	BDBM50116168 (CHEMBL3612244) Show SMILES Show InChI	PDB UniProtKB/TrEMBL GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	7.80E+4	n/a	n/a	n/a	n/a	n/a	n/a	n/a	n/a
Universidad de Salamanca Curated by ChEMBL					Assay Description Displacement of [3H]-diprenorphine from zebrafish mu opioid receptor expressed in HEK293 cells after 1 hr by liquid scintillation counting				Eur J Med Chem 101: 150-62 (2015) Article DOI: 10.1016/j.ejmech.2015.06.025 BindingDB Entry DOI: 10.7270/Q2JW8GPB
Universidad de Salamanca Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%