| Reaction Details |
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 | Report a problem with these data |
| Target | Fatty acid-binding protein, heart |
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| Ligand | BDBM50212873 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_455934 (CHEMBL887935) |
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| Ki | 250±n/a nM |
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| Citation |  Sulsky, R; Magnin, DR; Huang, Y; Simpkins, L; Taunk, P; Patel, M; Zhu, Y; Stouch, TR; Bassolino-Klimas, D; Parker, R; Harrity, T; Stoffel, R; Taylor, DS; Lavoie, TB; Kish, K; Jacobson, BL; Sheriff, S; Adam, LP; Ewing, WR; Robl, JA Potent and selective biphenyl azole inhibitors of adipocyte fatty acid binding protein (aFABP). Bioorg Med Chem Lett17:3511-5 (2007) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Fatty acid-binding protein, heart |
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| Name: | Fatty acid-binding protein, heart |
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| Synonyms: | FABP11 | FABP3 | FABPH_HUMAN | Fatty acid binding protein muscle | MDGI |
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| Type: | PROTEIN |
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| Mol. Mass.: | 14858.36 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1463784 |
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| Residue: | 133 |
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| Sequence: | MVDAFLGTWKLVDSKNFDDYMKSLGVGFATRQVASMTKPTTIIEKNGDILTLKTHSTFKN
TEISFKLGVEFDETTADDRKVKSIVTLDGGKLVHLQKWDGQETTLVRELIDGKLILTLTH
GTAVCTRTYEKEA
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| BDBM50212873 |
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| n/a |
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| Name | BDBM50212873 |
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| Synonyms: | ((2'-(5-ETHYL-3,4-DIPHENYL-1H-PYRAZOL-1-YL)-3-BIPHENYLYL)OXY)ACETIC ACID | BMS309403 | CHEMBL247920 | [2'-(5-Ethyl-3,4-diphenyl-pyrazol-1-yl)-biphenyl-3-yloxy]-acetic acid |
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| Type | Small organic molecule |
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| Emp. Form. | C31H26N2O3 |
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| Mol. Mass. | 474.5497 |
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| SMILES | CCc1c(c(nn1-c1ccccc1-c1cccc(OCC(O)=O)c1)-c1ccccc1)-c1ccccc1 |
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| Structure | 
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