The following articles (labelled with PubMed ID or TBD) are for your review
PMID | Data | Article Title | Organization |
1310118 |
32 |
Substituted 4,6-diaminoquinolines as inhibitors of C5a receptor binding. |
Merck Sharp and Dohme Research Laboratories |
25254640 |
64 |
Discovery of 2-[5-(4-Fluorophenylcarbamoyl)pyridin-2-ylsulfanylmethyl]phenylboronic Acid (SX-517): Noncompetitive Boronic Acid Antagonist of CXCR1 and CXCR2. |
Syntrix Biosystems |
19171482 |
22 |
Discovery of small molecule human C5a receptor antagonists. |
Astrazeneca |
18378452 |
64 |
Synthesis and characterization of 5,6,7,8-tetrahydroquinoline C5a receptor antagonists. |
Johnson & Johnson Prd |
11931608 |
17 |
Inhibition of protein-protein association by small molecules: approaches and progress. |
Pfizer |
| 36 |
A nonpeptidic agonist ligand of the human C5a receptor: Synthesis, binding affinity optimization and functional characterization |
TBA |
20527893 |
120 |
Selective hexapeptide agonists and antagonists for human complement C3a receptor. |
The University of Queensland |
20004096 |
49 |
Identification of a new class of small molecule C5a receptor antagonists. |
Wyeth Research |
| 21 |
New non peptidic C5a receptor antagonists |
TBA |
18809326 |
36 |
Small, non-peptide C5a receptor antagonists: part 1. |
Pfizer |
18804369 |
30 |
Small, non-peptide C5a receptor antagonists: part 2. |
Pfizer |
18595693 |
48 |
Design and optimization of aniline-substituted tetrahydroquinoline C5a receptor antagonists. |
Johnson & Johnson Pharmaceutical Research and Development |
16876401 |
48 |
Peptidomimetic C5a receptor antagonists with hydrophobic substitutions at the C-terminus: increased receptor specificity and in vivo activity. |
Jerini |
10354404 |
60 |
Low-molecular-weight peptidic and cyclic antagonists of the receptor for the complement factor C5a. |
University of Queensland |
9719594 |
13 |
Small molecular probes for G-protein-coupled C5a receptors: conformationally constrained antagonists derived from the C terminus of the human plasma protein C5a. |
University of Queensland |
7658455 |
43 |
Decapeptide agonists of human C5a: the relationship between conformation and neutrophil response. |
University of Nebraska Medical Center |
28977749 |
75 |
Chemical Approaches to Modulating Complement-Mediated Diseases. |
The University of Queensland |
2066977 |
8 |
Identification and synthesis of a receptor binding site of human anaphylatoxin C5a. |
Abbott Laboratories |
1732557 |
20 |
Improvements in the minimum binding sequence of C5a: examination of His-67. |
Abbott Laboratories |
1732540 |
10 |
Structure-function studies in a series of carboxyl-terminal octapeptide analogues of anaphylatoxin C5a. |
Abbott Laboratories |
23009604 |
17 |
Synthesis and characterization of 5,7-dihydroxyflavanone derivatives as novel protein tyrosine phosphatase 1B inhibitors. |
Yanbian University College of Pharmacy |