The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28256371 |
83 |
Synthesis of bulky-tailed sulfonamides incorporating pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-1(5H)-yl) moieties and evaluation of their carbonic anhydrases I, II, IV and IX inhibitory effects. |
University of Wollongong |
| 28161252 |
64 |
Synthesis and biological evaluation of cyclic imides incorporating benzenesulfonamide moieties as carbonic anhydrase I, II, IV and IX inhibitors. |
King Saud University |
| 28237553 |
76 |
Human carbonic anhydrase inhibitory profile of mono- and bis-sulfonamides synthesized via a direct sulfochlorination of 3- and 4-(hetero)arylisoxazol-5-amine scaffolds. |
Saint Petersburg State University |
| 28109946 |
84 |
Novel indolin-2-one-based sulfonamides as carbonic anhydrase inhibitors: Synthesis, in vitro biological evaluation against carbonic anhydrases isoforms I, II, IV and VII and molecular docking studies. |
Kafrelsheikh University |
| 28075587 |
102 |
Design and Synthesis of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Treatment of Rheumatoid Arthritis. |
University of Florence |
| 28111158 |
100 |
Synthesis of isoxazole-containing sulfonamides with potent carbonic anhydrase II and VII inhibitory properties. |
Abant Izzet Baysal University |
| 27919611 |
60 |
Discovery of 4-sulfamoyl-phenyl-ß-lactams as a new class of potent carbonic anhydrase isoforms I, II, IV and VII inhibitors: The first example of subnanomolar CA IV inhibitors. |
National Institute of Pharmaceutical Education and Research (NIPER) |
| 27876475 |
68 |
Microwave assisted synthesis of novel tetrazole/sulfonamide derivatives based on octahydroacridine, xanthene and chromene skeletons as inhibitors of the carbonic anhydrases isoforms I, II, IV and VII. |
Dumlupinar University |
| 27144971 |
60 |
PEGylated Bis-Sulfonamide Carbonic Anhydrase Inhibitors Can Efficiently Control the Growth of Several Carbonic Anhydrase IX-Expressing Carcinomas. |
Temple University |
| 27172398 |
20 |
An Unusual Natural Product Primary Sulfonamide: Synthesis, Carbonic Anhydrase Inhibition, and Protein X-ray Structures of Psammaplin C. |
Griffith University |
| 27298005 |
92 |
Microwave assisted synthesis of novel acridine-acetazolamide conjugates and investigation of their inhibition effects on human carbonic anhydrase isoforms hCA I, II, IV and VII. |
Dumlupinar University |
| 26498394 |
105 |
Inhibition of mammalian carbonic anhydrase isoforms I-XIV with a series of phenolic acid esters. |
Universit£ |
| 26498393 |
116 |
New natural product carbonic anhydrase inhibitors incorporating phenol moieties. |
Aristotle University of Thessaloniki |
| 26347950 |
32 |
Phosphate Chemical Probes Designed for Location Specific Inhibition of Intracellular Carbonic Anhydrases. |
Griffith University |
| 25468040 |
77 |
Inhibition studies of new ureido-substituted sulfonamides incorporating a GABA moiety against human carbonic anhydrase isoforms I-XIV. |
TBA |
| 25358084 |
143 |
Discovery and characterization of novel selective inhibitors of carbonic anhydrase IX. |
Vilnius University |
| 24689792 |
54 |
Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes. |
Griffith University |
| 23010455 |
108 |
Synthesis of C-cinnamoyl glycosides and their inhibitory activity against mammalian carbonic anhydrases. |
Universidad Nacional De La Plata |
| 23067387 |
105 |
Tricyclic sulfonamides incorporating benzothiopyrano[4,3-c]pyrazole and pyridothiopyrano[4,3-c]pyrazole effectively inhibita- andß-carbonic anhydrase: X-ray crystallography and solution investigations on 15 isoforms. |
Universit£ |
| 22687439 |
51 |
Synthesis and carbonic anhydrase inhibitory properties of novel bromophenols and their derivatives including natural products: vidalol B. |
Atat£Rk University |
| 22487176 |
109 |
Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins. |
Universit£ |
| 21211980 |
47 |
Characterization and anions inhibition studies of ana-carbonic anhydrase from the teleost fish Dicentrarchus labrax. |
Ondokuz Mayis University |
| 20674354 |
79 |
Carbonic anhydrase inhibitors. Antioxidant polyphenols effectively inhibit mammalian isoforms I-XV. |
Universit£ |
| 20605094 |
91 |
Carbonic anhydrase inhibitors. The X-ray crystal structure of human isoform II in adduct with an adamantyl analogue of acetazolamide resides in a less utilized binding pocket than most hydrophobic inhibitors. |
University of Florida |
| 20472429 |
80 |
Carbonic anhydrase inhibitors: crystallographic and solution binding studies for the interaction of a boron-containing aromatic sulfamide with mammalian isoforms I-XV. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
| 20363633 |
67 |
Thioether benzenesulfonamide inhibitors of carbonic anhydrases II and IV: structure-based drug design, synthesis, and biological evaluation. |
Pfizer |
| 20185318 |
132 |
Carbonic anhydrase inhibitors. Inhibition of mammalian isoforms I-XIV with a series of natural product polyphenols and phenolic acids. |
Universit£ |
| 19911821 |
273 |
Deciphering the mechanism of carbonic anhydrase inhibition with coumarins and thiocoumarins. |
Universita Degli Studi Di Firenze |
| 19854054 |
18 |
Nitric oxide-donating carbonic anhydrase inhibitors for the treatment of open-angle glaucoma. |
Nicox Research Institute |
| 20028100 |
78 |
The coumarin-binding site in carbonic anhydrase accommodates structurally diverse inhibitors: the antiepileptic lacosamide as an example and lead molecule for novel classes of carbonic anhydrase inhibitors. |
Universit£ |
| 19269822 |
75 |
Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I, II, III, VII and XIII with less investigated inorganic anions. |
Universit£ |
| 19186056 |
60 |
A thiabendazole sulfonamide shows potent inhibitory activity against mammalian and nematode alpha-carbonic anhydrases. |
Universit£ |
| 18990571 |
65 |
Carbonic anhydrase inhibitors: 2-substituted-1,3,4-thiadiazole-5-sulfamides act as powerful and selective inhibitors of the mitochondrial isozymes VA and VB over the cytosolic and membrane-associated carbonic anhydrases I, II and IV. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 18359629 |
84 |
Carbonic anhydrase inhibitors: the X-ray crystal structure of ethoxzolamide complexed to human isoform II reveals the importance of thr200 and gln92 for obtaining tight-binding inhibitors. |
Istituto Di Biostrutture E Bioimmagini-Cnr |
| 17475500 |
130 |
Carbonic anhydrases as targets for medicinal chemistry. |
Universit£ |
| 17376683 |
63 |
Carbonic anhydrase inhibitors. Inhibition of isoforms I, II, IV, VA, VII, IX, and XIV with sulfonamides incorporating fructopyranose-thioureido tails. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 17314045 |
11 |
Phosph(on)ate as a zinc-binding group in metalloenzyme inhibitors: X-ray crystal structure of the antiviral drug foscarnet complexed to human carbonic anhydrase I. |
Universit£ |
| 15686931 |
84 |
Carbonic anhydrase inhibitors. Inhibition of the membrane-bound human and bovine isozymes IV with sulfonamides. |
Universit£ |
| 15664814 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V, and IX with anions isosteric and isoelectronic with sulfate, nitrate, and carbonate. |
Universit£ |
| 15501038 |
68 |
Carbonic anhydrase inhibitors: inhibition of the membrane-bound human isozyme IV with anions. |
Universit£ |
| 15357993 |
82 |
Carbonic anhydrase inhibitors. Inhibition of the beta-class enzyme from the methanoarchaeon Methanobacterium thermoautotrophicum (Cab) with anions. |
Universit£ |
| 11229775 |
204 |
Carbonic anhydrase inhibitors: synthesis of sulfonamides incorporating dtpa tails and of their zinc complexes with powerful topical antiglaucoma properties. |
Universit£ |
| 22365761 |
144 |
New chemotypes acting as isozyme-selective carbonic anhydrase inhibitors with low affinity for the offtarget cytosolic isoform II. |
Universit£ |
| 22245047 |
135 |
Structure-activity relationships for the interaction of 5,10-dihydroindeno[1,2-b]indole derivatives with human and bovine carbonic anhydrase isoforms I, II, III, IV and VI. |
Ondokuz Mayis University |
| 22230050 |
82 |
Synthesis and carbonic anhydrase inhibitory properties of novel cyclohexanonyl bromophenol derivatives. |
Artvin£Oruh University |
| 21821413 |
65 |
Synthesis of rhodamine B-benzenesulfonamide conjugates and their inhibitory activity against humana- and bacterial/fungalß-carbonic anhydrases. |
Ecole Nationale Sup£Rieure De Chimie De Montpellier |
| 21515057 |
153 |
Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies. |
Universit£ |
| 21549597 |
71 |
Synthesis and crystallographic analysis of new sulfonamides incorporating NO-donating moieties with potent antiglaucoma action. |
U.O. Oculistica Az. Usl 3 |
| 21377369 |
60 |
Purification and inhibition studies with anions and sulfonamides of ana-carbonic anhydrase from the Antarctic seal Leptonychotes weddellii. |
Universit£ |
| 20590092 |
273 |
Polyamines inhibit carbonic anhydrases by anchoring to the zinc-coordinated water molecule. |
Universita Degli Studi Di Firenze |
| 19527930 |
53 |
The protein tyrosine kinase inhibitors imatinib and nilotinib strongly inhibit several mammalian alpha-carbonic anhydrase isoforms. |
University of Tampere and Tampere University Hospital |
| 19121582 |
15 |
Carbonic anhydrase inhibitors: inhibition studies of a coral secretory isoform with inorganic anions. |
Centre Scientifique De Monaco |
| 16759856 |
9 |
N-hydroxyurea--a versatile zinc binding function in the design of metalloenzyme inhibitors. |
Università |
| 15780631 |
55 |
Carbonic anhydrase inhibitors. Inhibition of isozymes I, II, IV, V and IX with complex fluorides, chlorides and cyanides. |
Università |
| 15745821 |
21 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with organic phosphates and phosphonates. |
University of Montpellier |
| 15664815 |
45 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with carboxylates. |
Università |
| 15501037 |
27 |
Carbonic anhydrase inhibitors. Interaction of isozymes I, II, IV, V, and IX with phosphates, carbamoyl phosphate, and the phosphonate antiviral drug foscarnet. |
Università |
| 32519851 |
164 |
Sulfonamide Inhibitors of Human Carbonic Anhydrases Designed through a Three-Tails Approach: Improving Ligand/Isoform Matching and Selectivity of Action. |
University of Firenze |
| 32435377 |
30 |
Glycomimetic Based Approach toward Selective Carbonic Anhydrase Inhibitors. |
Universit£ |
| 30996772 |
55 |
-Nitrosulfonamides as Carbonic Anhydrase Inhibitors: A Promising Chemotype for Targeting Chagas Disease and Leishmaniasis. |
University of Florence |
| 32364386 |
184 |
Phenyl(thio)phosphon(amid)ate Benzenesulfonamides as Potent and Selective Inhibitors of Human Carbonic Anhydrases II and VII Counteract Allodynia in a Mouse Model of Oxaliplatin-Induced Neuropathy. |
University of Florence |
| 32031797 |
96 |
Discovery of Potent Dual-Tailed Benzenesulfonamide Inhibitors of Human Carbonic Anhydrases Implicated in Glaucoma and in Vivo Profiling of Their Intraocular Pressure-Lowering Action. |
University of Wollongong |
| 31255926 |
46 |
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations. |
University of Sharjah |
| 31794211 |
138 |
"A Sweet Combination": Developing Saccharin and Acesulfame K Structures for Selectively Targeting the Tumor-Associated Carbonic Anhydrases IX and XII. |
University of Florence |
| 31515057 |
20 |
Highly hydrophilic 1,3-oxazol-5-yl benzenesulfonamide inhibitors of carbonic anhydrase II for reduction of glaucoma-related intraocular pressure. |
Saint Petersburg State University |
| 31476557 |
164 |
From random to rational: A discovery approach to selective subnanomolar inhibitors of human carbonic anhydrase IV based on the Castagnoli-Cushman multicomponent reaction. |
Saint Petersburg State University |
| 31401537 |
45 |
Synthesis of novel tellurides bearing benzensulfonamide moiety as carbonic anhydrase inhibitors with antitumor activity. |
University of Florence |
| 31287314 |
52 |
Synthesis and Evaluation of Carbonic Anhydrase Inhibitors with Carbon Monoxide Releasing Properties for the Management of Rheumatoid Arthritis. |
Universit£ |
| 31136893 |
176 |
Benzensulfonamides bearing spyrohydantoin moieties act as potent inhibitors of human carbonic anhydrases II and VII and show neuropathic pain attenuating effects. |
University of Florence |
| 31740053 |
1887 |
Halogenated and di-substituted benzenesulfonamides as selective inhibitors of carbonic anhydrase isoforms. |
Vilnius University |
| 31539777 |
92 |
Continued exploration and tail approach synthesis of benzenesulfonamides containing triazole and dual triazole moieties as carbonic anhydrase I, II, IV and IX inhibitors. |
Kurukshetra University |
| 30553625 |
761 |
Pyrrolidinone-bearing methylated and halogenated benzenesulfonamides as inhibitors of carbonic anhydrases. |
Kaunas University of Technology |
| 31413806 |
65 |
Bis-benzoxaboroles: Design, Synthesis, and Biological Evaluation as Carbonic Anhydrase Inhibitors. |
Universit£ |
| 26678172 |
70 |
Inhibition of carbonic anhydrase isoforms I, II, IV, VII and XII with carboxylates and sulfonamides incorporating phthalimide/phthalic anhydride scaffolds. |
King Saud University |
| 24300919 |
55 |
Combining the tail and the ring approaches for obtaining potent and isoform-selective carbonic anhydrase inhibitors: solution and X-ray crystallographic studies. |
Universit£ |
| 24103430 |
78 |
Inhibition of human carbonic anhydrase isoforms I-XIV with sulfonamides incorporating fluorine and 1,3,5-triazine moieties. |
Universit£ |
| 30496988 |
25 |
Pharmaceutical and medicinal significance of sulfur (S |
Wuhan University of Technology |
| 11831900 |
8 |
Structural aspects of isozyme selectivity in the binding of inhibitors to carbonic anhydrases II and IV. |
University of Pennsylvania |
| 30193219 |
114 |
Discovery of new 2, 5-disubstituted 1,3-selenazoles as selective human carbonic anhydrase IX inhibitors with potent anti-tumor activity. |
Department of University of Florence |
| 30344913 |
24 |
Famotidine, an Antiulcer Agent, Strongly Inhibits |
University of Florence |
| 29685656 |
8 |
Synthesis, structure and bioactivity of primary sulfamate-containing natural products. |
Griffith University |
| 29571155 |
124 |
Synthesis of novel 4-functionalized 1,5-diaryl-1,2,3-triazoles containing benzenesulfonamide moiety as carbonic anhydrase I, II, IV and IX inhibitors. |
Kurukshetra University |
| 28947945 |
72 |
Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors. |
University of Florence |
| 28802125 |
92 |
Novel 4/3-((4-oxo-5-(2-oxoindolin-3-ylidene)thiazolidin-2-ylidene)amino) benzenesulfonamides: Synthesis, carbonic anhydrase inhibitory activity, anticancer activity and molecular modelling studies. |
Kafrelsheikh University |
| 29746127 |
195 |
Discovery of Novel Nonsteroidal Anti-Inflammatory Drugs and Carbonic Anhydrase Inhibitors Hybrids (NSAIDs-CAIs) for the Management of Rheumatoid Arthritis. |
Ege University Bornova |
| 29305297 |
480 |
Benzimidazole design, synthesis, and docking to build selective carbonic anhydrase VA inhibitors. |
Vilnius University |
| 30006175 |
644 |
Design of two-tail compounds with rotationally fixed benzenesulfonamide ring as inhibitors of carbonic anhydrases. |
Vilnius University |
| 29909339 |
84 |
Design and synthesis of novel benzenesulfonamide containing 1,2,3-triazoles as potent human carbonic anhydrase isoforms I, II, IV and IX inhibitors. |
Kurukshetra University |
| 29684705 |
72 |
Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform. |
Egyptian Russian University |
| 29635168 |
140 |
2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering agents. |
University of Florence |
| 29912561 |
40 |
4-Substituted Benzenesulfonamides Incorporating Bi/Tricyclic Moieties Act as Potent and Isoform-Selective Carbonic Anhydrase II/IX Inhibitors. |
Universit£ |
| 29259736 |
70 |
Synthesis of Novel Selenides Bearing Benzenesulfonamide Moieties as Carbonic Anhydrase I, II, IV, VII, and IX Inhibitors. |
University of Florence |
| 29259754 |
76 |
Discovery of New Sulfonamide Carbonic Anhydrase IX Inhibitors Incorporating Nitrogenous Bases. |
University of Florence |
| 29057059 |
82 |
Lucky Switcheroo: Dramatic Potency and Selectivity Improvement of Imidazoline Inhibitors of Human Carbonic Anhydrase VII. |
Saint Petersburg State University |
| 28277280 |
43 |
Bortezomib inhibits mammalian carbonic anhydrases. |
Universit£ |
| 28302505 |
120 |
Evaluation of selenide, diselenide and selenoheterocycle derivatives as carbonic anhydrase I, II, IV, VII and IX inhibitors. |
Universit£ |
| 26773755 |
20 |
Synthesis and tyrosinase inhibition activity of trans-stilbene derivatives. |
Indian Institute of Integrative Medicine |
| 10945872 |
14 |
Pharmacological actions of a novel, high-affinity, and selective human dopamine D(3) receptor antagonist, SB-277011-A. |
Smithkline Beecham Pharmaceuticals |
| 7815325 |
65 |
Cloning and pharmacological characterization of human alpha-1 adrenergic receptors: sequence corrections and direct comparison with other species homologues. |
Duke University |
| 7796807 |
51 |
The 5-HT4 receptor: molecular cloning and pharmacological characterization of two splice variants. |
Synaptic Pharmaceutical |
| 3130534 |
3 |
7-[3-(4-[2,3-Dimethylphenyl]piperazinyl)propoxy]-2(1H)-quinolinone (OPC-4392), a presynaptic dopamine autoreceptor agonist and postsynaptic D2 receptor antagonist. |
Tokushima Research Institute |
| 2664084 |
17 |
Detection of a novel serotonin receptor subtype (5-HT1E) in human brain: interaction with a GTP-binding protein. |
Albany Medical College |
| 2547939 |
11 |
Characterization of the striatal M2 muscarinic receptor mediating inhibition of cyclic AMP using selective antagonists: a comparison with the brainstem M2 receptor. |
Abbott Laboratories |
| 2537406 |
2 |
Pharmacological characterization of the M1 muscarinic receptors expressed in murine fibroblast B82 cells. |
University of Arizona |
| 19900813 |
12 |
Optimization of (4,4-difluoro-1,2,3,4-tetrahydro-5H-1-benzazepine-5-ylidene)acetamide derivatives as arginine vasopressin V2 receptor agonists and discussion of their binding modes. |
Astellas Pharma |
| 18799592 |
17 |
Novel peroxisome proliferator-activated receptor alpha agonists lower low-density lipoprotein and triglycerides, raise high-density lipoprotein, and synergistically increase cholesterol excretion with a liver X receptor agonist. |
Bristol-Myers Squibb |
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