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62 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
27750148 7 Fragment-based discovery of novel pentacyclic triterpenoid derivatives as cholesteryl ester transfer protein inhibitors.EBI China Pharmaceutical University
27490022 29 Design, synthesis and biological evaluation of novel cholesteryl ester transfer protein inhibitors bearing a cycloalkene scaffold.EBI Shenyang Pharmaceutical University
27256912 36 Discovery of hydroxyl 1,2-diphenylethanamine analogs as potent cholesterol ester transfer protein inhibitors.EBI Bristol-Myers Squibb Pharmaceutical Research Institute
26985312 36 Discovery of Novel Indoline Cholesterol Ester Transfer Protein Inhibitors (CETP) through a Structure-Guided Approach.EBI Merck Research Laboratories
27010500 19 Design, synthesis and biological evaluation of N,N-3-phenyl-3-benzylaminopropanamide derivatives as novel cholesteryl ester transfer protein inhibitor.EBI Shenyang Pharmaceutical University
26993745 19 Discovery of novel N,N-3-phenyl-3-benzylaminopropionanilides as potent inhibitors of cholesteryl ester transfer protein in vivo.EBI Shenyang Pharmaceutical University
26200936 39 Applications of Fluorine in Medicinal Chemistry.EBI Bristol-Myers Squibb Research and Development
25127148 1 Some molecular targets for antihyperlipidemic drug research.EBI Banasthali University
25265559 19 Potent cholesteryl ester transfer protein inhibitors of reduced lipophilicity: 1,1'-spiro-substituted hexahydrofuroquinoline derivatives.EBI Boehringer Ingelheim Pharma
24424134 76 Diphenylpyridylethanamine (DPPE)-based aminoheterocycles as cholesteryl ester transfer protein inhibitors.EBI Bristol-Myers Squibb
22650305 64 Diphenylpyridylethanamine (DPPE) derivatives as cholesteryl ester transfer protein (CETP) inhibitors.EBI Bristol-Myers Squibb
22995620 60 Identification of a potent and metabolically stable series of fluorinated diphenylpyridylethanamine-based cholesteryl ester transfer protein inhibitors.EBI Bristol-Myers Squibb
22543028 39 Design and synthesis of new tetrahydroquinolines derivatives as CETP inhibitors.EBI Eli Lilly
22497761 59 Design, synthesis and structure-activity-relationship of 1,5-tetrahydronaphthyridines as CETP inhibitors.EBI Eli Lilly
18374566 129 2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis.EBI Bristol-Myers Squibb Pharmaceutical Research Institute
17521912 15 The biology and chemistry of hyperlipidemia.EBI Sinhgad College of Pharmacy
11000011 28 bis(2-(Acylamino)phenyl) disulfides, 2-(acylamino)benzenethiols, and S-(2-(acylamino)phenyl) alkanethioates as novel inhibitors of cholesteryl ester transfer protein.EBI Research Triangle Institute
 10 CETP inhibitory activity of ceramides, isolated from the gorgonian Acabaria UndulataEBI TBA
 13 Wiedendiol-A and -B, cholesteryl ester transfer protein inhibitors from the marine sponge Xestospongia wiedenmayeriEBI TBA
24900324 8 Discovery of substituted biphenyl oxazolidinone inhibitors of cholesteryl ester transfer protein.EBI TBA
22142541 24 SAR studies on the central phenyl ring of substituted biphenyl oxazolidinone-potent CETP inhibitors.EBI Merck Sharp & Dohme
21682257 11 Biphenyl-substituted oxazolidinones as cholesteryl ester transfer protein inhibitors: modifications of the oxazolidinone ring leading to the discovery of anacetrapib.EBI Merck Research Laboratories
21398121 51 2-(4-Carbonylphenyl)benzoxazole inhibitors of CETP: attenuation of hERG binding and improved HDLc-raising efficacy.EBI Merck Research Laboratories
21147531 44 2-(4-carbonylphenyl)benzoxazole inhibitors of CETP: scaffold design and advancement in HDLc-raising efficacy.EBI Merck Research Laboratories
21094047 69 2-Arylbenzoxazoles as CETP inhibitors: raising HDL-C in cynoCETP transgenic mice.EBI Merck Research Laboratories
21041082 18 Design of a novel class of biphenyl CETP inhibitors.EBI Merck Sharp & Dohme
20667734 18 Synthesis of a series of novel 2,4,5-trisubstituted selenazole compounds as potential PLTP inhibitors.EBI Beijing Institute of Pharmacology and Toxicology
20137927 43 Novel tetrahydrochinoline derived CETP inhibitors.EBI Bayer Healthcare
20036121 49 2-Arylbenzoxazoles as CETP inhibitors: substitution and modification of the alpha-alkoxyamide moiety.EBI Merck Research Laboratories
20089400 27 Synthesis and discovery of 2,3-dihydro-3,8-diphenylbenzo[1,4]oxazines as a novel class of potent cholesteryl ester transfer protein inhibitors.EBI Johnson & Johnson Pharmaceutical Research and Development
 12 Substituted 1,3,5-triazines as cholesteryl ester transfer protein inhibitorsEBI TBA
 8 Phosphonate-containing analogs of cholesteryl ester as novel inhibitors of cholesteryl ester transfer proteinEBI TBA
 14 Novel inhibitors of cholesteryl ester transfer proteinEBI TBA
19339179 24 Design and synthesis of potent inhibitors of cholesteryl ester transfer protein (CETP) exploiting a 1,2,3,4-tetrahydroquinoline platform.EBI Johnson & Johnson Pharmaceutical Research & Development
19236017 8 Design, synthesis, and biological evaluation of (2R,alphaS)-3,4-dihydro-2-[3-(1,1,2,2-tetrafluoroethoxy)phenyl]-5-[3-(trifluoromethoxy)-phenyl]-alpha-(trifluoromethyl)-1(2H)-quinolineethanol as potent and orally active cholesteryl ester transfer protein inhibitor.EBI Johnson and Johnson Pharmaceutical Research and Development
17604633 85 2D Quantitative structure-activity relationship studies on a series of cholesteryl ester transfer protein inhibitors.EBI Universidade Federal Da Bahia
17331716 40 Tetrazole and ester substituted tetrahydoquinoxalines as potent cholesteryl ester transfer protein inhibitors.EBI Array Biopharma
15975789 28 Dibenzodioxocinones--a new class of CETP inhibitors.EBI Bayer Healthcare Pharma Research
15109658 19 S-(2-(acylamino)phenyl) 2,2-dimethylpropanethioates as CETP inhibitors.EBI Central Pharmaceutical Research Institute
12747787 106 Discovery of a simple picomolar inhibitor of cholesteryl ester transfer protein.EBI Pfizer
12190312 67 Chiral N,N-disubstituted trifluoro-3-amino-2-propanols are potent inhibitors of cholesteryl ester transfer protein.EBI Pharmacia
11425523 20 Novel heteroaryl replacements of aromatic 3-tetrafluoroethoxy substituents in trifluoro-3-(tertiaryamino)-2-propanols as potent inhibitors of cholesteryl ester transfer protein.EBI Pharmacia
11101348 22 Discovery of chiral N,N-disubstituted trifluoro-3-amino-2-propanols as potent inhibitors of cholesteryl ester transfer protein.EBI Pfizer
31780304 7 Synthesis, biological evaluation and SAR studies of ursolic acid 3?-ester derivatives as novel CETP inhibitors.EBI Nanjing Medical University
31223447 44 Discovery of a Lead Triphenylethanamine Cholesterol Ester Transfer Protein (CETP) Inhibitor.EBI Bristol-Myers Squibb
9871749 3 A depsipeptide fungal metabolite inhibitor of cholesteryl ester transfer protein.EBI Schering-Plough Research Institute
11405654 1 Combinatorial synthesis of cholesterol ester transfer protein-mRNA ligands and screening by nondenaturating gel-electrophoresis.EBI Johann Wolfgang Goethe-Universit£T Frankfurt/Main
28802120 14 Discovery of pentacyclic triterpene 3?-ester derivatives as a new class of cholesterol ester transfer protein inhibitors.EBI China Pharmaceutical University
29035537 19 Discovery of a Novel Piperidine-Based Inhibitor of Cholesteryl Ester Transfer Protein (CETP) That Retains Activity in Hypertriglyceridemic Plasma.EBI Novartis Institutes For Biomedical Research
23327640 24 Phenolic compounds with pancreatic lipase inhibitory activity from Korean yam (Dioscorea opposita).BDB Seoul National University
15225695 64 4-Acylamino-6-arylfuro[2,3-d]pyrimidines: potent and selective glycogen synthase kinase-3 inhibitors.BDB Tsukuba Research Laboratories