Found 66 hits with Last Name = 'baltgalvis' and Initial = 'ka' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251456
![PNG](/data/jpeg/tenK5025/BindingDB_50251456.png) (CHEMBL4084955)Show InChI InChI=1S/C12H9N3/c1-4-13-5-2-9(1)11-7-15-12-8-14-6-3-10(11)12/h1-8,15H | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251453
![PNG](/data/jpeg/tenK5025/BindingDB_50251453.png) (CHEMBL4079572)Show InChI InChI=1S/C11H9N5/c12-11-14-4-2-9(16-11)8-5-15-10-6-13-3-1-7(8)10/h1-6,15H,(H2,12,14,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251457
![PNG](/data/jpeg/tenK5025/BindingDB_50251457.png) (CHEMBL4105629)Show InChI InChI=1S/C17H17N3/c1-2-13(1)6-10-20-12-16(14-3-7-18-8-4-14)15-5-9-19-11-17(15)20/h3-5,7-9,11-13H,1-2,6,10H2 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251509
![PNG](/data/jpeg/tenK5025/BindingDB_50251509.png) (CHEMBL4064316)Show InChI InChI=1S/C15H15N3/c1-11(2)18-10-14(12-3-6-16-7-4-12)13-5-8-17-9-15(13)18/h3-11H,1-2H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251436
![PNG](/data/jpeg/tenK5025/BindingDB_50251436.png) (CHEMBL4091320)Show InChI InChI=1S/C15H15N3O/c1-19-9-8-18-11-14(12-2-5-16-6-3-12)13-4-7-17-10-15(13)18/h2-7,10-11H,8-9H2,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251451
![PNG](/data/jpeg/tenK5025/BindingDB_50251451.png) (CHEMBL4069163)Show InChI InChI=1S/C19H14FN3/c20-16-3-1-14(2-4-16)12-23-13-18(15-5-8-21-9-6-15)17-7-10-22-11-19(17)23/h1-11,13H,12H2 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50081190
![PNG](/data/jpeg/tenK5008/BindingDB_50081190.png) (CHEMBL3421979)Show InChI InChI=1S/C12H10N4/c1-8-14-5-3-11(16-8)10-6-15-12-7-13-4-2-9(10)12/h2-7,15H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM100152
![PNG](/data/jpeg/tenK10/BindingDB_100152.png) (7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...)Show InChI InChI=1S/C13H12N2O/c1-8-13-11(5-6-14-8)10-4-3-9(16-2)7-12(10)15-13/h3-7,15H,1-2H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
DrugBank MCE KEGG PC cid PC sid PDB UniChem
Similars
| PDB Article PubMed
| n/a | n/a | 41 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | ![3D 3D](/images/Docked_3d.png) 3D Structure (crystal) |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251479
![PNG](/data/jpeg/tenK5025/BindingDB_50251479.png) (CHEMBL4073997)Show InChI InChI=1S/C12H9ClN4/c13-9-3-1-2-7-8(6-16-11(7)9)10-4-5-15-12(14)17-10/h1-6,16H,(H2,14,15,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 46 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251477
![PNG](/data/jpeg/tenK5025/BindingDB_50251477.png) (CHEMBL4075648)Show InChI InChI=1S/C12H8ClN3/c13-11-6-14-3-1-8(11)10-5-16-12-7-15-4-2-9(10)12/h1-7,16H | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251458
![PNG](/data/jpeg/tenK5025/BindingDB_50251458.png) (CHEMBL4087456)Show InChI InChI=1S/C13H9F3N4/c14-13(15,16)7-1-2-8-9(6-19-11(8)5-7)10-3-4-18-12(17)20-10/h1-6,19H,(H2,17,18,20) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 62 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251504
![PNG](/data/jpeg/tenK5025/BindingDB_50251504.png) (CHEMBL4098505)Show InChI InChI=1S/C12H8FN3/c13-12-5-8(1-4-15-12)10-6-16-11-7-14-3-2-9(10)11/h1-7,16H | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251485
![PNG](/data/jpeg/tenK5025/BindingDB_50251485.png) (CHEMBL4080488)Show InChI InChI=1S/C13H11N3/c1-9-6-10(2-5-15-9)12-7-16-13-8-14-4-3-11(12)13/h2-8,16H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50347796
![PNG](/data/jpeg/tenK5034/BindingDB_50347796.png) (CHEMBL1802963)Show InChI InChI=1S/C12H9BrN4/c13-9-3-1-2-7-8(6-16-11(7)9)10-4-5-15-12(14)17-10/h1-6,16H,(H2,14,15,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251452
![PNG](/data/jpeg/tenK5025/BindingDB_50251452.png) (CHEMBL4077010)Show InChI InChI=1S/C13H11N3/c1-16-9-12(10-2-5-14-6-3-10)11-4-7-15-8-13(11)16/h2-9H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 89 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251480
![PNG](/data/jpeg/tenK5025/BindingDB_50251480.png) (CHEMBL4086818)Show InChI InChI=1S/C13H10ClN3/c14-11-3-1-2-9-10(7-17-13(9)11)8-4-5-16-12(15)6-8/h1-7,17H,(H2,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 94 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251476
![PNG](/data/jpeg/tenK5025/BindingDB_50251476.png) (CHEMBL4095674)Show InChI InChI=1S/C19H22N4O/c1(8-22-10-12-24-13-11-22)9-23-15-18(16-2-5-20-6-3-16)17-4-7-21-14-19(17)23/h2-7,14-15H,1,8-13H2 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 109 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251478
![PNG](/data/jpeg/tenK5025/BindingDB_50251478.png) (CHEMBL4072138)Show InChI InChI=1S/C13H9N5/c14-6-8-2-1-3-9-10(7-17-12(8)9)11-4-5-16-13(15)18-11/h1-5,7,17H,(H2,15,16,18) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 138 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251475
![PNG](/data/jpeg/tenK5025/BindingDB_50251475.png) (CHEMBL4090889)Show InChI InChI=1S/C13H12N4O/c1-18-11-4-2-3-8-9(7-16-12(8)11)10-5-6-15-13(14)17-10/h2-7,16H,1H3,(H2,14,15,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 242 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251486
![PNG](/data/jpeg/tenK5025/BindingDB_50251486.png) (CHEMBL4066607)Show InChI InChI=1S/C16H11N3/c1-2-4-15-12(3-1)11(6-8-18-15)14-9-19-16-10-17-7-5-13(14)16/h1-10,19H | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 277 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251507
![PNG](/data/jpeg/tenK5025/BindingDB_50251507.png) (CHEMBL4094549)Show InChI InChI=1S/C13H10N4O2/c14-12-6-8(4-5-15-12)10-7-16-13-9(10)2-1-3-11(13)17(18)19/h1-7,16H,(H2,14,15) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 285 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251510
![PNG](/data/jpeg/tenK5025/BindingDB_50251510.png) (CHEMBL4095156)Show InChI InChI=1S/C13H11N3O/c1-17-13-6-9(2-5-15-13)11-7-16-12-8-14-4-3-10(11)12/h2-8,16H,1H3 | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 351 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251508
![PNG](/data/jpeg/tenK5025/BindingDB_50251508.png) (CHEMBL4065388)Show InChI InChI=1S/C12H9ClN4/c13-7-1-2-8-9(6-16-11(8)5-7)10-3-4-15-12(14)17-10/h1-6,16H,(H2,14,15,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 406 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251506
![PNG](/data/jpeg/tenK5025/BindingDB_50251506.png) (CHEMBL4095479)Show InChI InChI=1S/C13H12N4O/c1-18-8-2-3-9-10(7-16-12(9)6-8)11-4-5-15-13(14)17-11/h2-7,16H,1H3,(H2,14,15,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 443 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM10844
![PNG](/data/jpeg/tenK1/BindingDB_10844.png) (4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)Show InChI InChI=1S/C12H10N4/c13-12-14-6-5-11(16-12)9-7-15-10-4-2-1-3-8(9)10/h1-7,15H,(H2,13,14,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 588 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251509
![PNG](/data/jpeg/tenK5025/BindingDB_50251509.png) (CHEMBL4064316)Show InChI InChI=1S/C15H15N3/c1-11(2)18-10-14(12-3-6-16-7-4-12)13-5-8-17-9-15(13)18/h3-11H,1-2H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
| Article PubMed
| n/a | n/a | 660 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251503
![PNG](/data/jpeg/tenK5025/BindingDB_50251503.png) (CHEMBL4066075)Show InChI InChI=1S/C14H10N4/c15-7-10-2-1-3-11-12(8-18-14(10)11)9-4-5-17-13(16)6-9/h1-6,8,18H,(H2,16,17) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 790 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251451
![PNG](/data/jpeg/tenK5025/BindingDB_50251451.png) (CHEMBL4069163)Show InChI InChI=1S/C19H14FN3/c20-16-3-1-14(2-4-16)12-23-13-18(15-5-8-21-9-6-15)17-7-10-22-11-19(17)23/h1-11,13H,12H2 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.01E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251457
![PNG](/data/jpeg/tenK5025/BindingDB_50251457.png) (CHEMBL4105629)Show InChI InChI=1S/C17H17N3/c1-2-13(1)6-10-20-12-16(14-3-7-18-8-4-14)15-5-9-19-11-17(15)20/h3-5,7-9,11-13H,1-2,6,10H2 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251484
![PNG](/data/jpeg/tenK5025/BindingDB_50251484.png) (CHEMBL4074685)Show InChI InChI=1S/C12H10N4/c13-12-5-8(1-4-15-12)10-6-16-11-7-14-3-2-9(10)11/h1-7,16H,(H2,13,15) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.02E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251505
![PNG](/data/jpeg/tenK5025/BindingDB_50251505.png) (CHEMBL4068096)Show InChI InChI=1S/C14H13N3O/c1-18-12-4-2-3-10-11(8-17-14(10)12)9-5-6-16-13(15)7-9/h2-8,17H,1H3,(H2,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.14E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251482
![PNG](/data/jpeg/tenK5025/BindingDB_50251482.png) (CHEMBL4098364)Show InChI InChI=1S/C14H13N3O/c1-18-10-2-3-11-12(8-17-13(11)7-10)9-4-5-16-14(15)6-9/h2-8,17H,1H3,(H2,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251481
![PNG](/data/jpeg/tenK5025/BindingDB_50251481.png) (CHEMBL4069088)Show InChI InChI=1S/C13H10ClN3/c14-9-1-2-10-11(7-17-12(10)6-9)8-3-4-16-13(15)5-8/h1-7,17H,(H2,15,16) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 2.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251436
![PNG](/data/jpeg/tenK5025/BindingDB_50251436.png) (CHEMBL4091320)Show InChI InChI=1S/C15H15N3O/c1-19-9-8-18-11-14(12-2-5-16-6-3-12)13-4-7-17-10-15(13)18/h2-7,10-11H,8-9H2,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251502
![PNG](/data/jpeg/tenK5025/BindingDB_50251502.png) (CHEMBL4103831)Show InChI InChI=1S/C14H10F3N3/c15-14(16,17)9-1-2-10-11(7-20-12(10)6-9)8-3-4-19-13(18)5-8/h1-7,20H,(H2,18,19) | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251452
![PNG](/data/jpeg/tenK5025/BindingDB_50251452.png) (CHEMBL4077010)Show InChI InChI=1S/C13H11N3/c1-16-9-12(10-2-5-14-6-3-10)11-4-7-15-8-13(11)16/h2-9H,1H3 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 4.78E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251478
![PNG](/data/jpeg/tenK5025/BindingDB_50251478.png) (CHEMBL4072138)Show InChI InChI=1S/C13H9N5/c14-6-8-2-1-3-9-10(7-17-12(8)9)11-4-5-16-13(15)18-11/h1-5,7,17H,(H2,15,16,18) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 5.16E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251476
![PNG](/data/jpeg/tenK5025/BindingDB_50251476.png) (CHEMBL4095674)Show InChI InChI=1S/C19H22N4O/c1(8-22-10-12-24-13-11-22)9-23-15-18(16-2-5-20-6-3-16)17-4-7-21-14-19(17)23/h2-7,14-15H,1,8-13H2 | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 7.58E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human)) | BDBM50251483
![PNG](/data/jpeg/tenK5025/BindingDB_50251483.png) (CHEMBL4102903)Show InChI InChI=1S/C12H9N3/c1-2-9(6-13-4-1)11-7-15-12-8-14-5-3-10(11)12/h1-8,15H | PDB MMDB
Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human GST-tagged Dyrk1a expressed in baculovirus expression system using Alexa-Fluor tracer-236 incubated for 6... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251506
![PNG](/data/jpeg/tenK5025/BindingDB_50251506.png) (CHEMBL4095479)Show InChI InChI=1S/C13H12N4O/c1-18-8-2-3-9-10(7-16-12(9)6-8)11-4-5-15-13(14)17-11/h2-7,16H,1H3,(H2,14,15,17) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 7.96E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251456
![PNG](/data/jpeg/tenK5025/BindingDB_50251456.png) (CHEMBL4084955)Show InChI InChI=1S/C12H9N3/c1-4-13-5-2-9(1)11-7-15-12-8-14-6-3-10(11)12/h1-8,15H | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 9.23E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251477
![PNG](/data/jpeg/tenK5025/BindingDB_50251477.png) (CHEMBL4075648)Show InChI InChI=1S/C12H8ClN3/c13-11-6-14-3-1-8(11)10-5-16-12-7-15-4-2-9(10)12/h1-7,16H | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 9.61E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50347806
![PNG](/data/jpeg/tenK5034/BindingDB_50347806.png) (CHEMBL1802401)Show InChI InChI=1S/C12H9N5O2/c13-12-14-5-4-9(16-12)8-6-15-11-7(8)2-1-3-10(11)17(18)19/h1-6,15H,(H2,13,14,16) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| CHEMBL PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 9.95E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251508
![PNG](/data/jpeg/tenK5025/BindingDB_50251508.png) (CHEMBL4065388)Show InChI InChI=1S/C12H9ClN4/c13-7-1-2-8-9(6-16-11(8)5-7)10-3-4-15-12(14)17-10/h1-6,16H,(H2,14,15,17) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251453
![PNG](/data/jpeg/tenK5025/BindingDB_50251453.png) (CHEMBL4079572)Show InChI InChI=1S/C11H9N5/c12-11-14-4-2-9(16-11)8-5-15-10-6-13-3-1-7(8)10/h1-6,15H,(H2,12,14,16) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.23E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251482
![PNG](/data/jpeg/tenK5025/BindingDB_50251482.png) (CHEMBL4098364)Show InChI InChI=1S/C14H13N3O/c1-18-10-2-3-11-12(8-17-13(11)7-10)9-4-5-16-14(15)6-9/h2-8,17H,1H3,(H2,15,16) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251503
![PNG](/data/jpeg/tenK5025/BindingDB_50251503.png) (CHEMBL4066075)Show InChI InChI=1S/C14H10N4/c15-7-10-2-1-3-11-12(8-18-14(10)11)9-4-5-17-13(16)6-9/h1-6,8,18H,(H2,16,17) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.39E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM10844
![PNG](/data/jpeg/tenK1/BindingDB_10844.png) (4-(1H-indol-3-yl)pyrimidin-2-amine | Meridianin G)Show InChI InChI=1S/C12H10N4/c13-12-14-6-5-11(16-12)9-7-15-10-4-2-1-3-8(9)10/h1-7,15H,(H2,13,14,16) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| Purchase
MCE PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1.48E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251458
![PNG](/data/jpeg/tenK5025/BindingDB_50251458.png) (CHEMBL4087456)Show InChI InChI=1S/C13H9F3N4/c14-13(15,16)7-1-2-8-9(6-19-11(8)5-7)10-3-4-18-12(17)20-10/h1-6,19H,(H2,17,18,20) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Similars
| Article PubMed
| n/a | n/a | 1.53E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |
Glycogen synthase kinase-3 beta
(Homo sapiens (Human)) | BDBM50251475
![PNG](/data/jpeg/tenK5025/BindingDB_50251475.png) (CHEMBL4090889)Show InChI InChI=1S/C13H12N4O/c1-18-11-4-2-3-8-9(7-16-12(8)11)10-5-6-15-13(14)17-10/h2-7,16H,1H3,(H2,14,15,17) | PDB MMDB
NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![](/images/AffyNet_logo.png)
| PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| n/a | n/a | 1.58E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rigel Pharmaceuticals, Inc.
Curated by ChEMBL
| Assay Description Inhibition of full-length recombinant human His-tagged GSK3B recombinant in baculovirus expression system using Alexa-Fluor tracer-236 incubated for ... |
Bioorg Med Chem Lett 27: 2617-2621 (2017)
Article DOI: 10.1016/j.bmcl.2017.03.037 BindingDB Entry DOI: 10.7270/Q2SN0CFP |
More data for this Ligand-Target Pair | |