Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053109 (CHEMBL331755 | [1-Aminooxalyl-3-(2-benzyl-benzyl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053136 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosolic phospholipase A2 (Homo sapiens (Human)) | BDBM50085993 ((E)-N-(((2S,4R)-4-((biphenyl-2-ylmethyl)(isobutyl)...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay) | J Med Chem 43: 1041-4 (2000) BindingDB Entry DOI: 10.7270/Q27P8XMZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosolic phospholipase A2 (Homo sapiens (Human)) | BDBM50085984 (CHEMBL9161 | N-[1-[2-(2,4-Difluoro-benzoyl)-benzoy...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay) | J Med Chem 43: 1041-4 (2000) BindingDB Entry DOI: 10.7270/Q27P8XMZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053106 (CHEMBL120112 | [1-Aminooxalyl-2-ethyl-3-(3-trifluo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053108 ((1-Aminooxalyl-3-benzyl-2-methyl-indolizin-8-yloxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053137 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053102 (CHEMBL121245 | [1-Aminooxalyl-3-(3-chloro-benzyl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosolic phospholipase A2 (Homo sapiens (Human)) | BDBM50085986 (CHEMBL267258 | N-{4-(Biphenyl-2-ylmethyl-isobutyl-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay) | J Med Chem 43: 1041-4 (2000) BindingDB Entry DOI: 10.7270/Q27P8XMZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053114 ((1-Aminooxalyl-3-biphenyl-3-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053133 ((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053096 (CHEMBL123774 | [1-Aminooxalyl-3-(4-butyl-benzyl)-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053123 ((1-Aminooxalyl-2-ethyl-3-naphthalen-1-ylmethyl-ind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosolic phospholipase A2 (Homo sapiens (Human)) | BDBM50085987 (4-(2,4-Dioxo-thiazolidin-5-ylidenemethyl)-N-[1-[2-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay) | J Med Chem 43: 1041-4 (2000) BindingDB Entry DOI: 10.7270/Q27P8XMZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053137 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053102 (CHEMBL121245 | [1-Aminooxalyl-3-(3-chloro-benzyl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053109 (CHEMBL331755 | [1-Aminooxalyl-3-(2-benzyl-benzyl)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053147 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-cyclopropyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytosolic phospholipase A2 (Homo sapiens (Human)) | BDBM50085994 (CHEMBL8970 | N-{4-(Biphenyl-2-ylmethyl-isobutyl-am...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description Inhibition of Human cPLA2 alpha using Enzyme assay(PC/DOG assay) | J Med Chem 43: 1041-4 (2000) BindingDB Entry DOI: 10.7270/Q27P8XMZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053095 ((1-Aminooxalyl-2-ethyl-3-naphthalen-2-ylmethyl-ind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053108 ((1-Aminooxalyl-3-benzyl-2-methyl-indolizin-8-yloxy...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053136 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053133 ((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053147 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-cyclopropyl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053106 (CHEMBL120112 | [1-Aminooxalyl-2-ethyl-3-(3-trifluo...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053114 ((1-Aminooxalyl-3-biphenyl-3-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053140 ((1-Aminooxalyl-3-[2,2']bithiophenyl-4-ylmethyl-2-e...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053116 ((1-Aminooxalyl-3-cyclohexylmethyl-2-methyl-indoliz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053096 (CHEMBL123774 | [1-Aminooxalyl-3-(4-butyl-benzyl)-2...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053112 ((1-Aminooxalyl-2-ethyl-3-thiophen-2-ylmethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053140 ((1-Aminooxalyl-3-[2,2']bithiophenyl-4-ylmethyl-2-e...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053104 ((3-Benzyl-1-carbamoylmethyl-2-ethyl-indolizin-8-yl...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053112 ((1-Aminooxalyl-2-ethyl-3-thiophen-2-ylmethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053139 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methoxy-ind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053113 ((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-cyclopr...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053155 ((1-Aminooxalyl-3-biphenyl-4-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 13 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053125 ((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-ethyl-i...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053141 ((1-Aminooxalyl-3-cyclopentylmethyl-2-methyl-indoli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053125 ((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-ethyl-i...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 14 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053139 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methoxy-ind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053116 ((1-Aminooxalyl-3-cyclohexylmethyl-2-methyl-indoliz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053154 (CHEMBL121199 | [1-Carbamoylmethyl-3-(3-chloro-benz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053110 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methylsulfa...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053095 ((1-Aminooxalyl-2-ethyl-3-naphthalen-2-ylmethyl-ind...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053120 ((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053143 (CHEMBL123394 | [1-Aminooxalyl-2-ethyl-3-(2-methyl-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 17 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053155 ((1-Aminooxalyl-3-biphenyl-4-ylmethyl-2-ethyl-indol...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 18 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053132 ((1-Aminooxalyl-3-cyclopentylmethyl-2-ethyl-indoliz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay. | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053132 ((1-Aminooxalyl-3-cyclopentylmethyl-2-ethyl-indoliz...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phospholipase A2 (Homo sapiens (Human)) | BDBM50053146 (CHEMBL331184 | [1-Aminooxalyl-2-ethyl-3-((S)-3-pen...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Co., Ltd Curated by ChEMBL | Assay Description Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC). | J Med Chem 39: 3636-58 (1996) Article DOI: 10.1021/jm960395q BindingDB Entry DOI: 10.7270/Q2NC609M | |||||||||||
More data for this Ligand-Target Pair |
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