Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203869 (7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 0.900 | -51.5 | 3.40 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203875 (7-(3-((4-Borono-3-formylphenoxy)methyl)-1,5-dimeth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.20 | -50.7 | 4.20 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203870 (7-(3-((3-Acetyl-4-boronophenoxy)methyl)-1,5-dimeth...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.20 | -50.7 | 4.70 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91624 (alpha7 agonists 4t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.30 | -49.9 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203876 (Mcl-1 inhibitor 12) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.60 | -50.0 | 5.96 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91603 (4' | alpha7 agonists 4') | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2 | -48.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91615 (15q | alpha7 agonists 15q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4 | -47.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91615 (15q | alpha7 agonists 15q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 8 | -45.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91615 (15q | alpha7 agonists 15q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 13 | -44.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91615 (15q | alpha7 agonists 15q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 13 | -44.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203871 (7-(3-((3-formylphenoxy)methyl)-1,5-dimethyl-1H-pyr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 16 | -44.3 | 59.5 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91624 (alpha7 agonists 4t) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 16 | -43.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91621 (21q | alpha7 agonists 21q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 18 | -43.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91613 (13q | alpha7 agonists 13q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 20 | -43.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91601 (3' | alpha7 agonists 3') | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 24 | -42.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91629 (14t | alpha7 agonists 14t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 25 | -42.7 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91628 (13t | alpha7 agonists 13t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 26 | -42.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91621 (21q | alpha7 agonists 21q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 30 | -42.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91633 (18t | alpha7 agonists 18t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 30 | -42.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91599 (2' | alpha7 agonists 2') | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 40 | -41.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91621 (21q | alpha7 agonists 21q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 40 | -41.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91630 (15t | alpha7 agonists 15t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 40 | -41.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203873 (7-(3-((4-Boronophenoxy)methyl)-1,5-dimethyl-1H-pyr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 44 | -41.8 | 162 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91620 (20q | alpha7 agonists 20q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 50 | -41.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91614 (14q | alpha7 agonists 14q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 50 | -41.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91611 (11q | alpha7 agonists 11q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 50 | -41.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91619 (19q | alpha7 agonists 19q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 60 | -40.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91707 (alpha7 agonists 1') | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 60 | -40.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203872 (7-(3-((3-Acetylphenoxy)methyl)-1,5-dimethyl-1H-pyr...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 64 | -40.9 | 237 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91618 (18q | alpha7 agonists 18q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 70 | -40.2 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91613 (13q | alpha7 agonists 13q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 80 | -39.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91614 (14q | alpha7 agonists 14q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 96 | -39.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91603 (4' | alpha7 agonists 4') | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 100 | -39.3 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Induced myeloid leukemia cell differentiation protein Mcl-1 [171-327] (Homo sapiens (Human)) | BDBM203874 (Mcl-1 inhibitor 10) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 104 | -39.7 | 383 | n/a | n/a | n/a | n/a | 7.4 | 24 |
Oncology Innovative Medicines Unit | Assay Description TR-FRET assay was used to assess the ability of compounds to disrupt the interaction between recombinant human Mcl-1 and a labeled BIM peptide probe.... | Nat Chem Biol 12: 931-936 (2016) Article DOI: 10.1038/nchembio.2174 BindingDB Entry DOI: 10.7270/Q2FN1513 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91624 (alpha7 agonists 4t) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 109 | -39.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91630 (15t | alpha7 agonists 15t) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 110 | -39.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91613 (13q | alpha7 agonists 13q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 110 | -39.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91617 (17q | alpha7 agonists 17q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 110 | -39.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91619 (19q | alpha7 agonists 19q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 120 | -38.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91613 (13q | alpha7 agonists 13q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 120 | -38.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91620 (20q | alpha7 agonists 20q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 120 | -38.8 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91617 (17q | alpha7 agonists 17q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 130 | -38.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91614 (14q | alpha7 agonists 14q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 140 | -38.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91630 (15t | alpha7 agonists 15t) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 140 | -38.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91637 (22t | alpha7 agonists 22t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 141 | -38.4 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91622 (22q | alpha7 agonists 22q) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 160 | -38.1 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91707 (alpha7 agonists 1') | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 170 | -38.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91614 (14q | alpha7 agonists 14q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 170 | -38.0 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Soluble acetylcholine receptor (Aplysia Californica) | BDBM91622 (22q | alpha7 agonists 22q) | PDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 200 | -37.6 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Acetylcholine-binding protein (Lymnaea stagnalis) | BDBM91627 (12t | alpha7 agonists 12t) | PDB UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 210 | -37.5 | n/a | n/a | n/a | n/a | n/a | 7.4 | 20 |
University of California, San Diego | Assay Description Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ?l of 0.2 mg/ml an... | Taylor Research Group (2014) Article DOI: 10.1124/mol.112.080291 BindingDB Entry DOI: 10.7270/Q2805163 | |||||||||||
More data for this Ligand-Target Pair |
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