Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50292299 ((5S)-3-(3-fluoro-4-(3-methylisoxazol-5-yl)phenyl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Boston Curated by ChEMBL | Assay Description Inhibition human liver MAOA activity | Bioorg Med Chem Lett 17: 337-40 (2007) Article DOI: 10.1016/j.bmcl.2006.10.063 BindingDB Entry DOI: 10.7270/Q2HH6JQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159379 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26106 (CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | 540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26114 (CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents | PubMed | 800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Inhibitory activity against prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50292302 (CHEMBL390465 | N-(((S)-3-(3-fluoro-4-(3-methylisox...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Boston Curated by ChEMBL | Assay Description Inhibition human liver MAOA activity | Bioorg Med Chem Lett 17: 337-40 (2007) Article DOI: 10.1016/j.bmcl.2006.10.063 BindingDB Entry DOI: 10.7270/Q2HH6JQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159388 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50292301 ((5R)-5-((1H-1,2,3-triazol-1-yl)methyl)-3-(3-fluoro...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Boston Curated by ChEMBL | Assay Description Inhibition human liver MAOA activity | Bioorg Med Chem Lett 17: 337-40 (2007) Article DOI: 10.1016/j.bmcl.2006.10.063 BindingDB Entry DOI: 10.7270/Q2HH6JQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159382 ((R)-5-(4-Chloro-[1,2,3]triazol-1-ylmethyl)-3-[4-(1...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159372 (1-{(R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159385 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159370 (1-{(R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159380 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159375 (CHEMBL179191 | N-{(S)-3-[4-(1,1-Dioxo-1,2,3,6-tetr...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 5.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159378 ((R)-5-(4-Bromo-[1,2,3]triazol-1-ylmethyl)-3-[4-(1,...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50116067 ((Linezolid)N-[3-(3-Fluoro-4-morpholin-4-yl-phenyl)...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Boston Curated by ChEMBL | Assay Description Inhibition human liver MAOA activity | Bioorg Med Chem Lett 17: 337-40 (2007) Article DOI: 10.1016/j.bmcl.2006.10.063 BindingDB Entry DOI: 10.7270/Q2HH6JQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50292300 ((5R)-3-(3-fluoro-4-(3-methylisoxazol-5-yl)phenyl)-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca R&D Boston Curated by ChEMBL | Assay Description Inhibition human liver MAOA activity | Bioorg Med Chem Lett 17: 337-40 (2007) Article DOI: 10.1016/j.bmcl.2006.10.063 BindingDB Entry DOI: 10.7270/Q2HH6JQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159386 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 2.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159374 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159371 (CHEMBL360090 | Phosphoric acid 1-{(R)-3-[4-(1,1-di...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159373 ((R)-5-[4-(2,2-Dibromo-vinyl)-[1,2,3]triazol-1-ylme...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159377 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 1.02E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159376 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159387 ((1-{(R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159384 ((R)-5-[4-((E)-2-Bromo-vinyl)-[1,2,3]triazol-1-ylme...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159383 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] A (Homo sapiens (Human)) | BDBM50159381 ((R)-3-[4-(1,1-Dioxo-1,2,3,6-tetrahydro-1lambda*6*-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
AstraZeneca Discovery Curated by ChEMBL | Assay Description Binding affinity for human liver monoamine oxidase A | J Med Chem 48: 499-506 (2005) Article DOI: 10.1021/jm0400810 BindingDB Entry DOI: 10.7270/Q2VH5NBS | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042876 (CHEMBL332005 | [2,2']Bipyridinyl-5,5'-dicarboxylic...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 185 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042876 (CHEMBL332005 | [2,2']Bipyridinyl-5,5'-dicarboxylic...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 190 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042873 (5'-(4-Ethoxy-phenylcarbamoyl)-[2,2']bipyridinyl-5-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 320 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26106 (CHEMBL90852 | N-oxalyl glycine, 1a | NOG | Oxalylg...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 2.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042872 (3-phenylsulfonamidocarbonyl-6-(5-phenylsulfonamido...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM26114 (CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents | PubMed | n/a | n/a | 5.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM26114 (CHEMBL88972 | pyridine carboxylate, 6b | pyridine-...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents | PubMed | n/a | n/a | 5.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042875 (CHEMBL125345 | Potassium; [2,2']bipyridinyl-5-carb...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.32E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042877 (CHEMBL420149 | N-([2,2']Bipyridinyl-5-carbonyl)-be...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.38E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50042874 (2,2'-Bipyridin | 2,2'-bipyridine | 2,2'-bipyridyl ...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 3.42E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000866 (2-(Oxalyl-amino)-propionic acid (0.25H2O) | CHEMBL...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 3.82E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000865 (2-(Oxalyl-amino)-propionic acid | CHEMBL314979) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 9.07E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transmembrane prolyl 4-hydroxylase (Homo sapiens (Human)) | BDBM50000407 (2-carboxypyridine | CHEMBL72628 | alpha-picolinic ...) | PDB KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 1.12E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Zeneca Pharmaceuticals Curated by ChEMBL | Assay Description Inhibition of prolyl 4-hydroxylase by chromatographic determination of [14C]-succinic acid on ion-exchange minicolumna | J Med Chem 36: 3853-8 (1994) BindingDB Entry DOI: 10.7270/Q2RJ4HJV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000864 (CHEMBL314175 | N-(2-Methanesulfonylamino-2-oxo-eth...) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.14E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prolyl 4-hydroxylase subunit alpha-1 (Rattus norvegicus) | BDBM50000863 (2-(Oxalyl-amino)-propionic acid | CHEMBL88472) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 6.21E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
ICI Pharmaceuticals Curated by ChEMBL | Assay Description Compound was evaluated for the inhibition of prolyl 4-hydroxylase at 50 ug/mL | J Med Chem 35: 2652-8 (1992) BindingDB Entry DOI: 10.7270/Q28P5ZF9 | |||||||||||
More data for this Ligand-Target Pair |