Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM175970 (US10047103, 3 | US9605024, Example 3 | US9688695, ...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.00400 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of activating peptide-induced receptor activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM175970 (US10047103, 3 | US9605024, Example 3 | US9688695, ...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 0.0230 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of gamma-thrombin-induced receptor activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199438 (CHEMBL3931873) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of activating peptide-induced receptor activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199421 (CHEMBL3906197) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199421 (CHEMBL3906197) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199421 (CHEMBL3906197) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199420 (CHEMBL3933579) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199420 (CHEMBL3933579) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199420 (CHEMBL3933579) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 20 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199420 (CHEMBL3933579) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 21 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199416 (CHEMBL3936444) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced P-selectin activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199416 (CHEMBL3936444) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199416 (CHEMBL3936444) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199440 (CHEMBL3909608) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199440 (CHEMBL3909608) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 29 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199425 (CHEMBL3950308) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199425 (CHEMBL3950308) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 36 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199423 (CHEMBL3983476) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199423 (CHEMBL3983476) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 40 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199431 (CHEMBL3927486) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199431 (CHEMBL3927486) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 52 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199442 (CHEMBL3922644) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199442 (CHEMBL3922644) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 58 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199438 (CHEMBL3931873) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 59 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 (unknown origin) assessed as inhibition of gamma-thrombin-induced receptor activation | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024253 (CHEMBL3334887) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets after 10 mins by flow cytometric analysis | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024253 (CHEMBL3334887) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199433 (CHEMBL3902806) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199433 (CHEMBL3902806) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 69 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199428 (CHEMBL3890362) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 72 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199428 (CHEMBL3890362) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 73 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199418 (CHEMBL3973767) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199418 (CHEMBL3973767) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 83 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2D6 (Homo sapiens (Human)) | BDBM50536645 (CHEMBL4528799) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <100 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Inhibition of CYP2D6 in human liver microsomes incubated for 15 mins using dextromethorphan substrate in presence of NADPH by LC-MS/MS method | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cytochrome P450 2D6 (Homo sapiens (Human)) | BDBM50536646 (CHEMBL4557930) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 120 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Inhibition of CYP2D6 in human liver microsomes incubated for 15 mins using dextromethorphan substrate in presence of NADPH by LC-MS/MS method | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024254 (CHEMBL125021) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity PAR4 (unknown origin) | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024254 (CHEMBL125021) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50536642 (CHEMBL4566669) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 132 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity against PAR4 activating peptide domain in in human platelets assessed as inhibition of P-selectin activation | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024252 (CHEMBL1609104) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199437 (CHEMBL3912611) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 174 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199437 (CHEMBL3912611) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 175 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50536642 (CHEMBL4566669) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 178 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding... | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50536642 (CHEMBL4566669) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 180 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding... | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50536657 (CHEMBL4586027) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 204 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding... | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199427 (CHEMBL3937549) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 207 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199427 (CHEMBL3937549) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 209 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of activating peptide-induced PAC1 binding response preincubated for 20 mins fo... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50536657 (CHEMBL4586027) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 210 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture & Forestry University Curated by ChEMBL | Assay Description Antagonist activity against PAR4 activating peptide domain in human platelets assessed as inhibition of alpha2bbeta3 activation level by PAC1 binding... | J Med Chem 59: 7690-5 (2016) Article DOI: 10.1021/acs.jmedchem.6b00928 BindingDB Entry DOI: 10.7270/Q29C71XC | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199416 (CHEMBL3936444) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 229 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostaglandin G/H synthase 2 (Homo sapiens (Human)) | BDBM11639 (4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA | Assay Description Inhibition of COX-2 (unknown origin) assessed as reduction in PGH2 formation using arachidonic acid as substrate preincubated for 5 mins followed by ... | Citation and Details Article DOI: 10.1016/j.bmcl.2020.127743 BindingDB Entry DOI: 10.7270/Q23B63RC | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50199416 (CHEMBL3936444) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 246 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in human platelets assessed as inhibition of gamma-thrombin-induced PAC1 binding response preincubated for 20 mins follow... | Bioorg Med Chem Lett 26: 5481-5486 (2016) Article DOI: 10.1016/j.bmcl.2016.10.020 BindingDB Entry DOI: 10.7270/Q2P55QGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024255 (CHEMBL3334944) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 279 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair |
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