Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078977 (1-(3-{3-[N'-(4-Hydroxy-phenyl)-guanidino]-2-oxo-2,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Homo sapiens (Human)) | BDBM18656 ((2R,5S)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Astellas Pharma Inc. | Assay Description The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a... | J Med Chem 49: 716-26 (2006) Article DOI: 10.1021/jm050293c BindingDB Entry DOI: 10.7270/Q2P84952 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078965 (1-Benzothiazol-6-yl-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM18656 ((2R,5S)-4-[4-cyano-3-(trifluoromethyl)phenyl]-2,5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 6.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Astellas Pharma Inc. | Assay Description The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a... | J Med Chem 49: 716-26 (2006) Article DOI: 10.1021/jm050293c BindingDB Entry DOI: 10.7270/Q2P84952 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079009 (1-(3-{3-[N'-(4-Hydroxy-phenyl)-N''-methyl-guanidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078970 (1-(2-Fluoro-phenyl)-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079016 (1-Benzofuran-6-yl-3-{1-[3-(3-isopropyl-ureido)-ben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079015 (1-(2,4-Difluoro-phenyl)-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079012 (1-Benzo[b]thiophen-6-yl-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078958 (CHEMBL433216 | {3-[2-Oxo-3-(3-phenyl-ureido)-2,3,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078966 (1-Benzo[b]thiophen-5-yl-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Rattus norvegicus (Rat)) | BDBM18525 (Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | PDB Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Astellas Pharma Inc. | Assay Description The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a... | J Med Chem 49: 716-26 (2006) Article DOI: 10.1021/jm050293c BindingDB Entry DOI: 10.7270/Q2P84952 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078974 (1-Isopropyl-3-{3-[3-(N'-methyl-N''-phenyl-guanidin...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078994 (1-Benzooxazol-5-yl-3-{1-[3-(3-isopropyl-ureido)-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078971 (1-Indan-5-yl-3-{1-[3-(3-isopropyl-ureido)-benzyl]-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 17 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078981 (1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-{1-[3-(3-i...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078993 (1-(1H-Indol-5-yl)-3-{1-[3-(3-isopropyl-ureido)-ben...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Androgen receptor (Homo sapiens (Human)) | BDBM18525 (Bicalutamide | CHEMBL409 | N-[4-cyano-3-(trifluoro...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Astellas Pharma Inc. | Assay Description The Ki values were determined by the application of the Cheng-Prusoff equation: Ki=IC50/(1+[L]/Kd] where [L] is the concentration of labeled ligand a... | J Med Chem 49: 716-26 (2006) Article DOI: 10.1021/jm050293c BindingDB Entry DOI: 10.7270/Q2P84952 | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079017 (1-Benzothiazol-5-yl-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 24 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078995 (1-(1,3-Dioxo-2,3-dihydro-1H-isoindol-5-yl)-3-{1-[3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078959 (1-(1H-Indazol-5-yl)-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078975 (1-Benzo[1,3]dioxol-5-yl-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078985 (1-(4-Fluoro-phenyl)-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 29 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078957 (1-(3-{3-[N'-(4-Hydroxy-phenyl)-N''-isopropyl-guani...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078979 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079013 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 56 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078972 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-1,2,3,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 56 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078990 (1-(3-{3-[N'-(2-Hydroxy-ethyl)-N''-(4-hydroxy-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078967 (1-(4-Dimethylamino-phenyl)-3-{1-[3-(3-isopropyl-ur...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 66 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078998 (1-(4-Chloro-phenyl)-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 71 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078976 (1-{1-[3-(3-Isobutyl-ureido)-benzyl]-2-oxo-2,3,4,5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 75 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079002 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078969 (1-(4-Hydroxy-phenyl)-3-{1-[3-(3-isopropyl-ureido)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 82 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079011 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 83 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078996 (1-(3,5-Difluoro-phenyl)-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 86 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078987 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079010 (1-(2,3-Difluoro-phenyl)-3-{1-[3-(3-isopropyl-ureid...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078988 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078973 (1-{1-[3-(3-tert-Butyl-ureido)-benzyl]-2-oxo-2,3,4,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078956 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 150 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078960 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 160 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078984 (1-(4-Amino-phenyl)-3-{1-[3-(3-isopropyl-ureido)-be...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079004 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50079005 (CHEMBL314637 | Phenyl-carbamic acid 1-[3-(3-isopro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078968 (1-{9-[3-(3-Isopropyl-ureido)-benzyl]-8-oxo-6,7,8,9...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078963 (1-Biphenyl-4-yl-3-{1-[3-(3-isopropyl-ureido)-benzy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 610 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078992 (CHEMBL84632 | {3-[2-Oxo-3-(3-phenyl-ureido)-2,3,4,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078961 (1-Benzothiazol-2-yl-3-{1-[3-(3-isopropyl-ureido)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078964 (1-{1-[3-(3-Isopropyl-ureido)-benzyl]-2-oxo-2,3,4,5...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 780 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Neuropeptide Y receptor type 1 (Homo sapiens (Human)) | BDBM50078980 (1-{1-[3-(3-Cyclopropyl-ureido)-benzyl]-2-oxo-2,3,4...) | PDB Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 910 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Shionogi & Company, Ltd. Curated by ChEMBL | Assay Description In vitro binding affinity towards Neuropeptide Y receptor type 1 was determined as potency to displace [125I]-peptide YY binding to human neuroblasto... | J Med Chem 42: 2621-32 (1999) Article DOI: 10.1021/jm990044m BindingDB Entry DOI: 10.7270/Q2XK8DRQ | |||||||||||
More data for this Ligand-Target Pair |
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