Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50427221 (5-Aminonicotinic Acid | CHEMBL1491941) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Binding affinity to human recombinant DDO | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG38204, isoform CRA_d (Rattus norvegicus) | BDBM50427221 (5-Aminonicotinic Acid | CHEMBL1491941) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | 5.89E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of rat recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Mus musculus) | BDBM50427221 (5-Aminonicotinic Acid | CHEMBL1491941) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | 8.69E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of mouse recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121995 (CHEMBL3617316) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.51E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Binding affinity to human recombinant DDO | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Mus musculus) | BDBM50121995 (CHEMBL3617316) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.26E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of mouse recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG38204, isoform CRA_d (Rattus norvegicus) | BDBM50121995 (CHEMBL3617316) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.59E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of rat recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM14673 (Fragment 3 | Malonic Acid | propanedioic acid) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.53E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Binding affinity to human recombinant DDO | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Mus musculus) | BDBM14673 (Fragment 3 | Malonic Acid | propanedioic acid) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.22E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of mouse recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
RCG38204, isoform CRA_d (Rattus norvegicus) | BDBM14673 (Fragment 3 | Malonic Acid | propanedioic acid) | UniProtKB/TrEMBL GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 1.56E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of rat recombinant DDO using D-Asp | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122008 (CHEMBL3617314) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.34E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50427221 (5-Aminonicotinic Acid | CHEMBL1491941) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.19E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121995 (CHEMBL3617316) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.71E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50121996 (CHEMBL3617326) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50121997 (CHEMBL3322863) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50121998 (CHEMBL3322866) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122001 (CHEMBL3617320) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121996 (CHEMBL3617326) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121997 (CHEMBL3322863) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121998 (CHEMBL3322866) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122001 (CHEMBL3617320) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM197302 (Benzoic acid | SAMPL4, O1) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid PDB UniChem | DrugBank PDB Article PubMed | n/a | n/a | 1.34E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122006 (CHEMBL3617317) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.47E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50226518 (3-Aminobenzoesaeure | 3-aminobenzoic acid | CHEMBL...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 3.92E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50121995 (CHEMBL3617316) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM14673 (Fragment 3 | Malonic Acid | propanedioic acid) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase DrugBank KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 8.79E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122008 (CHEMBL3617314) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122000 (CHEBI:68572 | CHEMBL3322868) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122003 (CHEMBL3617319) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122018 (CHEMBL1529836) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122003 (CHEMBL3617319) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122000 (CHEBI:68572 | CHEMBL3322868) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50219484 (5-fluorosalicylic acid | CHEMBL229239) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 1.05E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM23515 (CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.13E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122007 (CHEMBL3617315) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.44E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50216534 (5-methylnicotinic acid | CHEMBL247132) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50052793 (CHEBI:68583 | CHEMBL3322864) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.36E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122011 (3-Hydroxypicolinic Acid | CHEBI:64342 | CHEMBL1234...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | 2.48E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50052793 (CHEBI:68583 | CHEMBL3322864) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >2.50E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50427221 (5-Aminonicotinic Acid | CHEMBL1491941) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | >2.50E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM23515 (CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 2.78E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50391823 (CHEMBL2146902) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE MMDB PC cid PC sid PDB UniChem | Article PubMed | n/a | n/a | 3.35E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50121999 (CHEMBL1588120) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.54E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50240969 (5-Chloro-2-hydroxy-benzoic acid | 5-Chlorosalicyli...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.67E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122010 (CHEMBL36767) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.93E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122007 (CHEMBL3617315) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.25E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-amino-acid oxidase (Homo sapiens (Human)) | BDBM50122002 (CHEMBL1383671) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >5.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122002 (CHEMBL1383671) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >5.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122006 (CHEMBL3617317) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >5.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50122014 (CHEMBL3617324) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | >5.00E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
D-aspartate oxidase (Homo sapiens (Human)) | BDBM50216534 (5-methylnicotinic acid | CHEMBL247132) | PDB KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 5.47E+6 | n/a | n/a | n/a | n/a | n/a | n/a |
Kitasato University Curated by ChEMBL | Assay Description Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ... | J Med Chem 58: 7328-40 (2015) Article DOI: 10.1021/acs.jmedchem.5b00871 BindingDB Entry DOI: 10.7270/Q2WM1G6R | |||||||||||
More data for this Ligand-Target Pair |
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