Found 324 hits with Last Name = 'lacoste' and Initial = 'jm' Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM81807
(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)Show InChI InChI=1S/C14H16N2/c1-2-14(13-9-15-10-16-13)7-11-5-3-4-6-12(11)8-14/h3-6,9-10H,2,7-8H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
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MCE PC cid PC sid UniChem
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Similars
| Article PubMed
| 0.126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(RAT) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.159 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]
(Rattus norvegicus (rat)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2B adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.251 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.346 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.562 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 0.631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473523
(CHEMBL167578)Show InChI InChI=1S/C14H16N2/c1-2-4-11-6-14(5-10(11)3-1)7-12(14)13-8-15-9-16-13/h1-4,9,12-13H,5-8H2,(H,15,16)/t12?,13-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 0.794 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(RAT) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
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| PubMed
| 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50473529
(CHEMBL165529)Show SMILES [H][C@]12CC[C@]3(CN=CN3)C[C@]1([H])Cc1ccccc1C2 |c:6| Show InChI InChI=1S/C16H20N2/c1-2-4-13-8-15-9-16(10-17-11-18-16)6-5-14(15)7-12(13)3-1/h1-4,11,14-15H,5-10H2,(H,17,18)/t14-,15+,16-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cell |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473526
(CHEMBL168201)Show InChI InChI=1S/C14H14N2/c1-2-4-13-7-11(5-6-12(13)3-1)8-14-9-15-10-16-14/h1-4,7,9-10H,5-6,8H2,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473556
(CHEMBL355467)Show InChI InChI=1S/C13H15FN2/c14-13-3-1-2-10-4-9(6-12(10)13)5-11-7-15-8-16-11/h1-3,8-9,11H,4-7H2,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473565
(CHEMBL436234)Show InChI InChI=1S/C14H15FN2/c15-13-4-3-11-2-1-10(5-12(11)7-13)6-14-8-16-9-17-14/h3-5,7,9,14H,1-2,6,8H2,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473533
(CHEMBL166690)Show InChI InChI=1S/C14H17ClN2/c15-14-3-1-2-11-5-4-10(7-13(11)14)6-12-8-16-9-17-12/h1-3,9-10,12H,4-8H2,(H,16,17) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031306
(8-chlorospiro[1,2,3,4-tetrahydronaphthalene-2,4'-(...)Show InChI InChI=1S/C12H13ClN2O/c13-10-3-1-2-8-4-5-12(6-9(8)10)7-16-11(14)15-12/h1-3H,4-7H2,(H2,14,15) | PDB
UniProtKB/SwissProt
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| 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Alpha-2B adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| PubMed
| 2.00 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473543
(CHEMBL353843)Show InChI InChI=1S/C13H16N2/c1-2-4-12-6-10(5-11(12)3-1)7-13-8-14-9-15-13/h1-4,9-10,13H,5-8H2,(H,14,15) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473534
(CHEMBL354611)Show SMILES [H][C@]1(CN=CN1)C1C[C@@]11CCc2ccccc2C1 |c:3| Show InChI InChI=1S/C15H18N2/c1-2-4-12-7-15(6-5-11(12)3-1)8-13(15)14-9-16-10-17-14/h1-4,10,13-14H,5-9H2,(H,16,17)/t13?,14-,15-/m0/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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| 2.04 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
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| PubMed
| 2.51 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031324
(5',7'-dichlorospiro[4,5-dihydro-1H-imidazole-4,2'-...)Show InChI InChI=1S/C12H12Cl2N2/c13-9-3-8-5-12(6-15-7-16-12)2-1-10(8)11(14)4-9/h3-4,7H,1-2,5-6H2,(H,15,16) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| PubMed
| 3.16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM81807
(ATIPAMEZOLE | CAS_104054-27-5 | NSC_71310)Show InChI InChI=1S/C14H16N2/c1-2-14(13-9-15-10-16-13)7-11-5-3-4-6-12(11)8-14/h3-6,9-10H,2,7-8H2,1H3,(H,15,16) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| Purchase
MCE PC cid PC sid UniChem
Patents
Similars
| Article PubMed
| 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cell |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50454831
(Napamezole)Show InChI InChI=1S/C14H16N2/c1-2-4-13-9-11(5-6-12(13)3-1)10-14-15-7-8-16-14/h1-4,9H,5-8,10H2,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| Purchase
PC cid PC sid UniChem
| Article PubMed
| 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50473534
(CHEMBL354611)Show SMILES [H][C@]1(CN=CN1)C1C[C@@]11CCc2ccccc2C1 |c:3| Show InChI InChI=1S/C15H18N2/c1-2-4-12-7-15(6-5-11(12)3-1)8-13(15)14-9-16-10-17-14/h1-4,10,13-14H,5-9H2,(H,16,17)/t13?,14-,15-/m0/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cell |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-1A adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 3.98 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50473543
(CHEMBL353843)Show InChI InChI=1S/C13H16N2/c1-2-4-12-6-10(5-11(12)3-1)7-13-8-14-9-15-13/h1-4,9-10,13H,5-8H2,(H,14,15) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cell |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2B adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 4.37 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473533
(CHEMBL166690)Show InChI InChI=1S/C14H17ClN2/c15-14-3-1-2-11-5-4-10(7-13(11)14)6-12-8-16-9-17-12/h1-3,9-10,12H,4-8H2,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 6.03 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473534
(CHEMBL354611)Show SMILES [H][C@]1(CN=CN1)C1C[C@@]11CCc2ccccc2C1 |c:3| Show InChI InChI=1S/C15H18N2/c1-2-4-12-7-15(6-5-11(12)3-1)8-13(15)14-9-16-10-17-14/h1-4,10,13-14H,5-9H2,(H,16,17)/t13?,14-,15-/m0/s1 | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM30130
(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)Show InChI InChI=1S/C17H18F3NO/c1-21-12-11-16(13-5-3-2-4-6-13)22-15-9-7-14(8-10-15)17(18,19)20/h2-10,16,21H,11-12H2,1H3 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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CHEMBL DrugBank MCE PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| 6.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description Binding affinity for human alpha-2 adrenergic receptor expressed in CHO cell |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-1A adrenergic receptor
(Rattus norvegicus (Rat)) | BDBM85709
(S18616)Show InChI InChI=1S/C12H14N2O/c13-11-14-12(8-15-11)6-5-9-3-1-2-4-10(9)7-12/h1-4H,5-8H2,(H2,13,14) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
Similars
| PubMed
| 6.31 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031311
(7'-methylspiro[4,5-dihydro-1H-imidazole-4,2'-(1',2...)Show InChI InChI=1S/C13H16N2/c1-10-2-3-11-4-5-13(7-12(11)6-10)8-14-9-15-13/h2-3,6,9H,4-5,7-8H2,1H3,(H,14,15) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50131357
(4-(5-Fluoro-indan-2-ylmethyl)-4,5-dihydro-1H-imida...)Show InChI InChI=1S/C13H15FN2/c14-12-2-1-10-3-9(4-11(10)6-12)5-13-7-15-8-16-13/h1-2,6,8-9,13H,3-5,7H2,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Patents
| Article PubMed
| 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473547
(CHEMBL166648)Show InChI InChI=1S/C15H20N2/c1-15(9-14-10-16-11-17-14)7-6-12-4-2-3-5-13(12)8-15/h2-5,11,14H,6-10H2,1H3,(H,16,17)/t14-,15-/m1/s1 | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM30130
(CHEMBL1201082 | CHEMBL41 | Fluoxetin | Fluoxetine ...)Show InChI InChI=1S/C17H18F3NO/c1-21-12-11-16(13-5-3-2-4-6-13)22-15-9-7-14(8-10-15)17(18,19)20/h2-10,16,21H,11-12H2,1H3 | PDB
KEGG
UniProtKB/SwissProt
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| Purchase
CHEMBL DrugBank MCE PC cid PC sid PDB UniChem
Patents
Similars
| Article PubMed
| 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473529
(CHEMBL165529)Show SMILES [H][C@]12CC[C@]3(CN=CN3)C[C@]1([H])Cc1ccccc1C2 |c:6| Show InChI InChI=1S/C16H20N2/c1-2-4-13-8-15-9-16(10-17-11-18-16)6-5-14(15)7-12(13)3-1/h1-4,11,14-15H,5-10H2,(H,17,18)/t14-,15+,16-/m1/s1 | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473560
(CHEMBL166748)Show InChI InChI=1S/C14H18N2/c1-2-4-13-7-11(5-6-12(13)3-1)8-14-9-15-10-16-14/h1-4,10-11,14H,5-9H2,(H,15,16) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031316
(5'-methoxyspiro[4,5-dihydro-1H-imidazole-4,2'-(1',...)Show InChI InChI=1S/C13H16N2O/c1-16-12-4-2-3-10-7-13(6-5-11(10)12)8-14-9-15-13/h2-4,9H,5-8H2,1H3,(H,14,15) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50031301
(8'-fluorospiro[4,5-dihydro-1H-imidazole-4,2'-(1',2...)Show InChI InChI=1S/C12H13FN2/c13-11-3-1-2-9-4-5-12(6-10(9)11)7-14-8-15-12/h1-3,8H,4-7H2,(H,14,15) | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
| CHEMBL PC cid PC sid UniChem
Similars
| PubMed
| 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by ChEMBL
| Assay Description Binding affinity towards Alpha-2A adrenergic receptor in human platelets using [3H]-RX-821002 as radioligand |
J Med Chem 38: 4056-69 (1995)
BindingDB Entry DOI: 10.7270/Q2DV1HXN |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473555
(CHEMBL352643)Show InChI InChI=1S/C13H14F2N2/c14-12-4-9-1-8(2-10(9)5-13(12)15)3-11-6-16-7-17-11/h4-5,7-8,11H,1-3,6H2,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473550
(CHEMBL354072)Show InChI InChI=1S/C15H18N2/c1-11-3-2-4-13-6-5-12(8-15(11)13)7-14-9-16-10-17-14/h2-4,8,10,14H,5-7,9H2,1H3,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473525
(CHEMBL167644)Show InChI InChI=1S/C12H12N2O/c1-2-4-12-9(3-1)5-11(15-12)6-10-7-13-8-14-10/h1-5,8,10H,6-7H2,(H,13,14) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2C adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
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CHEMBL MCE PC cid PC sid UniChem
Patents
Similars
| PubMed
| 15.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor
(Homo sapiens (Human)) | BDBM50241196
((R)-5-(1-(2,3-dimethylphenyl)ethyl)-1H-imidazole |...)Show InChI InChI=1S/C13H16N2/c1-9-5-4-6-12(10(9)2)11(3)13-7-14-8-15-13/h4-8,11H,1-3H3,(H,14,15)/t11-/m1/s1 | PDB
UniProtKB/SwissProt
antibodypedia GoogleScholar AffyNet
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CHEMBL MCE PC cid PC sid UniChem
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| PubMed
| 15.8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Centre de Recherches de Croissy
Curated by PDSP Ki Database
| |
J Pharmacol Exp Ther 295: 1192-205 (2000)
BindingDB Entry DOI: 10.7270/Q28P5Z2C |
More data for this Ligand-Target Pair | |
Sodium-dependent serotonin transporter
(Rattus norvegicus (rat)) | BDBM50473563
(CHEMBL352636)Show InChI InChI=1S/C15H18N2O/c1-18-15-4-2-3-12-6-5-11(8-14(12)15)7-13-9-16-10-17-13/h2-4,8,10,13H,5-7,9H2,1H3,(H,16,17) | PDB
KEGG
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against serotonin reuptake site of rat in presence of [3H]paroxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor
(RAT-NEONATAL RAT-Rattus norvegicus (rat)) | BDBM50473560
(CHEMBL166748)Show InChI InChI=1S/C14H18N2/c1-2-4-13-7-11(5-6-12(13)3-1)8-14-9-15-10-16-14/h1-4,10-11,14H,5-9H2,(H,15,16) | PDB
UniProtKB/SwissProt
GoogleScholar AffyNet
| PC cid PC sid UniChem
| Article PubMed
| 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity against alpha-2 adrenergic receptor of rat in presence of [3H]-RX 821002 radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |
Transporter
(Rattus norvegicus) | BDBM50335519
((S)-3,6-Diamino-hexanoic acid {(3S,9S,12S,15S)-3-(...)Show SMILES CN[C@H](CC(C)C)C(=O)N[C@@H]1[C@H](O)c2ccc(Oc3cc4cc(Oc5ccc(cc5Cl)[C@@H](O)[C@@H]5NC(=O)[C@H](NC(=O)[C@@H]4NC(=O)[C@H](CC(N)=O)NC1=O)c1ccc(O)c(c1)-c1c(O)cc(O)cc1[C@H](NC5=O)C(O)=O)c3O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1O[C@H]1C[C@](C)(N)[C@H](O)[C@H](C)O1)c(Cl)c2 |r| Show InChI InChI=1S/C66H75Cl2N9O24/c1-23(2)12-34(71-5)58(88)76-49-51(83)26-7-10-38(32(67)14-26)97-40-16-28-17-41(55(40)101-65-56(54(86)53(85)42(22-78)99-65)100-44-21-66(4,70)57(87)24(3)96-44)98-39-11-8-27(15-33(39)68)52(84)50-63(93)75-48(64(94)95)31-18-29(79)19-37(81)45(31)30-13-25(6-9-36(30)80)46(60(90)77-50)74-61(91)47(28)73-59(89)35(20-43(69)82)72-62(49)92/h6-11,13-19,23-24,34-35,42,44,46-54,56-57,65,71,78-81,83-87H,12,20-22,70H2,1-5H3,(H2,69,82)(H,72,92)(H,73,89)(H,74,91)(H,75,93)(H,76,88)(H,77,90)(H,94,95)/t24-,34+,35-,42+,44-,46+,47+,48-,49+,50-,51+,52+,53+,54-,56+,57+,65-,66-/m0/s1 | Reactome pathway KEGG
UniProtKB/TrEMBL
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CHEMBL DrugBank MCE PC cid PC sid UniChem
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| Article PubMed
| 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Institut de Recherches Servier
Curated by PDSP Ki Database
| Assay Description In vitro binding affinity was determined against NA (noradrenaline) reuptake site of rat in presence of [3H]nisoxetine radioligand |
J Med Chem 44: 787-805 (2001)
Article DOI: 10.1021/jm001040g BindingDB Entry DOI: 10.7270/Q2JQ13R9 |
More data for this Ligand-Target Pair | |