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Compile Data Set for Download or QSAR

Found 63 hits with Last Name = 'paramonova' and Initial = 'mp'   
Target/Host
(Institution)		LigandTarget/Host
Links		Ligand
Links		Trg + Lig
Links		Ki
nM		ΔG°
kJ/mole		IC50
nM		Kd
nM		EC50/IC50
nM		koff
s-1		kon
M-1s-1		pHTemp
°C
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM2483
PNG
((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Show SMILES FC(F)(F)[C@]1(OC(=O)Nc2ccc(Cl)cc12)C#CC1CC1 |r|
Show InChI InChI=1S/C14H9ClF3NO2/c15-9-3-4-11-10(7-9)13(14(16,17)18,21-12(20)19-11)6-5-8-1-2-8/h3-4,7-8H,1-2H2,(H,19,20)/t13-/m0/s1
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 10n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490649
PNG
(CHEMBL2337184)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3cc(C)cc(C)c3)c2=O)cc1
Show InChI InChI=1S/C22H24N2O3/c1-16-4-6-20(7-5-16)27-11-10-23-9-8-21(25)24(22(23)26)15-19-13-17(2)12-18(3)14-19/h4-9,12-14H,10-11,15H2,1-3H3
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 260n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490643
PNG
(CHEMBL2337196)
Show SMILES Cc1cc(Br)cc(Cn2c(=O)ccn(C\C=C\c3ccccc3)c2=O)c1
Show InChI InChI=1S/C21H19BrN2O2/c1-16-12-18(14-19(22)13-16)15-24-20(25)9-11-23(21(24)26)10-5-8-17-6-3-2-4-7-17/h2-9,11-14H,10,15H2,1H3/b8-5+
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 310n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490644
PNG
(CHEMBL2337195)
Show SMILES Brc1cc(Br)cc(Cn2c(=O)ccn(C\C=C\c3ccccc3)c2=O)c1
Show InChI InChI=1S/C20H16Br2N2O2/c21-17-11-16(12-18(22)13-17)14-24-19(25)8-10-23(20(24)26)9-4-7-15-5-2-1-3-6-15/h1-8,10-13H,9,14H2/b7-4+
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 310n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490669
PNG
(CHEMBL2337192)
Show SMILES Cc1cc(C)cc(Cn2c(=O)ccn(C\C=C\c3ccccc3)c2=O)c1
Show InChI InChI=1S/C22H22N2O2/c1-17-13-18(2)15-20(14-17)16-24-21(25)10-12-23(22(24)26)11-6-9-19-7-4-3-5-8-19/h3-10,12-15H,11,16H2,1-2H3/b9-6+
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 550n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490662
PNG
(CHEMBL2337194)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(C\C=C\c3ccccc3)c2=O)c1
Show InChI InChI=1S/C20H16Cl2N2O2/c21-17-11-16(12-18(22)13-17)14-24-19(25)8-10-23(20(24)26)9-4-7-15-5-2-1-3-6-15/h1-8,10-13H,9,14H2/b7-4+
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 670n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490648
PNG
(CHEMBL2337186)
Show SMILES Cc1ccc(OCCn2cc(C)c(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C21H22N2O3/c1-16-8-10-19(11-9-16)26-13-12-22-14-17(2)20(24)23(21(22)25)15-18-6-4-3-5-7-18/h3-11,14H,12-13,15H2,1-2H3
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 1.00E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490668
PNG
(CHEMBL2337189)
Show SMILES O=c1ccn(CCOc2ccc3ccccc3c2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C23H20N2O3/c26-22-12-13-24(23(27)25(22)17-18-6-2-1-3-7-18)14-15-28-21-11-10-19-8-4-5-9-20(19)16-21/h1-13,16H,14-15,17H2
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 1.00E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490646
PNG
(CHEMBL2337190)
Show SMILES Cc1ccc(OCCn2c3ccccc3c(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C24H22N2O3/c1-18-11-13-20(14-12-18)29-16-15-25-22-10-6-5-9-21(22)23(27)26(24(25)28)17-19-7-3-2-4-8-19/h2-14H,15-17H2,1H3
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 1.00E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 4.50E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490660
PNG
(CHEMBL2337187)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(CCc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C21H22N2O3/c1-17-7-9-19(10-8-17)26-16-15-22-13-12-20(24)23(21(22)25)14-11-18-5-3-2-4-6-18/h2-10,12-13H,11,14-16H2,1H3
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 6.50E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490665
PNG
(CHEMBL2337181)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3cccc(C)c3)c2=O)cc1
Show InChI InChI=1S/C21H22N2O3/c1-16-6-8-19(9-7-16)26-13-12-22-11-10-20(24)23(21(22)25)15-18-5-3-4-17(2)14-18/h3-11,14H,12-13,15H2,1-2H3
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 6.60E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490642
PNG
(CHEMBL2337197)
Show SMILES O=c1ccn(C\C=C\c2ccccc2)c(=O)n1Cc1cccc2ccccc12
Show InChI InChI=1S/C24H20N2O2/c27-23-15-17-25(16-7-10-19-8-2-1-3-9-19)24(28)26(23)18-21-13-6-12-20-11-4-5-14-22(20)21/h1-15,17H,16,18H2/b10-7+
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 6.60E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM1434
PNG
(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Show SMILES Cc1ccnc2N(C3CC3)c3ncccc3C(=O)Nc12
Show InChI InChI=1S/C15H14N4O/c1-9-6-8-17-14-12(9)18-15(20)11-3-2-7-16-13(11)19(14)10-4-5-10/h2-3,6-8,10H,4-5H2,1H3,(H,18,20)
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 7.20E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490659
PNG
(CHEMBL2337174)
Show SMILES O=c1ccn(CCOc2ccc(cc2)-c2ccccc2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C25H22N2O3/c28-24-15-16-26(25(29)27(24)19-20-7-3-1-4-8-20)17-18-30-23-13-11-22(12-14-23)21-9-5-2-6-10-21/h1-16H,17-19H2
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 8.10E+3n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490650
PNG
(CHEMBL2337183)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3cc(C)ccc3C)c2=O)cc1
Show InChI InChI=1S/C22H24N2O3/c1-16-5-8-20(9-6-16)27-13-12-23-11-10-21(25)24(22(23)26)15-19-14-17(2)4-7-18(19)3/h4-11,14H,12-13,15H2,1-3H3
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 1.00E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490647
PNG
(CHEMBL2337188)
Show SMILES CC(c1ccccc1)n1c(=O)ccn(CCOc2ccc(C)cc2)c1=O
Show InChI InChI=1S/C21H22N2O3/c1-16-8-10-19(11-9-16)26-15-14-22-13-12-20(24)23(21(22)25)17(2)18-6-4-3-5-7-18/h3-13,17H,14-15H2,1-2H3
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 1.20E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490645
PNG
(CHEMBL2337193)
Show SMILES Fc1cc(F)cc(Cn2c(=O)ccn(C\C=C\c3ccccc3)c2=O)c1
Show InChI InChI=1S/C20H16F2N2O2/c21-17-11-16(12-18(22)13-17)14-24-19(25)8-10-23(20(24)26)9-4-7-15-5-2-1-3-6-15/h1-8,10-13H,9,14H2/b7-4+
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 1.20E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490653
PNG
(CHEMBL2337173)
Show SMILES CC(C)(C)c1ccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C23H26N2O3/c1-23(2,3)19-9-11-20(12-10-19)28-16-15-24-14-13-21(26)25(22(24)27)17-18-7-5-4-6-8-18/h4-14H,15-17H2,1-3H3
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 1.50E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 1.54E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 1.59E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase L100I mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 2.00E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase G190A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490658
PNG
(CHEMBL2337175)
Show SMILES Clc1ccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C19H17ClN2O3/c20-16-6-8-17(9-7-16)25-13-12-21-11-10-18(23)22(19(21)24)14-15-4-2-1-3-5-15/h1-11H,12-14H2
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 2.20E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490663
PNG
(CHEMBL2337191)
Show SMILES O=c1ccn(C\C=C\c2ccccc2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C20H18N2O2/c23-19-13-15-21(14-7-12-17-8-3-1-4-9-17)20(24)22(19)16-18-10-5-2-6-11-18/h1-13,15H,14,16H2/b12-7+
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 2.90E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490657
PNG
(CHEMBL2337182)
Show SMILES Cc1ccc(Cn2c(=O)ccn(CCOc3ccc(C)cc3)c2=O)cc1
Show InChI InChI=1S/C21H22N2O3/c1-16-3-7-18(8-4-16)15-23-20(24)11-12-22(21(23)25)13-14-26-19-9-5-17(2)6-10-19/h3-12H,13-15H2,1-2H3
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 4.70E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490652
PNG
(CHEMBL2337177)
Show SMILES O=c1ccn(CCOc2ccc(cc2)C#N)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C20H17N3O3/c21-14-16-6-8-18(9-7-16)26-13-12-22-11-10-19(24)23(20(22)25)15-17-4-2-1-3-5-17/h1-11H,12-13,15H2
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 5.10E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490654
PNG
(CHEMBL2337201)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C20H20N2O3/c1-16-7-9-18(10-8-16)25-14-13-21-12-11-19(23)22(20(21)24)15-17-5-3-2-4-6-17/h2-12H,13-15H2,1H3
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 5.20E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 6.33E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase K103N mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 6.76E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase V106A mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer compl...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490656
PNG
(CHEMBL2337198)
Show SMILES O=c1ccn(CCOc2ccccc2)c(=O)n1Cc1ccccc1
Show InChI InChI=1S/C19H18N2O3/c22-18-11-12-20(13-14-24-17-9-5-2-6-10-17)19(23)21(18)15-16-7-3-1-4-8-16/h1-12H,13-15H2
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 6.80E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063002
PNG
(CHEMBL3398101)
Show SMILES Clc1cc(Cl)cc(Cn2c(=O)ccn(CC(=O)Nc3ccccc3Cl)c2=O)c1
Show InChI InChI=1S/C19H14Cl3N3O3/c20-13-7-12(8-14(21)9-13)10-25-18(27)5-6-24(19(25)28)11-17(26)23-16-4-2-1-3-15(16)22/h1-9H,10-11H2,(H,23,26)
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 6.99E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 reverse transcriptase K103N/Y181C mutant using radioactively-labeled [alpha-32P]ATP substrate and activated DNA as template-primer...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490661
PNG
(CHEMBL2337176)
Show SMILES Fc1ccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)cc1
Show InChI InChI=1S/C19H17FN2O3/c20-16-6-8-17(9-7-16)25-13-12-21-11-10-18(23)22(19(21)24)14-15-4-2-1-3-5-15/h1-11H,12-14H2
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 7.10E+4n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063018
PNG
(CHEMBL3398086)
Show SMILES Cn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2ccc(Cl)cc2)c1=O
Show InChI InChI=1S/C20H18ClN3O4/c1-23-19(26)10-11-24(20(23)27)12-14-4-2-3-5-17(14)28-13-18(25)22-16-8-6-15(21)7-9-16/h2-11H,12-13H2,1H3,(H,22,25)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063017
PNG
(CHEMBL3398085)
Show SMILES Cn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2cccc(Cl)c2)c1=O
Show InChI InChI=1S/C20H18ClN3O4/c1-23-19(26)9-10-24(20(23)27)12-14-5-2-3-8-17(14)28-13-18(25)22-16-7-4-6-15(21)11-16/h2-11H,12-13H2,1H3,(H,22,25)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063010
PNG
(CHEMBL3398082)
Show SMILES Cn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2ccccc2)c1=O
Show InChI InChI=1S/C20H19N3O4/c1-22-19(25)11-12-23(20(22)26)13-15-7-5-6-10-17(15)27-14-18(24)21-16-8-3-2-4-9-16/h2-12H,13-14H2,1H3,(H,21,24)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063019
PNG
(CHEMBL3398087)
Show SMILES Cn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2cc(Cl)ccc2Cl)c1=O
Show InChI InChI=1S/C20H17Cl2N3O4/c1-24-19(27)8-9-25(20(24)28)11-13-4-2-3-5-17(13)29-12-18(26)23-16-10-14(21)6-7-15(16)22/h2-10H,11-12H2,1H3,(H,23,26)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490670
PNG
(CHEMBL2337180)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3ccccc3C)c2=O)cc1
Show InChI InChI=1S/C21H22N2O3/c1-16-7-9-19(10-8-16)26-14-13-22-12-11-20(24)23(21(22)25)15-18-6-4-3-5-17(18)2/h3-12H,13-15H2,1-2H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063020
PNG
(CHEMBL3398088)
Show SMILES CCCn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2ccccc2Cl)c1=O
Show InChI InChI=1S/C22H22ClN3O4/c1-2-12-26-21(28)11-13-25(22(26)29)14-16-7-3-6-10-19(16)30-15-20(27)24-18-9-5-4-8-17(18)23/h3-11,13H,2,12,14-15H2,1H3,(H,24,27)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063023
PNG
(CHEMBL3398090)
Show SMILES Cc1cn(Cc2ccccc2OCC(=O)Nc2ccccc2Cl)c(=O)n(C)c1=O
Show InChI InChI=1S/C21H20ClN3O4/c1-14-11-25(21(28)24(2)20(14)27)12-15-7-3-6-10-18(15)29-13-19(26)23-17-9-5-4-8-16(17)22/h3-11H,12-13H2,1-2H3,(H,23,26)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490655
PNG
(CHEMBL2337199)
Show SMILES Cc1ccccc1OCCn1ccc(=O)n(Cc2ccccc2)c1=O
Show InChI InChI=1S/C20H20N2O3/c1-16-7-5-6-10-18(16)25-14-13-21-12-11-19(23)22(20(21)24)15-17-8-3-2-4-9-17/h2-12H,13-15H2,1H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063001
PNG
(CHEMBL3398091)
Show SMILES Cn1c(=O)c(F)cn(Cc2ccccc2OCC(=O)Nc2ccccc2Cl)c1=O
Show InChI InChI=1S/C20H17ClFN3O4/c1-24-19(27)15(22)11-25(20(24)28)10-13-6-2-5-9-17(13)29-12-18(26)23-16-8-4-3-7-14(16)21/h2-9,11H,10,12H2,1H3,(H,23,26)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490667
PNG
(CHEMBL2337200)
Show SMILES Cc1cccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)c1
Show InChI InChI=1S/C20H20N2O3/c1-16-6-5-9-18(14-16)25-13-12-21-11-10-19(23)22(20(21)24)15-17-7-3-2-4-8-17/h2-11,14H,12-13,15H2,1H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490666
PNG
(CHEMBL2337178)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)cc1C
Show InChI InChI=1S/C21H22N2O3/c1-16-8-9-19(14-17(16)2)26-13-12-22-11-10-20(24)23(21(22)25)15-18-6-4-3-5-7-18/h3-11,14H,12-13,15H2,1-2H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490664
PNG
(CHEMBL2337185)
Show SMILES Cc1ccc(OCCn2ccc(=O)n(Cc3c(C)cc(C)cc3C)c2=O)cc1
Show InChI InChI=1S/C23H26N2O3/c1-16-5-7-20(8-6-16)28-12-11-24-10-9-22(26)25(23(24)27)15-21-18(3)13-17(2)14-19(21)4/h5-10,13-14H,11-12,15H2,1-4H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063003
PNG
(CHEMBL3398092)
Show SMILES Cn1c(=O)c(Cl)cn(Cc2ccccc2OCC(=O)Nc2ccccc2Cl)c1=O
Show InChI InChI=1S/C20H17Cl2N3O4/c1-24-19(27)15(22)11-25(20(24)28)10-13-6-2-5-9-17(13)29-12-18(26)23-16-8-4-3-7-14(16)21/h2-9,11H,10,12H2,1H3,(H,23,26)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063022
PNG
(CHEMBL3398089)
Show SMILES Clc1ccccc1NC(=O)COc1ccccc1Cn1ccc(=O)n(CC=C)c1=O
Show InChI InChI=1S/C22H20ClN3O4/c1-2-12-26-21(28)11-13-25(22(26)29)14-16-7-3-6-10-19(16)30-15-20(27)24-18-9-5-4-8-17(18)23/h2-11,13H,1,12,14-15H2,(H,24,27)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063013
PNG
(CHEMBL3398083)
Show SMILES Cc1ccccc1NC(=O)COc1ccccc1Cn1ccc(=O)n(C)c1=O
Show InChI InChI=1S/C21H21N3O4/c1-15-7-3-5-9-17(15)22-19(25)14-28-18-10-6-4-8-16(18)13-24-12-11-20(26)23(2)21(24)27/h3-12H,13-14H2,1-2H3,(H,22,25)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50063014
PNG
(CHEMBL3398084)
Show SMILES Cn1c(=O)ccn(Cc2ccccc2OCC(=O)Nc2ccccc2Cl)c1=O
Show InChI InChI=1S/C20H18ClN3O4/c1-23-19(26)10-11-24(20(23)27)12-14-6-2-5-9-17(14)28-13-18(25)22-16-8-4-3-7-15(16)21/h2-11H,12-13H2,1H3,(H,22,25)
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM50490651
PNG
(CHEMBL2337179)
Show SMILES Cc1cc(C)cc(OCCn2ccc(=O)n(Cc3ccccc3)c2=O)c1
Show InChI InChI=1S/C21H22N2O3/c1-16-12-17(2)14-19(13-16)26-11-10-22-9-8-20(24)23(21(22)25)15-18-6-4-3-5-7-18/h3-9,12-14H,10-11,15H2,1-2H3
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>1.00E+5n/an/an/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Non-competitive inhibition of wild type HIV1 reverse transcriptase p66/p51 after 30 mins by liquid scintillation counting

Bioorg Med Chem 21: 1150-8 (2013)


Article DOI: 10.1016/j.bmc.2012.12.027
BindingDB Entry DOI: 10.7270/Q2NZ8BKZ
More data for this
Ligand-Target Pair
Reverse transcriptase


(Human immunodeficiency virus 1)		BDBM2483
PNG
((4S)-6-chloro-4-(2-cyclopropylethynyl)-4-(trifluor...)
Show SMILES FC(F)(F)[C@]1(OC(=O)Nc2ccc(Cl)cc12)C#CC1CC1 |r|
Show InChI InChI=1S/C14H9ClF3NO2/c15-9-3-4-11-10(7-9)13(14(16,17)18,21-12(20)19-11)6-5-8-1-2-8/h3-4,7-8H,1-2H2,(H,19,20)/t13-/m0/s1
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n/an/a 22n/an/an/an/an/an/a



Volgograd State Medical University

Curated by ChEMBL


Assay Description
Inhibition of HIV1 recombinant wild type reverse transcriptase p66/p51 pre-incubated with compound before enzyme addition using poly(rA) template and...

Bioorg Med Chem 23: 1069-81 (2015)


Article DOI: 10.1016/j.bmc.2015.01.002
BindingDB Entry DOI: 10.7270/Q2RR20XW
More data for this
Ligand-Target Pair
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