Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Translocator protein (Rattus norvegicus (rat)) | BDBM50186098 (CHEMBL3822812) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186176 (CHEMBL3823275) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 2.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186171 (CHEMBL3823116) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 5.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50185956 (CHEMBL3824124) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186173 (CHEMBL3823482) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186196 (CHEMBL3823216) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 13 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186218 (CHEMBL3822930) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 14 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186177 (CHEMBL3823486) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186191 (CHEMBL3823161) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186170 (CHEMBL3822955) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 38 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186168 (CHEMBL3823157) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186189 (CHEMBL3823037) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 59 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186100 (CHEMBL3823703) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 88 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186179 (CHEMBL3824014) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 95 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186155 (CHEMBL3824260) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 127 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186099 (CHEMBL3824329) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 397 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-PK11195 from TSPO in rat C6 cell lysate after 2 hrs by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50185956 (CHEMBL3824124) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186099 (CHEMBL3824329) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186100 (CHEMBL3823703) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186155 (CHEMBL3824260) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186168 (CHEMBL3823157) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186098 (CHEMBL3822812) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186218 (CHEMBL3822930) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186196 (CHEMBL3823216) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186191 (CHEMBL3823161) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186189 (CHEMBL3823037) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186179 (CHEMBL3824014) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186177 (CHEMBL3823486) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186176 (CHEMBL3823275) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186170 (CHEMBL3822955) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186171 (CHEMBL3823116) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Translocator protein (Rattus norvegicus (rat)) | BDBM50186173 (CHEMBL3823482) | PDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Displacement of [3H]-flunitrazepam from TSPO in rat C6 cell lysate by liquid scintillation counting | Bioorg Med Chem Lett 26: 3472-7 (2016) Article DOI: 10.1016/j.bmcl.2016.06.041 BindingDB Entry DOI: 10.7270/Q2B27X7C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024253 (CHEMBL3334887) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 66 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024254 (CHEMBL125021) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024252 (CHEMBL1609104) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 140 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50278662 (CHEMBL4172540) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 245 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK293 cells co-expressing Galpha15 assessed as decrease in glutamate-induced calcium mobil... | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024255 (CHEMBL3334944) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 279 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024258 (CHEMBL3334941) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 336 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512690 (CHEMBL4451520) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 520 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024259 (CHEMBL3334940) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 646 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024260 (CHEMBL3334939) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 785 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Proteinase-activated receptor 4 (Homo sapiens (Human)) | BDBM50024257 (CHEMBL3334942) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 793 | n/a | n/a | n/a | n/a | n/a | n/a |
Northwest Agriculture& Forestry University Curated by ChEMBL | Assay Description Antagonist activity at PAR4 in PAR-4-AP-stimulated human platelets compound pretreated for 5 mins by fluorescent PAC1 integrin alpha2bb3 activation a... | Bioorg Med Chem Lett 24: 4708-13 (2014) Article DOI: 10.1016/j.bmcl.2014.08.021 BindingDB Entry DOI: 10.7270/Q29P336C | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512692 (CHEMBL4474204) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 920 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50278662 (CHEMBL4172540) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.28E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux preincuba... | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512694 (CHEMBL4554871) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512683 (CHEMBL4468538) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amino acid transporter (Rattus norvegicus) | BDBM50140134 (CHEMBL3753869) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512682 (CHEMBL4520808) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Metabotropic glutamate receptor 3 (Rattus norvegicus (Rat)) | BDBM50512698 (CHEMBL4572957) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Curated by ChEMBL | Assay Description Negative allosteric modulation of rat mGlu3R expressed in HEK cells harboring GIRK assessed as reduction in glutamate-induced thallium flux | Bioorg Med Chem Lett 29: 2670-2674 (2019) Article DOI: 10.1016/j.bmcl.2019.07.030 BindingDB Entry DOI: 10.7270/Q2KP85HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amino acid transporter (Rattus norvegicus) | BDBM50140131 (CHEMBL3752249) | UniProtKB/TrEMBL GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Vanderbilt University Medical Center Curated by ChEMBL | Assay Description Inhibition of ASCT2-mediated glutamine transport in rat C6 cells using [3H]-glutamine after 15 mins by scintillation counting | Bioorg Med Chem Lett 26: 1044-7 (2016) Article DOI: 10.1016/j.bmcl.2015.12.031 BindingDB Entry DOI: 10.7270/Q2MC91V1 | |||||||||||
More data for this Ligand-Target Pair |
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