Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Endothelin-1 receptor (Mus musculus) | BDBM50304494 (3-Benzo[1,3]dioxol-5-yl-4-[3-(2-bromoethoxy)-4,5-d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.240 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304495 (2-{4-[4-(Benzo[1,3]dioxol-5-yl)-2-hydroxy-5-oxo-3-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.360 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304496 (3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.09 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304496 (3-Benzo[1,3]dioxol-5-yl-4-[3-(2-fluoroethoxy)-4,5-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304497 (2-(5-{[4-(Benzo[1,3]dioxol-5-yl)-2-hydroxy-2-(4-me...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.26 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336694 (3-Benzo[1,3]dioxol-5-yl-4-{3-(2-(2-(2-(2-fluoroeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336695 (3-Benzo[1,3]dioxol-5-yl-4-{3-[1-(2-{2-[2-(2-fluoro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304498 (3-Benzo[1,3]dioxol-5-yl-5-[4-(2-fluoroethoxy)pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.43 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336697 (3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{4-[4-(2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336699 (CHEMBL1672884 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336696 (3-Benzo[1,3]dioxol-5-yl-4-[3-(2-{2-[2-(2-{1-[2-(2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336698 (CHEMBL1672885 | N-[1-(2-{2-[2-(2-{5-[4-Benzo[1,3]d...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50336700 (3-Benzo[1,3]dioxol-5-yl-4-{3-[2-(2-{2-[2-(4-fluoro...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital Mu£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from ETA receptor in CD1 Nu/Nu mouse myocardial ventricles membranes after 2 hrs by gamma counting | J Med Chem 54: 939-48 (2011) Article DOI: 10.1021/jm101110w BindingDB Entry DOI: 10.7270/Q2V69JW4 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50304499 (3-Benzo[1,3]dioxol-5-yl-5-hydroxy-5-[4-(2-bromoeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50034267 (3-(benzo[d][1,3]dioxol-5-yl)-5-hydroxy-5-(4-methox...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
University Hospital M£nster Curated by ChEMBL | Assay Description Displacement of [125I]ET1 from endothelin A receptor in DBA mouse microsomes | Bioorg Med Chem 17: 7197-208 (2009) Article DOI: 10.1016/j.bmc.2009.08.058 BindingDB Entry DOI: 10.7270/Q27S7NVF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281579 ((S)-3-{2-[((R)-2-Acetylamino-3-phenyl-propionyl)-b...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281576 ((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(1H-indol-3-yl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281577 ((S)-3-{(S)-2-[(R)-2-Acetylamino-3-(4-hydroxy-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 26 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281586 ((R)-3-{[(R)-1-((R)-2-Acetylamino-3-phenyl-propiony...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 45 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281580 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 57 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281581 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 70 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281582 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281575 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 77 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281585 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 79 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281587 ((S)-3-[(R)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281583 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 114 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281584 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description The compound was tested for the binding affinity against eEndothelin A receptor in murine 3T3 cells using [125I]-ET-1 as a radioligand | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281910 ((S)-3-[(S)-5-((S)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cells | Bioorg Med Chem Lett 3: 1253-1256 (1993) Article DOI: 10.1016/S0960-894X(00)80326-1 BindingDB Entry DOI: 10.7270/Q2ZC82S8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281911 ((R)-3-[(R)-5-((S)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cells | Bioorg Med Chem Lett 3: 1253-1256 (1993) Article DOI: 10.1016/S0960-894X(00)80326-1 BindingDB Entry DOI: 10.7270/Q2ZC82S8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281578 ((S)-3-[(S)-2-((R)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 270 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibition of [125I]-ET-1 binding to Endothelin A receptor of murine 3T3 cells | Bioorg Med Chem Lett 3: 519-524 (1993) Article DOI: 10.1016/S0960-894X(01)81219-1 BindingDB Entry DOI: 10.7270/Q27081C5 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Endothelin-1 receptor (Mus musculus) | BDBM50281912 ((S)-3-[(R)-5-((S)-2-Acetylamino-3-phenyl-propionyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article | n/a | n/a | 900 | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Binding affinity of the compound for Endothelin A receptor was determined in murine 3T3 cells | Bioorg Med Chem Lett 3: 1253-1256 (1993) Article DOI: 10.1016/S0960-894X(00)80326-1 BindingDB Entry DOI: 10.7270/Q2ZC82S8 | |||||||||||
More data for this Ligand-Target Pair |