Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM50009723![]() (2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Effect of Phosphatidylserine on inhibition of Protein kinase C alpha | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM2579![]() ((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PubMed | n/a | n/a | 2.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
cAMP-dependent protein kinase catalytic subunit alpha (Rattus norvegicus (rat)) | BDBM2579![]() ((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | PDB PubMed | n/a | n/a | 27 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of cAMP-dependent kinase PKA(Protein kinase A) catalytic subunit at 100 uM | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | ![]() 3D Structure (crystal) | ||||||||||||
cAMP-dependent protein kinase catalytic subunit alpha (Rattus norvegicus (rat)) | BDBM83205![]() ((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase MCE KEGG PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 98 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of cAMP-dependent kinase PKA(Protein kinase A) catalytic subunit at 100 uM | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM50009723![]() (2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Effect of PMA on inhibition of PKC alpha (Protein kinase C) | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha type (Rattus norvegicus (Rat)) | BDBM50009723![]() (2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...) | PDB MMDB Reactome pathway UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1.90E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Effect of PMA on inhibition of PKC alpha (Protein kinase C) | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50009723![]() (2,6-Diamino-hexanoic acid (1-tridecanoyl-piperidin...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229926![]() (CHEMBL319584) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229931![]() (CHEMBL100713) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229920![]() (CHEMBL101142) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229930![]() (CHEMBL97997) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase C | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229928![]() (CHEMBL97998) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase C | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229917![]() (CHEMBL100289) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229921![]() (CHEMBL99372) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | PubMed | n/a | n/a | 4.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229932![]() (CHEMBL97921) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229922![]() (CHEMBL98968) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of [3H]-phorbol dibutyrate binding to Protein kinase C alpha | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229924![]() (CHEMBL99156) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229929![]() (CHEMBL98337) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 5.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM83205![]() ((E,2S,3R)-2-amino-4-octadecene-1,3-diol | (E,2S,3R...) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | Purchase MCE KEGG PC cid PC sid PDB UniChem Similars | PubMed | n/a | n/a | 5.70E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229927![]() (CHEMBL319666) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 6.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229933![]() (CHEMBL98542) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229916![]() (CHEMBL322371) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 7.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229915![]() (CHEMBL101358) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 9.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229925![]() (CHEMBL433408) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.02E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229923![]() (CHEMBL317827) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.54E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description Inhibition of PMA and [Ca2+] induced 32P incorporation into histones by partially purified rat brain Protein kinase C | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229919![]() (CHEMBL101538) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 1.59E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Protein kinase C alpha/beta/gamma type (Rattus norvegicus (Rat)-Rattus norvegicus (rat)) | BDBM50229918![]() (CHEMBL101731) | PDB UniProtKB/SwissProt GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.99E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Nova Pharmaceutical Corporation Curated by ChEMBL | Assay Description In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat... | J Med Chem 34: 2928-31 (1991) BindingDB Entry DOI: 10.7270/Q2KH0NZG | |||||||||||
More data for this Ligand-Target Pair |