Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394450 (2-(6-amino-5-(8-(5- | US10308614, Example 51) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394468 (2-(6-amino-5-(8- | US10308614, Example 69) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394474 (2-(6-amino-5-(8-(5- | US10308614, Example 75) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394469 (2-(6-amino-5-(8-(pyridin- | US10308614, Example 70) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.10 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394462 (2-(6-amino-5-(8-phenyl-3,8- | US10308614, Example ...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394446 (2-(6-amino-5-(8-(2- | US10308614, Example 47) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase PC cid PC sid UniChem | US Patent | n/a | n/a | 4.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394470 (2-(6-amino-5-(8- | US10308614, Example 71) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469320 (CHEMBL4293567) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469331 (CHEMBL4282980) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469324 (CHEMBL4286345) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469330 (CHEMBL4295096) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem | Article PubMed | n/a | n/a | <5 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469329 (CHEMBL4278436) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394589 (2-(6-amino-5-(1-(1- | US10308614, Example 192) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394476 (2-(6-amino-5-(8-(thiazol- | US10308614, Example 77) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394585 (2-(6-amino-5-(1-(1- | US10308614, Example 188) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.60 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394475 (2-(6-amino-5-(8-(4- | US10308614, Example 76) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 6.70 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394427 ((trans-4a,8a)-2-(3-amino-6- | US10308614, Example ...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 (Homo sapiens (Human)) | BDBM50469325 (CHEMBL4294655) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 10 | n/a | n/a | n/a | n/a | n/a | n/a |
Novartis Institutes for Biomedical Research Curated by ChEMBL | Assay Description Inhibition of recombinant His6-tagged BRG1 ATPase-SnAC (658 to 1361 residues) (unknown origin) expressed in insect sf9 cells preincubated for 5 mins ... | J Med Chem 61: 10155-10172 (2018) Article DOI: 10.1021/acs.jmedchem.8b01318 BindingDB Entry DOI: 10.7270/Q2TH8QDB | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394528 (1-(4-(3-amino-6-(2- | US10308614, Example 129) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394449 (2-(6-amino-5-(8- | US10308614, Example 50) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394473 (2-(6-amino-5-((1R,4R)-5- | US10308614, Example 74) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 10.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394485 (Enantiomer 1 and Enantiomer 2 of (trans-4a,8a)-2-(...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394441 (1-(3-amino-6-(2- | US10308614, Example 42) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394461 ((4-(3-amino-6-(2- | US10308614, Example 62) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 11.7 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394595 (2-(6-amino-5-(trans-2-phenylcyclopropyl)pyridazin-...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12.1 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394575 (2-(6-amino-5-(2- | US10308614, Example 178) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12.2 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394537 ((4-(3-amino-6-(2- | US10308614, Example 138) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394584 (2-(6-amino-5-(1-methyl- | US10308614, Example 187) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 12.8 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394605 (2-(6-amino-5-cyclohexylpyridazin-3-yl)phenol | US1...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394571 (2-(6-amino-5- | US10308614, Example 174) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 14.8 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394458 (1-(3-amino-6-(2- | US10308614, Example 59) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 15.8 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394427 ((trans-4a,8a)-2-(3-amino-6- | US10308614, Example ...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.2 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394580 (2-(6-amino-5-((1- | US10308614, Example 183) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.2 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394424 (2-(6-amino-5-(4-methyl- | US10308614, Example 25) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394587 (2-(6-amino-5- | US10308614, Example 190) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394508 (2-(6-amino-5-(3-methyl- | US10308614, Example 109) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394456 (2-(6-amino-5-(3- | US10308614, Example 57) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 17.7 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394492 ((S)-2-(6-amino-5-(3-methyl-4-((1-methyl-1H-imidazo...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 18.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394621 (2-(6-amino-5-((1,4-trans)-4-methylcyclohexyl)pyrid...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394481 (Enantiomer 1 and Enantiomer 2 of 2-(6-amino-5-(4-(...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19.1 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394442 (2-(6-amino-5-(8- | US10308614, Example 43) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19.3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394510 (2-(6-amino-5-(4- | US10308614, Example 111) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 19.7 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394525 ((3-(3-amino-6-(2- | US10308614, Example 126) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.3 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394619 (2-(6-amino-5-(1-benzyl-1,2,3,6-tetrahydropyridin-4...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.5 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394542 ((4-(3-amino-6-(2- | US10308614, Example 143) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.6 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394430 (1-(3-amino-6-(2- | US10308614, Example 31) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.8 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394622 (2-(6-amino-5-((1,4-trans)-4-methylcyclohexyl)pyrid...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.9 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394414 (2-(6-amino-5-(4-(1- | US10308614, Example 15) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 20.9 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394399 (US10308614, Example 1 | tert-butyl 4-(3-amino-6-(2...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid PDB UniChem | US Patent | n/a | n/a | 21.4 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcription activator BRG1 [1448-1575] (Homo sapiens (Human)) | BDBM394592 ((2R)-2-[4-[3-amino- 6-(2- hydroxyphenyl) pyridazin...) | PDB MMDB KEGG UniProtKB/SwissProt GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | n/a | n/a | 21.7 | n/a | n/a | n/a | n/a | n/a | n/a |
The Institute of Cancer Research | Assay Description His-BRG1 (A1448-S1575; Swiss Prot P51532; mhhhhhhgslvpr\gsAEKLSPNPP NLTKKMKKIVDAVIKYKDSSSGRQLSEVFIQLPSRKELPEYYELIRKPVDFKKIKERIRNH KYRSLNDLEKDVMLLCQNA... | J Med Chem 52: 2255-64 (2009) BindingDB Entry DOI: 10.7270/Q26112NJ | |||||||||||
More data for this Ligand-Target Pair |
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