Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Calmodulin-1 (Human) | BDBM50346822 (CHEMBL66917) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.38E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50001888 ((chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL DrugBank MCE KEGG MMDB PC cid PC sid PDB UniChem Patents Similars | Article PubMed | n/a | n/a | 1.03E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346811 (CHEMBL1796022) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 1.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346820 (CHEMBL1796013) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.84E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346810 (CHEMBL268559) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346806 (CHEMBL1796026) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.29E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346819 (CHEMBL1796014) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346821 (CHEMBL1796012) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.13E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346805 (CHEMBL1796027) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.25E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346818 (CHEMBL1796015) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.63E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346809 (CHEMBL1796023) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.77E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346815 (CHEMBL1796017) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.61E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346814 (CHEMBL1796018) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.47E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346812 (CHEMBL1796021) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.47E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346813 (CHEMBL1796020) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.62E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346808 (CHEMBL1796024) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.73E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346807 (CHEMBL1796025) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.27E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346817 (CHEMBL1796016) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.59E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346823 (GIGANTOL) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.14E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Calmodulin-1 (Human) | BDBM50346816 (CHEMBL467338) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.46E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
Universidad Nacional Aut£noma de M£xico Curated by ChEMBL | Assay Description Inhibition of Calmodulin-dependent PDE1 activity assessed as inorganic phosphate release after 30 min | Eur J Med Chem 46: 2699-708 (2011) Article DOI: 10.1016/j.ejmech.2011.03.057 BindingDB Entry DOI: 10.7270/Q2MW2HGD | |||||||||||
More data for this Ligand-Target Pair |