Affinity Data by PubMed id=16603348

PubMed code 16603348

Found 12 hits of Enzyme Inhibition Constant Data
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50185156 (CHEMBL210439 \| Hmb-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50185159 (CHEMBL208162 \| Hmb-Phe-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	32	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50185155 (CHEMBL207774 \| H-Phe-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	42	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50370717 (EPOXOMYCIN \| Epoxomicin) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	47	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50185157 (CHEMBL210901 \| benzyl (S)-4-methyl-1-((S)-4-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	61	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50185158 (CHEMBL210091 \| H-Tyr-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	83	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50370717 (EPOXOMYCIN \| Epoxomicin) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	Purchase PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	980	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50185159 (CHEMBL208162 \| Hmb-Phe-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.23E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-2 (Homo sapiens (Human))	BDBM50185157 (CHEMBL210901 \| benzyl (S)-4-methyl-1-((S)-4-methyl...) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	2.43E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of trypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50185155 (CHEMBL207774 \| H-Phe-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.15E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50185158 (CHEMBL210091 \| H-Tyr-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	4.32E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair
Proteasome subunit beta type-5 (Homo sapiens (Human))	BDBM50185156 (CHEMBL210439 \| Hmb-Val-Gln-Leu-VE) Show SMILES Show InChI	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	Article PubMed	n/a	n/a	6.67E+3	n/a	n/a	n/a	n/a	n/a	n/a
University of Ferrara Curated by ChEMBL					Assay Description Inhibition of chymotrypsin like activity of proteasome				Bioorg Med Chem Lett 16: 3125-30 (2006) Article DOI: 10.1016/j.bmcl.2006.03.070 BindingDB Entry DOI: 10.7270/Q2TX3G5J
University of Ferrara Curated by ChEMBL					More data for this Ligand-Target Pair

* indicates data uncertainty>20%