| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
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| Ligand | BDBM50259839 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_2298857 |
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| EC50 | 3.0±n/a nM |
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| Citation |  Wei, L; Xiang, K; Kang, H; Yu, Y; Fan, H; Zhou, H; Hou, T; Ge, Y; Wang, J; Guo, Z; Chen, Y; Zhao, Y; Liang, X Development and Characterization of Fluorescent Probes for the G Protein-Coupled Receptor 35. ACS Med Chem Lett14:411-416 (2023) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 35 |
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| Name: | G-protein coupled receptor 35 |
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| Synonyms: | G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 34085.57 |
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| Organism: | Homo sapiens (Human) |
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| Description: | gi_33695097 |
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| Residue: | 309 |
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| Sequence: | MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
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| BDBM50259839 |
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| n/a |
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| Name | BDBM50259839 |
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| Synonyms: | CHEMBL4100677 |
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| Type | Small organic molecule |
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| Emp. Form. | C10H4BrN5O5 |
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| Mol. Mass. | 354.073 |
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| SMILES | Oc1c(Br)cc2cc(-c3nnn[nH]3)c(=O)oc2c1[N+]([O-])=O |
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| Structure | 
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