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TargetNuclear receptor subfamily 4 group A member 1
LigandBDBM50378798
Substrate/Competitorn/a
Meas. Tech.ChEMBL_650684 (CHEMBL1227264)
Kd 1510±n/a nM
Citation Zhan, YDu, XChen, HLiu, JZhao, BHuang, DLi, GXu, QZhang, MWeimer, BCChen, DCheng, ZZhang, LLi, QLi, SZheng, ZSong, SHuang, YYe, ZSu, WLin, SCShen, YWu, Q Cytosporone B is an agonist for nuclear orphan receptor Nur77. Nat Chem Biol4:548-56 (2008) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Nuclear receptor subfamily 4 group A member 1
Name:Nuclear receptor subfamily 4 group A member 1
Synonyms:GFRP1 | HMR | NAK1 | NR4A1 | NR4A1_HUMAN | nuclear receptor subfamily 4, group A, member 1
Type:Enzyme Catalytic Domain
Mol. Mass.:64467.13
Organism:Homo sapiens (Human)
Description:gi_27894344
Residue:598
Sequence:
MPCIQAQYGTPAPSPGPRDHLASDPLTPEFIKPTMDLASPEAAPAAPTALPSFSTFMDGY
TGEFDTFLYQLPGTVQPCSSASSSASSTSSSSATSPASASFKFEDFQVYGCYPGPLSGPV
DEALSSSGSDYYGSPCSAPSPSTPSFQPPQLSPWDGSFGHFSPSQTYEGLRAWTEQLPKA
SGPPQPPAFFSFSPPTGPSPSLAQSPLKLFPSQATHQLGEGESYSMPTAFPGLAPTSPHL
EGSGILDTPVTSTKARSGAPGGSEGRCAVCGDNASCQHYGVRTCEGCKGFFKRTVQKNAK
YICLANKDCPVDKRRRNRCQFCRFQKCLAVGMVKEVVRTDSLKGRRGRLPSKPKQPPDAS
PANLLTSLVRAHLDSGPSTAKLDYSKFQELVLPHFGKEDAGDVQQFYDLLSGSLEVIRKW
AEKIPGFAELSPADQDLLLESAFLELFILRLAYRSKPGEGKLIFCSGLVLHRLQCARGFG
DWIDSILAFSRSLHSLLVDVPAFACLSALVLITDRHGLQEPRRVEELQNRIASCLKEHVA
AVAGEPQPASCLSRLLGKLPELRTLCTQGLQRIFYLKLEDLVPPPPIIDKIFMDTLPF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50378798
n/a
NameBDBM50378798
Synonyms:CYTOSPORONE B
TypeSmall organic molecule
Emp. Form.C18H26O5
Mol. Mass.322.396
SMILESCCCCCCCC(=O)c1c(O)cc(O)cc1CC(=O)OCC
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: