The following articles (labelled with PubMed ID or TBD) are for your review
| PMID | Data | Article Title | Organization |
|---|
| 28107736 |
53 |
Crystal structures, binding interactions, and ADME evaluation of brain penetrant N-substituted indazole-5-carboxamides as subnanomolar, selective monoamine oxidase B and dual MAO-A/B inhibitors. |
Ntz Lab |
| 3968682 |
20 |
Enzyme-activated irreversible inhibitors of monoamine oxidase: phenylallylamine structure-activity relationships. |
TBA |
| 6864731 |
38 |
Synthesis and monoamine oxidase inhibitory activities of alpha-allenic amines in vivo and in vitro. Different activities of two enantiomeric allenes. |
TBA |
| 27692996 |
84 |
Neuroprotective effects of benzyloxy substituted small molecule monoamine oxidase B inhibitors in Parkinson's disease. |
China Pharmaceutical University |
| 27578245 |
46 |
2-Benzylidene-1-indanone derivatives as inhibitors of monoamine oxidase. |
North-West University |
| 26652247 |
60 |
3-(Piperidin-4-ylmethoxy)pyridine Containing Compounds Are Potent Inhibitors of Lysine Specific Demethylase 1. |
Baylor College of Medicine |
| 26107513 |
172 |
Structure-Based Design and Optimization of Multitarget-Directed 2H-Chromen-2-one Derivatives as Potent Inhibitors of Monoamine Oxidase B and Cholinesterases. |
Universit£ |
| 25466194 |
34 |
a-Ketoamino acid ester derivatives as promising MAO inhibitors. |
King Saud University |
| 25627172 |
150 |
Novel arylalkenylpropargylamines as neuroprotective, potent, and selective monoamine oxidase B inhibitors for the treatment of Parkinson's disease. |
A* Star |
| 25418133 |
51 |
N-Methyl-N-((1-methyl-5-(3-(1-(2-methylbenzyl)piperidin-4-yl)propoxy)-1H-indol-2-yl)methyl)prop-2-yn-1-amine, a new cholinesterase and monoamine oxidase dual inhibitor. |
Laboratorio De Quimica Medica (Iqog, Csic) |
| 25600407 |
26 |
Reversible and irreversible small molecule inhibitors of monoamine oxidase B (MAO-B) investigated by biophysical techniques. |
Dart Neuroscience |
| 24955776 |
166 |
Indazole- and indole-5-carboxamides: selective and reversible monoamine oxidase B inhibitors with subnanomolar potency. |
University of Bonn |
| 25462230 |
80 |
In silico design of novel 2H-chromen-2-one derivatives as potent and selective MAO-B inhibitors. |
Universit£ |
| 24813882 |
41 |
Donepezil + propargylamine + 8-hydroxyquinoline hybrids as new multifunctional metal-chelators, ChE and MAO inhibitors for the potential treatment of Alzheimer's disease. |
Okayama University |
| 23353756 |
23 |
Synthesis, pharmacological evaluation and QSAR modeling of mono-substituted 4-phenylpiperidines and 4-phenylpiperazines. |
Neurosearch Sweden |
| 23437843 |
30 |
Discovery, biological evaluation, and structure-activity and -selectivity relationships of 6'-substituted (E)-2-(benzofuran-3(2H)-ylidene)-N-methylacetamides, a novel class of potent and selective monoamine oxidase inhibitors. |
Universit£ |
| 16884303 |
27 |
Structural insights into monoamine oxidase inhibitory potency and selectivity of 7-substituted coumarins from ligand- and target-based approaches. |
Universit£ |
| 11543689 |
34 |
Coumarins derivatives as dual inhibitors of acetylcholinesterase and monoamine oxidase. |
Universit£ |
| 11123983 |
112 |
Inhibition of monoamine oxidases by functionalized coumarin derivatives: biological activities, QSARs, and 3D-QSARs. |
Universit£ |
| 23043306 |
69 |
Systematic in vivo screening of a series of 1-propyl-4-arylpiperidines against dopaminergic and serotonergic properties in rat brain: a scaffold-jumping approach. |
Neurosearch Sweden |
| 22385498 |
24 |
Synthesis and evaluation of a set of para-substituted 4-phenylpiperidines and 4-phenylpiperazines as monoamine oxidase (MAO) inhibitors. |
Neurosearch Sweden |
| 22282722 |
10 |
Molecular Insights into Human Monoamine Oxidase B Inhibition by the Glitazone Anti-Diabetes Drugs. |
TBA |
| 22503231 |
66 |
Multipotent MAO and cholinesterase inhibitors for the treatment of Alzheimer's disease: synthesis, pharmacological analysis and molecular modeling of heterocyclic substituted alkyl and cycloalkyl propargyl amine. |
Laboratorio De Radicales Libres Y Qu�Mica Computacional (Iqog, Csic) |
| 22475561 |
42 |
Synthesis and inhibitory effect of piperine derivates on monoamine oxidase. |
General Hospital of Pla |
| 20123154 |
48 |
2-Arylthiomorpholine derivatives as potent and selective monoamine oxidase B inhibitors. |
University of Chile |
| 19243954 |
36 |
Naphthylisopropylamine and N-benzylamphetamine derivatives as monoamine oxidase inhibitors. |
University of Chile |
| 17611112 |
36 |
A new therapeutic approach in Alzheimer disease: some novel pyrazole derivatives as dual MAO-B inhibitors and antiinflammatory analgesics. |
Hacettepe University |
| 15689151 |
112 |
Alkylamino derivatives of 4-aminomethylpyridine as inhibitors of copper-containing amine oxidases. |
Universit£ |
| 9258353 |
45 |
Selective inhibitors of monoamine oxidase. 4. SAR of tricyclic N-methylcarboxamides and congeners binding at the tricyclics' hydrophilic binding site. |
Wellcome Research Laboratories |
| 8487255 |
84 |
5-[4-(benzyloxy)phenyl]-1,3,4-oxadiazol-2(3H)-one derivatives and related analogues: new reversible, highly potent, and selective monamine oxidase type B inhibitors. |
Universit£ |
| 1433183 |
32 |
Aliphatic propargylamines: potent, selective, irreversible monoamine oxidase B inhibitors. |
University of Saskatchewan |
| 7200144 |
2 |
(+/-)-4-Aryl-4,5-dihydro-3H-1,3-benzodiazepines. 1. Synthesis and evaluation of (+/-)-4,5-dihydro-2,3-dimethyl-4-phenyl-3H-1,3-benzodiazepine and analogues as potential antidepressant agents. |
TBA |
| | 51 |
Synthesis of coumarins as subtype-selective inhibitors of monoamine oxidase |
TBA |
| 22023459 |
42 |
Synthesis, biological evaluation, and molecular modeling of donepezil and N-[(5-(benzyloxy)-1-methyl-1H-indol-2-yl)methyl]-N-methylprop-2-yn-1-amine hybrids as new multipotent cholinesterase/monoamine oxidase inhibitors for the treatment of Alzheimer's disease. |
Universitat Aut£Noma De Barcelona |
| 21377879 |
44 |
Development of selective and reversible pyrazoline based MAO-B inhibitors: virtual screening, synthesis and biological evaluation. |
Birla Institute of Technology |
| 20117937 |
56 |
Design of novel nicotinamides as potent and selective monoamine oxidase a inhibitors. |
Nanjing University |
| 19969454 |
7 |
Proposed structural basis of interaction of piperine and related compounds with monoamine oxidases. |
University of Cambridge |
| 19945874 |
24 |
Towards development of selective and reversible pyrazoline based MAO-inhibitors: Synthesis, biological evaluation and docking studies. |
Institute of Technology |
| 19682910 |
48 |
Synthesis and molecular modeling of some novel hexahydroindazole derivatives as potent monoamine oxidase inhibitors. |
Hacettepe University |
| 19810674 |
93 |
Discovery of a novel class of potent coumarin monoamine oxidase B inhibitors: development and biopharmacological profiling of 7-[(3-chlorobenzyl)oxy]-4-[(methylamino)methyl]-2H-chromen-2-one methanesulfonate (NW-1772) as a highly potent, selective, reversible, and orally active monoamine oxidase B |
Universita Degli Studi Di Bari |
| 19091581 |
128 |
New pyrazoline bearing 4(3H)-quinazolinone inhibitors of monoamine oxidase: synthesis, biological evaluation, and structural determinants of MAO-A and MAO-B selectivity. |
Hacettepe University |
| 19064321 |
37 |
Ultrasound promoted synthesis of 2-imidazolines in water: a greener approach toward monoamine oxidase inhibitors. |
Universidade Federal De Santa Maria |
| 18980841 |
72 |
Pyrazoline-based mycobactin analogues as MAO-inhibitors. |
Institute of Technology |
| 17824599 |
39 |
Solid-phase synthesis and insights into structure-activity relationships of safinamide analogues as potent and selective inhibitors of type B monoamine oxidase. |
University of Bari |
| 17521909 |
15 |
Human and rat monoamine oxidase-A are differentially inhibited by (S)-4-alkylthioamphetamine derivatives: insights from molecular modeling studies. |
University of Santiago De Chile |
| 16942031 |
4 |
3-[5-(4,5-dihydro-1H-imidazol-2-yl)-furan-2-yl]phenylamine (Amifuraline), a promising reversible and selective peripheral MAO-A inhibitor. |
Università |
| 16759116 |
8 |
Synthesis, structural reassignment, and biological activity of type B MAO inhibitors based on the 5H-indeno[1,2-c]pyridazin-5-one core. |
FacultéS Universitaires N.D. De La Paix |
| 16356714 |
16 |
Synthesis of 3-benzyl-2-substituted quinoxalines as novel monoamine oxidase A inhibitors. |
University of Alexandria |
| 15974574 |
56 |
Design, synthesis, and biological activities of pyrrolylethanoneamine derivatives, a novel class of monoamine oxidases inhibitors. |
Sapienza University of Rome |
| 15801832 |
38 |
Sulfur-substituted alpha-alkyl phenethylamines as selective and reversible MAO-A inhibitors: biological activities, CoMFA analysis, and active site modeling. |
Universidad De Chile |
| 15189042 |
24 |
Novel pyridazino[4,3-b]indoles with dual inhibitory activity against Mycobacterium tuberculosis and monoamine oxidase. |
Russian Academy of Sciences |
| 11591508 |
18 |
Synthesis of N-propargylphenelzine and analogues as neuroprotective agents. |
Cv Technologies |
| 32031378 |
17 |
Acetylene Group, Friend or Foe in Medicinal Chemistry. |
St. John'S University |
| 31864798 |
42 |
Propargylamine-derived multi-target directed ligands for Alzheimer's disease therapy. |
Universidade De Lisboa |
| 30920216 |
6 |
Bioactive Dimeric Acylphloroglucinols from the Mexican Fern Elaphoglossum paleaceum. |
Universidad Aut£Noma Del Estado De Morelos |
| 27575476 |
30 |
Potent selective monoamine oxidase B inhibition by maackiain, a pterocarpan from the roots of Sophora flavescens. |
Sunchon National University |
| 10794685 |
42 |
Molecular determinants of MAO selectivity in a series of indolylmethylamine derivatives: biological activities, 3D-QSAR/CoMFA analysis, and computational simulation of ligand recognition. |
Universitat AutòNoma De Barcelona |
| 30686752 |
35 |
Osthenol, a prenylated coumarin, as a monoamine oxidase A inhibitor with high selectivity. |
Sunchon National University |
| 30522087 |
63 |
(Pyrrolo-pyridin-5-yl)benzamides: BBB permeable monoamine oxidase B inhibitors with neuroprotective effect on cortical neurons. |
Ntz Lab |
| 31185168 |
144 |
Functionalized 6-(Piperidin-1-yl)-8,9-Diphenyl Purines as Peripherally Restricted Inverse Agonists of the CB1 Receptor. |
Rti International |
| 31103902 |
41 |
Multi-target design strategies for the improved treatment of Alzheimer's disease. |
China Pharmaceutical University |
| 9748356 |
28 |
Inhibition of monoamine oxidase-B by condensed pyridazines and pyrimidines: effects of lipophilicity and structure-activity relationships. |
Université |
| 30744931 |
170 |
Anti-cholinesterase hybrids as multi-target-directed ligands against Alzheimer's disease (1998-2018). |
Csir-Central Drug Research Institute |
| 9622553 |
42 |
Selective inhibitors of monoamine oxidase (MAO). 5. 1-Substituted phenoxathiin inhibitors containing no nitrogen that inhibit MAO A by binding it to a hydrophobic site. |
The Wellcome Research Laboratories |
| 31082225 |
26 |
Rational Design of Multitarget-Directed Ligands: Strategies and Emerging Paradigms. |
China Pharmaceutical University |
| 8627609 |
51 |
Selective inhibitors of monoamine oxidase. 3. Structure-activity relationship of tricyclics bearing imidazoline, oxadiazole, or tetrazole groups. |
Wellcome Research Laboratories |
| 24231308 |
80 |
Fine molecular tuning at position 4 of 2H-chromen-2-one derivatives in the search of potent and selective monoamine oxidase B inhibitors. |
Universit£ |
| 24012182 |
28 |
Inhibition of monoamine oxidase by 3,4-dihydro-2(1H)-quinolinone derivatives. |
North-West University |
| 8027990 |
25 |
Selective inhibitors of monoamine oxidase. 2. Arylamide SAR. |
Burroughs Wellcome |
| 23860591 |
38 |
Selected furanochalcones as inhibitors of monoamine oxidase. |
North-West University |
| 23374869 |
49 |
Inhibition of monoamine oxidase by phthalide analogues. |
North-West University |
| 7562919 |
132 |
Inhibition of monoamine oxidase-B by 5H-indeno[1,2-c]pyridazines: biological activities, quantitative structure-activity relationships (QSARs) and 3D-QSARs. |
Université |
| 7490728 |
87 |
Selective and potent monoamine oxidase type B inhibitors: 2-substituted 5-aryltetrazole derivatives. |
Université |
| 30243151 |
23 |
Donepezil-based multi-functional cholinesterase inhibitors for treatment of Alzheimer's disease. |
China Pharmaceutical University |
| 3735309 |
50 |
Selective monoamine oxidase inhibitors. 3. Cyclic compounds related to 4-aminophenethylamine. Preparation and neuron-selective action of some 5-(2-aminoethyl)-2,3-dihydroindoles. |
TBA |
| 30143367 |
38 |
Design, synthesis and biological evaluation of lazabemide derivatives as inhibitors of monoamine oxidase. |
Hainan Normal University |
| 29126721 |
81 |
Synthesis, monoamine oxidase inhibition activity and molecular docking studies of novel 4-hydroxy-N'-[benzylidene or 1-phenylethylidene]-2-H/methyl/benzyl-1,2-benzothiazine-3-carbohydrazide 1,1-dioxides. |
Government College University |
| 1895310 |
9 |
A selective, reversible, competitive inhibitor of monoamine oxidase A containing no nitrogen, with negligible potentiation of tyramine-induced blood pressure rise. |
Burroughs Wellcome |
| 27855360 |
23 |
Benzyloxynitrostyrene analogues - A novel class of selective and highly potent inhibitors of monoamine oxidase B. |
North-West University |
| 14709324 |
20 |
Pharmacological profile of YM348, a novel, potent and orally active 5-HT2C receptor agonist. |
Yamanouchi Pharmaceutical |
| 17373783 |
62 |
Discovery, synthesis, and in vivo activity of a new class of pyrazoloquinazolines as selective inhibitors of aurora B kinase. |
Astrazeneca |
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