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20 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDDataArticle TitleOrganization
28105277 33 Design and Synthesis of Novel Meta-Linked Phenylglycine Macrocyclic FVIIa Inhibitors.EBI Bristol-Myers Squibb
27994741 48 Discovery of Phenylglycine Lactams as Potent Neutral Factor VIIa Inhibitors.EBI Bristol-Myers Squibb R & D
27612545 37 Synthesis and P1' SAR exploration of potent macrocyclic tissue factor-factor VIIa inhibitors.EBI Bristol-Myers Squibb Research & Development
27455395 66 Discovery of a Highly Potent, Selective, and Orally Bioavailable Macrocyclic Inhibitor of Blood Coagulation Factor VIIa-Tissue Factor Complex.EBI Bristol-Myers Squibb R & D
27015008 51 Atropisomer Control in Macrocyclic Factor VIIa Inhibitors.EBI Bristol-Myers Squibb Research & Development
26200936 39 Applications of Fluorine in Medicinal Chemistry.EBI Bristol-Myers Squibb Research and Development
26151189 56 Structure-Based Design of Macrocyclic Coagulation Factor VIIa Inhibitors.EBI TBA
23845220 53 Nonbenzamidine acylsulfonamide tissue factor-factor VIIa inhibitors.EBI Bristol-Myers Squibb R & D
16289811 56 The discovery of fluoropyridine-based inhibitors of the factor VIIa/TF complex--Part 2.EBI Pfizer
19483697 23 Phage-encoded combinatorial chemical libraries based on bicyclic peptides.EBI Laboratory of Molecular Biology, Medical Research Council
20650636 118 Discovery of a factor Xa inhibitor (3R,4R)-1-(2,2-difluoro-ethyl)-pyrrolidine-3,4-dicarboxylic acid 3-[(5-chloro-pyridin-2-yl)-amide] 4-[[2-fluoro-4-(2-oxo-2H-pyridin-1-yl)-phenyl]-amide] as a clinical candidate.EBI F. Hoffmann-La Roche
17064913 29 Design, synthesis and biological activity of selective and orally available TF/FVIIa complex inhibitors containing non-amidine P1 ligands.EBI Astellas Pharma
16793264 13 Potent 4-amino-5-azaindole factor VIIa inhibitors.EBI Celera Genomics
16455251 11 Factor VIIa inhibitors: improved pharmacokinetic parameters.EBI Celera Genomics
16412633 9 Factor VIIa inhibitors: chemical optimization, preclinical pharmacokinetics, pharmacodynamics, and efficacy in an arterial baboon thrombosis model.EBI Celera Genomics
16125385 55 The discovery of fluoropyridine-based inhibitors of the Factor VIIa/TF complex.EBI Pfizer
11527709 19 Optimization of a screening lead for factor VIIa/TF.EBI Axys Pharmaceuticals
25764119 15 Discovery of novel P1 groups for coagulation factor VIIa inhibition using fragment-based screening.EBI Bristol-Myers Squibb
29072911 16 Design of Small-Molecule Active-Site Inhibitors of the S1A Family Proteases as Procoagulant and Anticoagulant Drugs.EBI University of Nottingham
29407959 82 The selectivity and bioavailability improvement of novel oral anticoagulants: An overview.EBI Hefei University of Technology