Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Cysteine protease (Trypanosoma brucei rhodesiense) | BDBM50505323![]() (CHEMBL4556848) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei rhodesiense rhodesain | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteine protease (Trypanosoma brucei rhodesiense) | BDBM50505321![]() (CHEMBL2402091) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Inhibition of Trypanosoma brucei rhodesiense rhodesain | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50396164![]() (CHEMBL2171751) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 8 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of human KLK1 using Pro-Phe-Arg-MCA as substrate for 2 mins by spectrophotometric analysis | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Procathepsin L (Homo sapiens (Human)) | BDBM50505321![]() (CHEMBL2402091) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 33 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Inhibition of human cathepsin L | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112584![]() (2-(2-{2-[2-(2-{2-[2-(2-Amino-3-methyl-pentanoylami...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50396166![]() (CHEMBL2171749) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of human KLK1 | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostate-specific antigen (Homo sapiens (Human)) | BDBM50298759![]() ((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of human KLK3 using Mu-SRKSQQY-AMC as substrate by fluorometric analysis | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Procathepsin L (Homo sapiens (Human)) | BDBM50229129![]() (4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 80 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Irreversible inhibition of human cathepsin L | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50370072![]() (CHEMBL1790422) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50396165![]() (CHEMBL2171750) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of human KLK1 | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112580![]() (CHEMBL268148 | PWGF(CH2NH)WWFW) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cruzipain (Trypanosoma cruzi) | BDBM50229129![]() (4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...) | PDB MMDB UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 220 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Irreversible inhibition of Trypanosoma cruzi cruzipain | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cysteine protease (Trypanosoma brucei rhodesiense) | BDBM50229129![]() (4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 270 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Irreversible inhibition of Trypanosoma brucei rhodesiense rhodesain | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446220![]() (CHEMBL3109164) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostate-specific antigen (Homo sapiens (Human)) | BDBM50396162![]() (CHEMBL2171878) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 300 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of KLK3 | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cathepsin B (Homo sapiens (Human)) | BDBM50229129![]() (4-Methyl-piperazine-1-carboxylic acid [(S)-1-((E)-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 390 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Irreversible inhibition of human cathepsin B | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446221![]() (CHEMBL3109163) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112597![]() (2-{2-[2-(2-{2-[2-[2-(2-Amino-3-carboxy-propionylam...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Prostate-specific antigen (Homo sapiens (Human)) | BDBM50396161![]() (CHEMBL2171879) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of KLK3 | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112581![]() (6-Amino-2-(2-{2-[2-(6-amino-2-{2-[6-amino-2-(2-ami...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446218![]() (CHEMBL3109166) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Procathepsin L (Homo sapiens (Human)) | BDBM50505323![]() (CHEMBL4556848) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | PC cid PC sid UniChem | Article PubMed | 690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of S£o Paulo Curated by ChEMBL | Assay Description Inhibition of human cathepsin L | J Med Chem 62: 10497-10525 (2019) Article DOI: 10.1021/acs.jmedchem.9b00683 BindingDB Entry DOI: 10.7270/Q2K93BT1 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446219![]() (CHEMBL3109165) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112596![]() (6-Amino-2-{2-[2-(2-{2-[2-[6-amino-2-(2-amino-3-car...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112594![]() (CHEMBL266692 | ChaALF(CH2NH)YMYY) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446218![]() (CHEMBL3109166) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446219![]() (CHEMBL3109165) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-2 (Homo sapiens (Human)) | BDBM50396163![]() (CHEMBL2171880) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | 1.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universit£ degli Studi di Napoli Federico II Curated by ChEMBL | Assay Description Inhibition of human KLK2 after 1 hr by phage-display based Immunofluorometric Assay | J Med Chem 55: 6669-86 (2012) Article DOI: 10.1021/jm300407t BindingDB Entry DOI: 10.7270/Q2N017N9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-2 (Homo sapiens (Human)) | BDBM50292533![]() (CHEMBL446790 | Fukugetin) | PDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Mixed-type inhibition of human tissue kallikrein-2 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446228![]() (CHEMBL3109061) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446227![]() (CHEMBL3109056) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391075![]() (CHEMBL2087343) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446220![]() (CHEMBL3109164) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446224![]() (CHEMBL3109160) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446211![]() (CHEMBL3109058) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446228![]() (CHEMBL3109061) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446224![]() (CHEMBL3109160) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446221![]() (CHEMBL3109163) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446211![]() (CHEMBL3109058) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50391078![]() (CHEMBL2087346) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do Tri£ngulo Mineiro Curated by ChEMBL | Assay Description Competitive inhibition of recombinant human KLK7 expressed in insect cell/baculovirus using Abz-KLYSSKQ-EDDnp as substrate by Dixon plot analysis | Bioorg Med Chem Lett 22: 6072-5 (2012) Article DOI: 10.1016/j.bmcl.2012.08.047 BindingDB Entry DOI: 10.7270/Q2SF2X8R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-5 [D153N] (Homo sapiens (Human)) | BDBM50446229![]() (CHEMBL3109060) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-1 (Homo sapiens (Human)) | BDBM50292533![]() (CHEMBL446790 | Fukugetin) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet ![]() | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Campus Inc Curated by ChEMBL | Assay Description Mixed-type inhibition of human tissue kallikrein-1 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated fo... | Bioorg Med Chem Lett 26: 1485-9 (2016) Article DOI: 10.1016/j.bmcl.2016.01.039 BindingDB Entry DOI: 10.7270/Q2862J9K | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446229![]() (CHEMBL3109060) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Kallikrein-7 (Homo sapiens (Human)) | BDBM50446230![]() (CHEMBL3109059) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Universidade Federal do ABC Curated by ChEMBL | Assay Description Competitive inhibition of human recombinant KLK7 expressed in baculovirus-infected insect cell system using Abz-KLYSSKQ-Eddnp as substrate incubated ... | ACS Med Chem Lett 5: 128-32 (2014) Article DOI: 10.1021/ml4003698 BindingDB Entry DOI: 10.7270/Q2W37XSV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112583![]() (1-{2-[2-[2-(6-Amino-2-{2-[2-(2-amino-3-methyl-pent...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112579![]() (6-Amino-2-(2-{2-[2-(6-amino-2-{2-[2-(2-amino-3-cyc...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112591![]() (2-(2-{2-[2-(2-{2-[2-(2-Amino-4-methylsulfanyl-buty...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112585![]() (2-[3-Cyclohexyl-2-(2-{2-[2-(3-(3H-imidazol-4-yl)-2...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 6.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50112582![]() (6-Amino-2-[2-(2-{2-[2-(2-{6-amino-2-[(pyrrolidine-...) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Genome polyprotein (Human rhinovirus B) | BDBM50370073![]() (CHEMBL1790421) | PDB MMDB UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | PubMed | 1.01E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Carlsberg Laboratory Curated by ChEMBL | Assay Description Inhibition of Leishmania mexicana Cysteine protease B (CPB2.8deltaCTE) was obtained in a solution-phase assay | J Med Chem 45: 1971-82 (2002) BindingDB Entry DOI: 10.7270/Q29887QH | |||||||||||
More data for this Ligand-Target Pair |
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