Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Epidermal growth factor receptor (Homo sapiens (Human)) | BDBM50276903 (CHEMBL4171764) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.60 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toledo Curated by ChEMBL | Assay Description Inhibition of EGFR1 (unknown origin) after 1 hr in presence of adenosine 5'[gamma-33P]triphosphate by microbeta microplate counting method | Eur J Med Chem 138: 1053-1065 (2017) Article DOI: 10.1016/j.ejmech.2017.07.028 BindingDB Entry DOI: 10.7270/Q2794760 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242619 (CHEMBL4105091) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242620 (CHEMBL4097381) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242621 (CHEMBL4070204) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242622 (CHEMBL4065204) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242618 (CHEMBL4099804) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242619 (CHEMBL4105091) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242620 (CHEMBL4097381) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242621 (CHEMBL4070204) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242622 (CHEMBL4065204) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242618 (CHEMBL4099804) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242619 (CHEMBL4105091) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242623 (CHEMBL4080858) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242621 (CHEMBL4070204) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242622 (CHEMBL4065204) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242618 (CHEMBL4099804) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242619 (CHEMBL4105091) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242623 (CHEMBL4080858) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242621 (CHEMBL4070204) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242622 (CHEMBL4065204) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242618 (CHEMBL4099804) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242619 (CHEMBL4105091) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242623 (CHEMBL4080858) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242621 (CHEMBL4070204) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242624 (CHEMBL4081787) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242622 (CHEMBL4065204) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242623 (CHEMBL4080858) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242624 (CHEMBL4081787) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity protein kinase CLK1 (Mus musculus) | BDBM50242623 (CHEMBL4080858) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant mouse GST-fused CLK1 expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of ATP by scinti... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242624 (CHEMBL4081787) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-T1/Cyclin-dependent kinase 9 (Homo sapiens (Human)) | BDBM50242620 (CHEMBL4097381) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK9/cyclin T expressed in insect cells using YSPTSPSYSPTSPSYSPTSPSKKKK as substrate after 30 mins in presence of ATP... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242624 (CHEMBL4081787) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-dependent kinase 5 activator 1 (Homo sapiens (Human)) | BDBM50242620 (CHEMBL4097381) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK5/p25 expressed in Escherichia coli using histone H1 as substrate after 30 mins in presence of ATP by scintillatio... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242624 (CHEMBL4081787) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM50242620 (CHEMBL4097381) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Cyclin-A2/Cyclin-dependent kinase 2 (Homo sapiens (Human)) | BDBM100152 (7-methoxy-1-methyl-9H-beta-carboline;hydrochloride...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia antibodypedia GoogleScholar AffyNet | Purchase DrugBank MCE KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant human CDK2/cyclin A using histone H1 as substrate after 30 mins in presence of ATP by scintillation counting method | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dual specificity tyrosine-phosphorylation-regulated kinase 1A (Homo sapiens (Human)) | BDBM50242618 (CHEMBL4099804) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | <1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
Rajiv Gandhi Proudyogiki Vishwavidyalaya Curated by ChEMBL | Assay Description Inhibition of recombinant full length human GST-fused DYRK1A expressed in Escherichia coli using RS peptide as substrate after 30 mins in presence of... | Bioorg Med Chem Lett 27: 2663-2667 (2017) Article DOI: 10.1016/j.bmcl.2017.04.080 BindingDB Entry DOI: 10.7270/Q28P62X6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Fibroblast growth factor receptor 1 (Homo sapiens (Human)) | BDBM50307261 (CHEMBL597990 | [2-Methoxy-4-(7-methyl-4-oxo-3,4,5,...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Toledo Curated by ChEMBL | Assay Description Inhibition of FGFR1 kinase domain (unknown origin) by caliper mobility shift assay | Eur J Med Chem 138: 1053-1065 (2017) Article DOI: 10.1016/j.ejmech.2017.07.028 BindingDB Entry DOI: 10.7270/Q2794760 | |||||||||||
More data for this Ligand-Target Pair |