Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161472 (US9108978, 2.02) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 30 | -44.7 | 203 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Escherichia coli) | BDBM50039492 (CHEMBL1231498) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | DrugBank PDB Article PubMed | 87 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of Escherichia coli recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysis | ACS Med Chem Lett 6: 216-20 (2015) Article DOI: 10.1021/ml500475n BindingDB Entry DOI: 10.7270/Q2VT1TTQ | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161468 (US9108978, 6.09) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem Similars | PDB US Patent | 90 | -41.8 | 530 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92383 (Biotin triazole, 14) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 90 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388931 (CHEMBL2063402) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 140 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50039492 (CHEMBL1231498) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL DrugBank PC cid PC sid PDB UniChem Patents Similars | Article PubMed | 182 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human recombinant BPL using 3H-biotin as substrate after 10 mins by liquid scintillation counting analysis | ACS Med Chem Lett 6: 216-20 (2015) Article DOI: 10.1021/ml500475n BindingDB Entry DOI: 10.7270/Q2VT1TTQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388933 (CHEMBL2063403) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Escherichia coli) | BDBM161472 (US9108978, 2.02) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 225 | -39.5 | n/a | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Escherichia coli) | BDBM161472 (US9108978, 2.02) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 420 | -37.9 | n/a | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161470 (US9108978, 4.01) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid PDB UniChem | PDB US Patent | 660 | -36.7 | 4.00E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161469 (US9108978, 6.07) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | US Patent | 1.17E+3 | -35.2 | 7.00E+3 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92378 (Biotin triazole, 5) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92382 (Biotin triazole, 13) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 1.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161467 (US9108978, 3.25) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | 1.83E+3 | -34.1 | 1.16E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388934 (CHEMBL2063404) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 3.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388927 (CHEMBL2063398) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | 3.85E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388932 (CHEMBL2062535) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.43E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM161471 (US9108978, 6.34) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | US Patent | >1.00E+4 | >-29.7 | >5.00E+4 | n/a | n/a | n/a | n/a | 8.0 | 37 |
Monash University; Adelaide Research & Innovation Pty Ltd US Patent | Assay Description Quantitation of BPL catalysed 3H-biotin incorporation into the biotin domain substrate was performed as previously described by Polyak et al, J. Biol... | US Patent US9108978 (2015) BindingDB Entry DOI: 10.7270/Q2T43RVW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92379 (Biotin triazole, 10) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92380 (Biotin triazole, 11) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92384 (Biotin triazole, 15) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92385 (Biotin triazole, 16) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Bifunctional ligase/repressor BirA (Staphylococcus aureus) | BDBM92381 (Biotin triazole, 12) | PDB KEGG UniProtKB/TrEMBL B.MOAD GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide | Assay Description In vitro enzyme inhibition using biotin protein ligase. | J Biol Chem 287: 17823-32 (2012) Article DOI: 10.1074/jbc.M112.356576 BindingDB Entry DOI: 10.7270/Q2DJ5D7V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388935 (CHEMBL2063405) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201192 (CHEMBL3932681) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201209 (CHEMBL3914868) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201208 (CHEMBL3892750) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201207 (CHEMBL3910734) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201206 (CHEMBL3960176) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201205 (CHEMBL3914706) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201204 (CHEMBL3927537) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201203 (CHEMBL3905724) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201202 (CHEMBL3971239) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201201 (CHEMBL3901708) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201200 (CHEMBL3905875) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201186 (CHEMBL3923732) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201187 (CHEMBL3976601) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201188 (CHEMBL3891635) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201189 (CHEMBL3984675) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201190 (CHEMBL3942705) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201191 (CHEMBL3951442) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201210 (CHEMBL3933745) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201193 (CHEMBL3974372) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201194 (CHEMBL3932600) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201195 (CHEMBL3972792) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201196 (CHEMBL3961751) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201197 (CHEMBL3895686) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201198 (CHEMBL3968104) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid PDB UniChem Patents Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50201199 (CHEMBL3934430) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Adelaide Curated by ChEMBL | Assay Description Inhibition of human biotin protein ligase assessed as reduction in 3H-biotin incorporation into pyruvate carboxylase biotin domain after 10 mins by l... | ACS Med Chem Lett 7: 1068-1072 (2016) Article DOI: 10.1021/acsmedchemlett.6b00248 BindingDB Entry DOI: 10.7270/Q2QV3PGF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Biotin--protein ligase (Homo sapiens (Human)) | BDBM50388930 (CHEMBL2063401) | Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Displacement of [3H]-biotin from human BPL after 20 mins by scintillation counting | ACS Med Chem Lett 3: 509-514 (2012) Article DOI: 10.1021/ml300106p BindingDB Entry DOI: 10.7270/Q2DZ09CN | |||||||||||
More data for this Ligand-Target Pair |
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