Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194448 (CHEMBL3972289) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 32 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194466 (CHEMBL3958557) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194475 (CHEMBL3889586) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 35 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194259 (CHEMBL3939958) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 37 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194476 (CHEMBL3942693) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 47 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194477 (CHEMBL3916023) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 56 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194258 (CHEMBL3934881) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 61 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194458 (CHEMBL3987134) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 63 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194457 (CHEMBL3969494) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 75 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194474 (CHEMBL3953637) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 81 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194450 (CHEMBL3933207) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 130 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194257 (CHEMBL3925993) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 220 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194260 (CHEMBL3973366) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 230 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194462 (CHEMBL3898460) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 240 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194469 (CHEMBL3937936) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 250 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194471 (CHEMBL3943850) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 570 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194256 (CHEMBL3944916) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 740 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194447 (CHEMBL3978944) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50538815 (CHEMBL4640937) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 1.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assay | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115176 BindingDB Entry DOI: 10.7270/Q26W9FM9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194255 (CHEMBL3935965) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50157430 (CHEMBL3781271) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Binding affinity to N-terminal His6-tagged human CBX7 (8 to 62) expressed in Escherichia coli BL21 using FITC-peptide-3 as competitive binding probe ... | ACS Med Chem Lett 7: 139-44 (2016) Article DOI: 10.1021/acsmedchemlett.5b00378 BindingDB Entry DOI: 10.7270/Q2222WNZ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194262 (CHEMBL3949885) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50538816 (CHEMBL4642464) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assay | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115176 BindingDB Entry DOI: 10.7270/Q26W9FM9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50157430 (CHEMBL3781271) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assay | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115176 BindingDB Entry DOI: 10.7270/Q26W9FM9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194465 (CHEMBL3980951) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194449 (CHEMBL3905193) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50194261 (CHEMBL3970686) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Antagonist activity at recombinant human C-terminal His-tagged CBX7 chromodomain (8 to 62 residues) expressed in Escherichia coli Rosetta BL21(DE3)pL... | J Med Chem 59: 8913-8923 (2016) Article DOI: 10.1021/acs.jmedchem.6b00801 BindingDB Entry DOI: 10.7270/Q2H1340D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009510 (CHEMBL3234188) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009456 (CHEMBL3234138) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009468 (CHEMBL3234150) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009512 (CHEMBL3234189) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009463 (CHEMBL3234145) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009517 (CHEMBL3234435) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009518 (CHEMBL3234436) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009455 (CHEMBL3234137) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009489 (CHEMBL3234171) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50179360 (CHEMBL3040216) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Connecticut Curated by ChEMBL | Assay Description Inhibition of Cbx7 (unknown origin) using FITC-labeled SETDB1-K1170me3 peptide as probe by fluorescence polarization assay | Eur J Med Chem 136: 14-35 (2017) Article DOI: 10.1016/j.ejmech.2017.04.047 BindingDB Entry DOI: 10.7270/Q2F76G3G | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50538817 (CHEMBL4646032) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | n/a | n/a | 8.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) assessed as inhibition of CBX4 disruption by competitive FP assay | Bioorg Med Chem 28: (2020) Article DOI: 10.1016/j.bmc.2019.115176 BindingDB Entry DOI: 10.7270/Q26W9FM9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009488 (CHEMBL3234170) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009469 (CHEMBL3234151) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009523 (CHEMBL3234438) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 8.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50009475 (CHEMBL3234157) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Victoria Curated by ChEMBL | Assay Description Displacement of FITC-labeled H3K27me3 from CBX7 (unknown origin) after 15 mins by fluorescence polarization assay | J Med Chem 57: 2874-83 (2014) Article DOI: 10.1021/jm401487x BindingDB Entry DOI: 10.7270/Q2571DJ3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440605 (CHEMBL2424677) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440606 (CHEMBL2426376) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440607 (CHEMBL2426375) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440608 (CHEMBL2426374) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440609 (CHEMBL2426373) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440610 (CHEMBL2426368) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440611 (CHEMBL2426367) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Chromobox protein homolog 7 (Homo sapiens (Human)) | BDBM50440612 (CHEMBL2426366) | PDB KEGG UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | >1.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
University of North Carolina at Chapel Hill Curated by ChEMBL | Assay Description Inhibition of CBX7 (unknown origin) after 30 mins by AlphaScreen assay | J Med Chem 56: 7358-71 (2013) Article DOI: 10.1021/jm400919p BindingDB Entry DOI: 10.7270/Q2B27WRP | |||||||||||
More data for this Ligand-Target Pair |
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