Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kcal/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Melatonin receptor type 1C (Xenopus) | BDBM50423058 (CHEMBL244471) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 282 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423056 (CHEMBL243002) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423059 (CHEMBL244472) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.41E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423057 (CHEMBL242573) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.51E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423062 (CHEMBL242786) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.59E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423063 (CHEMBL396501) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423061 (CHEMBL243003) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.04E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423055 (CHEMBL244957) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.19E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM85065 (CAS_117946-91-5 | Luzindole | NSC_122162) | UniProtKB/SwissProt GoogleScholar AffyNet | Purchase MCE PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 2.46E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423064 (CHEMBL244263) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.68E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423060 (CHEMBL241928) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.13E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50423065 (CHEMBL242806) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.17E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Melatonin receptor type 1C (Xenopus) | BDBM50411361 (CHEMBL396991) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
University of Athens Curated by ChEMBL | Assay Description Antagonist activity in Xenopus laevis melanophores assessed as melatoninergic activity after 60 mins | Eur J Med Chem 42: 1004-13 (2007) Article DOI: 10.1016/j.ejmech.2007.01.005 BindingDB Entry DOI: 10.7270/Q2B859BK | |||||||||||
More data for this Ligand-Target Pair |