Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350660 (CHEMBL1813552) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350661 (CHEMBL1813553) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 2.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350666 (CHEMBL1813558) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350659 (CHEMBL1813551) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350669 (CHEMBL1813546) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350649 (CHEMBL1813536) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350670 (CHEMBL1813559) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350653 (CHEMBL1813540) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350648 (CHEMBL1813535) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.10E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350654 (CHEMBL1813541) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350657 (CHEMBL1813547) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.50E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350650 (CHEMBL1813537) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.30E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350668 (CHEMBL1813545) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.90E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350652 (CHEMBL1813539) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350665 (CHEMBL1813557) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350662 (CHEMBL1813554) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.47E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350647 (CHEMBL1813534) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350664 (CHEMBL1813556) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350658 (CHEMBL1813550) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 3.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350656 (CHEMBL1813544) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350651 (CHEMBL1813538) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350663 (CHEMBL1813555) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 6.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350655 (CHEMBL1813542) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350646 (CHEMBL1813533) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350667 (CHEMBL1813560) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 8.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Transcriptional activator protein LuxR (Vibrio fischeri) | BDBM50350645 (CHEMBL1813532) | UniProtKB/SwissProt GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.53E+5 | n/a | n/a | n/a | n/a | n/a | n/a |
INSA Lyon Curated by ChEMBL | Assay Description Antagonist activity at Vibrio fischeri LuxR assessed as inhibition of 3-oxo-C6-HSL-induced quorum sensing activation mediated bioluminescence | Bioorg Med Chem 19: 4868-75 (2011) Article DOI: 10.1016/j.bmc.2011.06.075 BindingDB Entry DOI: 10.7270/Q2CC112H | |||||||||||
More data for this Ligand-Target Pair |