Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431782 (CHEMBL2347039) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431785 (CHEMBL2347036) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431784 (CHEMBL2347037) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431791 (CHEMBL2346926) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431786 (CHEMBL2347035) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431788 (CHEMBL2346929) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 15 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431783 (CHEMBL2347038) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 16 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431793 (CHEMBL2346924) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 28 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50381853 (CHEMBL2023067) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431794 (CHEMBL2346923) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431795 (CHEMBL2346922) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 44 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431792 (CHEMBL2346925) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 48 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431787 (CHEMBL2346930) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 53 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431789 (CHEMBL2346928) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 60 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431790 (CHEMBL2346927) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 139 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431781 (CHEMBL2346919) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 212 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431796 (CHEMBL2346921) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 460 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Dipeptidyl peptidase 4 (Homo sapiens (Human)) | BDBM50431797 (CHEMBL2346920) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 860 | n/a | n/a | n/a | n/a | n/a | n/a |
Chinese Academy of Science Curated by ChEMBL | Assay Description Inhibition of human DPP4 using Gly-Pro-AMC as substrate treated with enzyme 10 mins prior to substrate addition measured after 10 mins | Bioorg Med Chem 21: 1749-55 (2013) Article DOI: 10.1016/j.bmc.2013.01.062 BindingDB Entry DOI: 10.7270/Q2R78GMR | |||||||||||
More data for this Ligand-Target Pair |