Compile Data Set for Download or QSAR

Found 68 hits Enz. Inhib. hit(s) with all data for assayid = 1 entry = 2398   

Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	koff s-1	kon M-1s-1	pH	Temp °C
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364220 (US9856257, 5) Show SMILES Cc1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C18H13F3N4O/c1-10-4-2-3-5-11(10)14-6-15-12(7-22-14)16-13(8-23-24-16)17(26)25(15)9-18(19,20)21/h2-8H,9H2,1H3,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	3	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364234 (US9856257, 19) Show SMILES CNS(=O)(=O)c1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C18H14F3N5O3S/c1-22-30(28,29)15-5-3-2-4-10(15)13-6-14-11(7-23-13)16-12(8-24-25-16)17(27)26(14)9-18(19,20)21/h2-8,22H,9H2,1H3,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	4	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364246 (US9856257, 31) Show SMILES CN1CCN(CC1)c1ccc(cn1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C21H20F3N7O/c1-29-4-6-30(7-5-29)18-3-2-13(9-26-18)16-8-17-14(10-25-16)19-15(11-27-28-19)20(32)31(17)12-21(22,23)24/h2-3,8-11H,4-7,12H2,1H3,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	5	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364272 (US9856257, 57) Show SMILES OCCc1ccccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C19H15F3N4O2/c20-19(21,22)10-26-15-7-12(13-4-2-1-3-11(13)5-6-27)8-23-17(15)16-14(18(26)28)9-24-25-16/h1-4,7-9,27H,5-6,10H2,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364248 (US9856257, 33) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1cccnc1N1CCCC1 Show InChI InChI=1S/C20H17F3N6O/c21-20(22,23)11-29-16-8-15(12-4-3-5-24-18(12)28-6-1-2-7-28)25-9-13(16)17-14(19(29)30)10-26-27-17/h3-5,8-10H,1-2,6-7,11H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	6	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364237 (US9856257, 22) Show SMILES CS(=O)(=O)Nc1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C18H14F3N5O3S/c1-30(28,29)25-13-5-3-2-4-10(13)14-6-15-11(7-22-14)16-12(8-23-24-16)17(27)26(15)9-18(19,20)21/h2-8,25H,9H2,1H3,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	8	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364255 (US9856257, 40) Show SMILES CN1CCN(CC1)c1cc(ccn1)-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C21H20F3N7O/c1-29-4-6-30(7-5-29)17-9-13(2-3-25-17)14-8-16-19(26-10-14)18-15(11-27-28-18)20(32)31(16)12-21(22,23)24/h2-3,8-11H,4-7,12H2,1H3,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364216 (US9856257, 1) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1cccnc1Cl Show InChI InChI=1S/C16H9ClF3N5O/c17-14-8(2-1-3-21-14)11-4-12-9(5-22-11)13-10(6-23-24-13)15(26)25(12)7-16(18,19)20/h1-6H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	11	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364249 (US9856257, 34) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1cccnc1N1CCCNCC1 Show InChI InChI=1S/C21H20F3N7O/c22-21(23,24)12-31-17-9-16(27-10-14(17)18-15(20(31)32)11-28-29-18)13-3-1-5-26-19(13)30-7-2-4-25-6-8-30/h1,3,5,9-11,25H,2,4,6-8,12H2,(H,28,29)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	12	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364268 (US9856257, 53) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ncccc1Cl Show InChI InChI=1S/C16H9ClF3N5O/c17-10-2-1-3-21-12(10)8-4-11-14(22-5-8)13-9(6-23-24-13)15(26)25(11)7-16(18,19)20/h1-6H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364229 (US9856257, 14) Show SMILES COc1ccc(c(F)c1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C18H12F4N4O2/c1-28-9-2-3-10(13(19)4-9)14-5-15-11(6-23-14)16-12(7-24-25-16)17(27)26(15)8-18(20,21)22/h2-7H,8H2,1H3,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	19	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364221 (US9856257, 6) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccccc1C(F)(F)F Show InChI InChI=1S/C18H10F6N4O/c19-17(20,21)8-28-14-5-13(9-3-1-2-4-12(9)18(22,23)24)25-6-10(14)15-11(16(28)29)7-26-27-15/h1-7H,8H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364281 (US9856257, 66) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ccc(cc1)C(=O)C1CC1 Show InChI InChI=1S/C21H15F3N4O2/c22-21(23,24)10-28-16-7-14(8-25-18(16)17-15(20(28)30)9-26-27-17)11-1-3-12(4-2-11)19(29)13-5-6-13/h1-4,7-9,13H,5-6,10H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364231 (US9856257, 16) Show SMILES CNC(=O)c1cc(ccc1F)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C19H13F4N5O2/c1-24-17(29)10-4-9(2-3-13(10)20)14-5-15-11(6-25-14)16-12(7-26-27-16)18(30)28(15)8-19(21,22)23/h2-7H,8H2,1H3,(H,24,29)(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50097412 (CHEMBL3586448 | US9856257, 37) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1cccnc1Cl Show InChI InChI=1S/C16H9ClF3N5O/c17-14-9(2-1-3-21-14)8-4-11-13(22-5-8)12-10(6-23-24-12)15(26)25(11)7-16(18,19)20/h1-6H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Patents Similars	US Patent	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364262 (US9856257, 47) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ccccc1CNC1CC1 Show InChI InChI=1S/C21H18F3N5O/c22-21(23,24)11-29-17-7-13(9-26-19(17)18-16(20(29)30)10-27-28-18)15-4-2-1-3-12(15)8-25-14-5-6-14/h1-4,7,9-10,14,25H,5-6,8,11H2,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	21	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50097401 (CHEMBL3586459 | US9856257, 3) Show SMILES CN1CCN(CC1)c1cc(ccn1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C21H20F3N7O/c1-29-4-6-30(7-5-29)18-8-13(2-3-25-18)16-9-17-14(10-26-16)19-15(11-27-28-19)20(32)31(17)12-21(22,23)24/h2-3,8-11H,4-7,12H2,1H3,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	US Patent	n/a	n/a	24	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364257 (US9856257, 42) Show SMILES Nc1cccc(n1)-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C16H11F3N6O/c17-16(18,19)7-25-11-4-8(10-2-1-3-12(20)23-10)5-21-14(11)13-9(15(25)26)6-22-24-13/h1-6H,7H2,(H2,20,23)(H,22,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	26	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364259 (US9856257, 44) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ncccc1C(F)(F)F Show InChI InChI=1S/C17H9F6N5O/c18-16(19,20)7-28-11-4-8(12-10(17(21,22)23)2-1-3-24-12)5-25-14(11)13-9(15(28)29)6-26-27-13/h1-6H,7H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364253 (US9856257, 38) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ccccn1 Show InChI InChI=1S/C16H10F3N5O/c17-16(18,19)8-24-12-5-9(11-3-1-2-4-20-11)6-21-14(12)13-10(15(24)25)7-22-23-13/h1-7H,8H2,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	28	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364251 (US9856257, 36) Show SMILES Fc1ncccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C16H9F4N5O/c17-14-8(2-1-3-21-14)11-4-12-9(5-22-11)13-10(6-23-24-13)15(26)25(12)7-16(18,19)20/h1-6H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	31	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364256 (US9856257, 41) Show SMILES COC(=O)c1ncccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C18H12F3N5O3/c1-29-17(28)14-10(3-2-4-22-14)9-5-12-15(23-6-9)13-11(7-24-25-13)16(27)26(12)8-18(19,20)21/h2-7H,8H2,1H3,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	34	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364270 (US9856257, 55) Show SMILES Nc1ccccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C17H12F3N5O/c18-17(19,20)8-25-13-5-9(10-3-1-2-4-12(10)21)6-22-15(13)14-11(16(25)26)7-23-24-14/h1-7H,8,21H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	37	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364254 (US9856257, 39) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ccncc1 Show InChI InChI=1S/C16H10F3N5O/c17-16(18,19)8-24-12-5-10(9-1-3-20-4-2-9)6-21-14(12)13-11(15(24)25)7-22-23-13/h1-7H,8H2,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	37	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364276 (US9856257, 61) Show SMILES Nc1cnccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C16H11F3N6O/c17-16(18,19)7-25-12-3-8(9-1-2-21-6-11(9)20)4-22-14(12)13-10(15(25)26)5-23-24-13/h1-6H,7,20H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	37	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364267 (US9856257, 52) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ccc(Cl)cn1 Show InChI InChI=1S/C16H9ClF3N5O/c17-9-1-2-11(21-5-9)8-3-12-14(22-4-8)13-10(6-23-24-13)15(26)25(12)7-16(18,19)20/h1-6H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	38	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364224 (US9856257, 9) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1cccc2cccnc12 Show InChI InChI=1S/C20H12F3N5O/c21-20(22,23)10-28-16-7-15(12-5-1-3-11-4-2-6-24-17(11)12)25-8-13(16)18-14(19(28)29)9-26-27-18/h1-9H,10H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	38	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364250 (US9856257, 35) Show SMILES CCN(C)c1ncccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C19H17F3N6O/c1-3-27(2)17-11(5-4-6-23-17)14-7-15-12(8-24-14)16-13(9-25-26-16)18(29)28(15)10-19(20,21)22/h4-9H,3,10H2,1-2H3,(H,25,26)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	38	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364261 (US9856257, 46) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1cccnc1C#N Show InChI InChI=1S/C17H9F3N6O/c18-17(19,20)8-26-13-4-9(10-2-1-3-22-12(10)5-21)6-23-15(13)14-11(16(26)27)7-24-25-14/h1-4,6-7H,8H2,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	40	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364280 (US9856257, 65) Show SMILES CC(=O)c1ccccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C19H13F3N4O2/c1-10(27)12-4-2-3-5-13(12)11-6-15-17(23-7-11)16-14(8-24-25-16)18(28)26(15)9-19(20,21)22/h2-8H,9H2,1H3,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	41	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364238 (US9856257, 23) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1cccc(c1)-n1cccn1 Show InChI InChI=1S/C20H13F3N6O/c21-20(22,23)11-28-17-8-16(12-3-1-4-13(7-12)29-6-2-5-26-29)24-9-14(17)18-15(19(28)30)10-25-27-18/h1-10H,11H2,(H,25,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	41	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364245 (US9856257, 30) Show SMILES CCNS(=O)(=O)c1ccc(cc1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C19H16F3N5O3S/c1-2-25-31(29,30)12-5-3-11(4-6-12)15-7-16-13(8-23-15)17-14(9-24-26-17)18(28)27(16)10-19(20,21)22/h3-9,25H,2,10H2,1H3,(H,24,26)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	42	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364222 (US9856257, 7) Show SMILES Fc1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C17H10F4N4O/c18-12-4-2-1-3-9(12)13-5-14-10(6-22-13)15-11(7-23-24-15)16(26)25(14)8-17(19,20)21/h1-7H,8H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	45	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364269 (US9856257, 54) Show SMILES Cc1cc(nc(N)n1)-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C16H12F3N7O/c1-7-2-10(24-15(20)23-7)8-3-11-13(21-4-8)12-9(5-22-25-12)14(27)26(11)6-16(17,18)19/h2-5H,6H2,1H3,(H,22,25)(H2,20,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	45	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364277 (US9856257, 62) Show SMILES CCCC(=O)Nc1ccccc1-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C21H18F3N5O2/c1-2-5-17(30)27-15-7-4-3-6-13(15)12-8-16-19(25-9-12)18-14(10-26-28-18)20(31)29(16)11-21(22,23)24/h3-4,6-10H,2,5,11H2,1H3,(H,26,28)(H,27,30)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	46	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364233 (US9856257, 18) Show SMILES CCOCc1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C20H17F3N4O2/c1-2-29-10-12-5-3-4-6-13(12)16-7-17-14(8-24-16)18-15(9-25-26-18)19(28)27(17)11-20(21,22)23/h3-9H,2,10-11H2,1H3,(H,25,26)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	49	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM50097411 (CHEMBL3586449 | US9856257, 67) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1cccnc1 Show InChI InChI=1S/C16H10F3N5O/c17-16(18,19)8-24-12-4-10(9-2-1-3-20-5-9)6-21-14(12)13-11(15(24)25)7-22-23-13/h1-7H,8H2,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	CHEMBL PC cid PC sid UniChem Similars	US Patent	n/a	n/a	52	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364239 (US9856257, 24) Show SMILES Cc1nc(Cl)ccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C17H11ClF3N5O/c1-8-9(2-3-14(18)24-8)12-4-13-10(5-22-12)15-11(6-23-25-15)16(27)26(13)7-17(19,20)21/h2-6H,7H2,1H3,(H,23,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	54	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364274 (US9856257, 59) Show SMILES Cc1cc(ncn1)-c1cnc2c3[nH]ncc3c(=O)n(CC(F)(F)F)c2c1 Show InChI InChI=1S/C16H11F3N6O/c1-8-2-11(22-7-21-8)9-3-12-14(20-4-9)13-10(5-23-24-13)15(26)25(12)6-16(17,18)19/h2-5,7H,6H2,1H3,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	58	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364223 (US9856257, 8) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccncc1 Show InChI InChI=1S/C16H10F3N5O/c17-16(18,19)8-24-13-5-12(9-1-3-20-4-2-9)21-6-10(13)14-11(15(24)25)7-22-23-14/h1-7H,8H2,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	60	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364273 (US9856257, 58) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1ncccc1C#N Show InChI InChI=1S/C17H9F3N6O/c18-17(19,20)8-26-12-4-10(13-9(5-21)2-1-3-22-13)6-23-15(12)14-11(16(26)27)7-24-25-14/h1-4,6-7H,8H2,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	61	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364235 (US9856257, 20) Show SMILES Oc1c(Cl)cccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C17H10ClF3N4O2/c18-11-3-1-2-8(15(11)26)12-4-13-9(5-22-12)14-10(6-23-24-14)16(27)25(13)7-17(19,20)21/h1-6,26H,7H2,(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	61	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364263 (US9856257, 48) Show SMILES FC(F)(F)Cn1c2cc(cnc2c2[nH]ncc2c1=O)-c1cncnc1C1CCCC1 Show InChI InChI=1S/C20H17F3N6O/c21-20(22,23)9-29-15-5-12(6-25-18(15)17-14(19(29)30)8-27-28-17)13-7-24-10-26-16(13)11-3-1-2-4-11/h5-8,10-11H,1-4,9H2,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	62	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364240 (US9856257, 25) Show SMILES CC(C)NS(=O)(=O)c1ccc(cc1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C20H18F3N5O3S/c1-11(2)27-32(30,31)13-5-3-12(4-6-13)16-7-17-14(8-24-16)18-15(9-25-26-18)19(29)28(17)10-20(21,22)23/h3-9,11,27H,10H2,1-2H3,(H,25,26)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	62	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364217 (US9856257, 2) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccccn1 Show InChI InChI=1S/C16H10F3N5O/c17-16(18,19)8-24-13-5-12(11-3-1-2-4-20-11)21-6-9(13)14-10(15(24)25)7-22-23-14/h1-7H,8H2,(H,22,23)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	64	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364225 (US9856257, 10) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccccc1OC(F)(F)F Show InChI InChI=1S/C18H10F6N4O2/c19-17(20,21)8-28-13-5-12(9-3-1-2-4-14(9)30-18(22,23)24)25-6-10(13)15-11(16(28)29)7-26-27-15/h1-7H,8H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	72	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364232 (US9856257, 17) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccccc1CN1CCOCC1 Show InChI InChI=1S/C22H20F3N5O2/c23-22(24,25)13-30-19-9-18(26-10-16(19)20-17(21(30)31)11-27-28-20)15-4-2-1-3-14(15)12-29-5-7-32-8-6-29/h1-4,9-11H,5-8,12-13H2,(H,27,28)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	75	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364227 (US9856257, 12) Show SMILES FC(F)(F)Cn1c2cc(ncc2c2[nH]ncc2c1=O)-c1ccc(cc1)N1CCOCC1 Show InChI InChI=1S/C21H18F3N5O2/c22-21(23,24)12-29-18-9-17(25-10-15(18)19-16(20(29)30)11-26-27-19)13-1-3-14(4-2-13)28-5-7-31-8-6-28/h1-4,9-11H,5-8,12H2,(H,26,27)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	75	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364244 (US9856257, 29) Show SMILES CN(C)S(=O)(=O)c1ccccc1-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C19H16F3N5O3S/c1-26(2)31(29,30)16-6-4-3-5-11(16)14-7-15-12(8-23-14)17-13(9-24-25-17)18(28)27(15)10-19(20,21)22/h3-9H,10H2,1-2H3,(H,24,25)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	82	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair
Methionine aminopeptidase 2 (Homo sapiens (Human))	BDBM364228 (US9856257, 13) Show SMILES Nc1ccc(cn1)-c1cc2n(CC(F)(F)F)c(=O)c3cn[nH]c3c2cn1 Show InChI InChI=1S/C16H11F3N6O/c17-16(18,19)7-25-12-3-11(8-1-2-13(20)22-4-8)21-5-9(12)14-10(15(25)26)6-23-24-14/h1-6H,7H2,(H2,20,22)(H,23,24)	PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar AffyNet	PC cid PC sid UniChem	US Patent	n/a	n/a	102	n/a	n/a	n/a	n/a	n/a	n/a
Wyeth Research					Assay Description For the enzymatic test, human MetAP2 protein was obtained from a culture supernatant of insect cells (sf9) infected with MetAP2 recombinant baculovir...				Bioorg Med Chem 15: 3321-33 (2007) BindingDB Entry DOI: 10.7270/Q26T0PZK
					More data for this Ligand-Target Pair

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