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| Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091104 (CHEMBL29422 | N-[2'-(3,4-Dimethyl-isoxazol-5-ylsul...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet  | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091101 (4'-Oxazol-4-yl-biphenyl-2-sulfonic acid (3,4-dimet...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091105 (4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 1.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091108 (4'-(4-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091109 (4'-Oxazol-5-yl-biphenyl-2-sulfonic acid (3,4-dimet...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 3.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50068674 (2'-Amino-4'-isobutyl-biphenyl-2-sulfonic acid (3,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091106 (4'-(5-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 4.70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091107 (4'-(5-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091103 (4'-(4,5-Dimethyl-oxazol-2-yl)-biphenyl-2-sulfonic ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50068742 (4'-Isobutyl-biphenyl-2-sulfonic acid (3,4-dimethyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 18 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091102 (4'-Oxazol-2-ylmethyl-biphenyl-2-sulfonic acid (3,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 19 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50034435 (5-Dimethylamino-naphthalene-1-sulfonic acid (3,4-d...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 55 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091099 (4'-(2-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 70 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50068742 (4'-Isobutyl-biphenyl-2-sulfonic acid (3,4-dimethyl...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin-1 receptor (Homo sapiens (Human)) | BDBM50091100 (4'-Benzooxazol-2-yl-biphenyl-2-sulfonic acid (3,4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 2.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inhibition of Human Endothelin A receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091104 (CHEMBL29422 | N-[2'-(3,4-Dimethyl-isoxazol-5-ylsul...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 4.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091107 (4'-(5-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091103 (4'-(4,5-Dimethyl-oxazol-2-yl)-biphenyl-2-sulfonic ...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091105 (4''-Oxazol-2-yl-biphenyl-2-sulfonic acid (3,4-dime...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | 1.87E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091101 (4'-Oxazol-4-yl-biphenyl-2-sulfonic acid (3,4-dimet...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091102 (4'-Oxazol-2-ylmethyl-biphenyl-2-sulfonic acid (3,4...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 3.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091109 (4'-Oxazol-5-yl-biphenyl-2-sulfonic acid (3,4-dimet...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 7.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091106 (4'-(5-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 9.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091100 (4'-Benzooxazol-2-yl-biphenyl-2-sulfonic acid (3,4-...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | 9.40E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091108 (4'-(4-Methyl-oxazol-2-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
| Endothelin receptor type B (Homo sapiens (Human)) | BDBM50091099 (4'-(2-Methyl-oxazol-4-yl)-biphenyl-2-sulfonic acid...) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | 1.10E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Bristol-Myers Squibb Pharmaceutical Research Institute Curated by ChEMBL | Assay Description Inihibition of Human Endothelin B receptor expressed in CHO Cells. | J Med Chem 43: 3111-7 (2000) BindingDB Entry DOI: 10.7270/Q2DF6QFM | |||||||||||
| More data for this Ligand-Target Pair | |||||||||||||
