Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500893 (CHEMBL3797662) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500901 (CHEMBL3799266) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 1.60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500908 (CHEMBL3797537) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50175665 ((R)-(4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500894 (CHEMBL3799578) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50380884 (CHEMBL2018954) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500902 (CHEMBL3798452) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500896 (CHEMBL3799393) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500910 (CHEMBL3799025) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500898 (CHEMBL3797567) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 20 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500906 (CHEMBL3798263) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500903 (CHEMBL3799865) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500907 (CHEMBL3797980) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500909 (CHEMBL3799514) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500900 (CHEMBL3798949) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500899 (CHEMBL3798941) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500905 (CHEMBL3798539) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500897 (CHEMBL3799904) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500912 (CHEMBL3797946) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 126 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500904 (CHEMBL3797678) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 316 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500911 (CHEMBL3797555) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Displacement of [125I]-TARC from human recombinant CCR4 expressed in CHO cell membranes by scintillation counting method | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50175665 ((R)-(4-(4-(2,4-dichlorobenzylamino)pyrimidin-2-yl)...) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Antagonist activity at human CCR4 expressed in CHO cells by [35S]GTPgammaS assay | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500901 (CHEMBL3799266) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Antagonist activity at human CCR4 expressed in CHO cells by [35S]GTPgammaS assay | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500893 (CHEMBL3797662) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Antagonist activity at human CCR4 expressed in CHO cells by [35S]GTPgammaS assay | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500894 (CHEMBL3799578) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | 7.90 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Antagonist activity at human CCR4 expressed in CHO cells by [35S]GTPgammaS assay | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500902 (CHEMBL3798452) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 13 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500896 (CHEMBL3799393) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 6.30 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500893 (CHEMBL3797662) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 158 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500895 (CHEMBL3797462) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 398 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50500894 (CHEMBL3799578) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | n/a | n/a | n/a | n/a | 16 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
C-C chemokine receptor type 4 (Homo sapiens (Human)) | BDBM50380881 (CHEMBL2018953) | UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | CHEMBL MCE PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | n/a | n/a | 10 | n/a | n/a | n/a | n/a |
GlaxoSmithKline Medicines Research Centre Curated by ChEMBL | Assay Description Induction of CCR4 internalisation in human HUT78 cells after 30 mins by flow cytometry | Eur J Med Chem 115: 14-25 (2016) Article DOI: 10.1016/j.ejmech.2016.02.058 BindingDB Entry DOI: 10.7270/Q24J0J4S | |||||||||||
More data for this Ligand-Target Pair |