BDBM5446
| - 3-phosphoinositide dependent protein kinase-1
- 5'-AMP-activated protein kinase catalytic subunit alpha-1
- ABL Mutant (T315I)
- ABL1(Q252H)
- ALK tyrosine kinase receptor
- AMPK subunit alpha-2
- AP2-associated protein kinase 1
- ATP-binding cassette sub-family G member 2
- Activin receptor type-1
- Activin receptor type-1B
- Activin receptor type-2A
- Activin receptor type-2B
- Activin receptor-like kinase 3 (ALK-3)
- Adrenergic Alpha
- Ankyrin repeat and protein kinase domain-containing protein 1
- Apoptosis Signal-regulating Kinase 1 (ASK1)
- Aurora Kinase C (Aurora-C)
- Aurora kinase A
- Aurora kinase B
- BDNF/NT-3 growth factors receptor
- BIKE
- BMP-2-inducible protein kinase
- BR serine/threonine-protein kinase 1
- BR serine/threonine-protein kinase 2
- Bile salt export pump
- Bone morphogenetic protein receptor type-1B (BMPR1B)
- Bone morphogenetic protein receptor type-2
- CAMK2A
- CAMK2B
- CDC2-like kinase 3 (CLK3)
- CDK7/Cyclin H/MNAT1
- CDKL2
- CaM kinase I alpha
- CaM kinase I delta
- CaM kinase I gamma
- CaM kinase II
- CaM kinase IV
- CaM-kinase kinase alpha
- CaM-kinase kinase beta
- Calcium-dependent protein kinase 1
- Calcium/calmodulin-dependent protein kinase type II subunit delta
- Casein kinase I
- Casein kinase I delta/epsilon
- Casein kinase I isoform alpha
- Casein kinase I isoform alpha-like
- Casein kinase I isoform delta
- Casein kinase I isoform gamma-3
- Casein kinase II alpha
- Casein kinase II subunit alpha
- Cell division control protein 2 homolog
- Chaperone activity of bc1 complex-like, mitochondrial
- Citron Rho-interacting kinase
- Cyclin-Dependent Kinase 5 (CDK5)
- Cyclin-dependent kinase 11A
- Cyclin-dependent kinase 13
- Cyclin-dependent kinase 15
- Cyclin-dependent kinase 19
- Cyclin-dependent kinase 2
- Cyclin-dependent kinase 3 (CDK3)
- Cyclin-dependent kinase 4
- Cyclin-dependent kinase 8
- Cyclin-dependent kinase 9
- Cyclin-dependent kinase-like 1
- Cyclin-dependent kinase-like 3
- Cyclin-dependent kinase-like 5
- Cytochrome P450 3A
- Death-associated protein kinase 1
- Death-associated protein kinase 2
- Death-associated protein kinase 3
- Discoidin domain-containing receptor 2
- Dual serine/threonine and tyrosine protein kinase
- Dual specificity mitogen-activated protein kinase kinase 1
- Dual specificity mitogen-activated protein kinase kinase 2
- Dual specificity mitogen-activated protein kinase kinase 3
- Dual specificity mitogen-activated protein kinase kinase 4
- Dual specificity mitogen-activated protein kinase kinase 5
- Dual specificity mitogen-activated protein kinase kinase 6
- Dual specificity mitogen-activated protein kinase kinase 7 (MAP2K7)
- Dual specificity protein kinase CLK2
- Dual specificity protein kinase CLK4
- Dual specificity protein kinase TTK
- Dual specificity testis-specific protein kinase 1
- Dual specificty protein kinase CLK1
- Dual-specificity tyrosine-phosphorylation regulated kinase 1A
- Dual-specificity tyrosine-phosphorylation regulated kinase 2
- Dual-specificity tyrosine-regulated kinases 1B
- EGF-R Tyrosine Kinase
- EGF-R Tyrosine Kinase Mutant (G719C)
- EGF-R Tyrosine Kinase Mutant (T790M)
- EGFR(L858R)
- EPHA8
- EPHB1
- Ephrin receptor
- Ephrin type-A receptor 1 (EPHA1)
- Ephrin type-A receptor 3 (EPHA3)
- Ephrin type-A receptor 7
- Ephrin type-B receptor 3 (EPHB3)
- Ephrin type-B receptor 4 (EphB4)
- Epidermal growth factor receptor
- Epithelial discoidin domain-containing receptor 1
- Eukaryotic translation initiation factor 2-alpha kinase 1
- Eukaryotic translation initiation factor 2-alpha kinase 4
- Extracellular signal-regulated kinase 5 (ERK5)
- FLT3(D835H)
- FLT3(D835Y)
- Ferrochelatase R115L (FECH)
- Fibroblast growth factor receptor 1
- Fibroblast growth factor receptor 2
- Fibroblast growth factor receptor 3
- Fibroblast growth factor receptor 4
- Focal adhesion kinase 1
- Focal adhesion kinase 1/vascular endothelial growth factor receptor 3
- G protein-coupled receptor kinase 4
- G protein-coupled receptor kinase 7
- GCN2(Kin.Dom.2 S808G)
- Glycogen synthase kinase-3
- Glycogen synthase kinase-3 beta
- Hepatocyte growth factor receptor
- High affinity nerve growth factor receptor
- Homeodomain-interacting protein kinase 1
- Homeodomain-interacting protein kinase 2 (HIPK2)
- Homeodomain-interacting protein kinase 3
- Homeodomain-interacting protein kinase 4
- Hormonally up-regulated neu tumor-associated kinase
- Inhibitor of NF-kappa-B kinase (IKK)
- Inhibitor of nuclear factor kappa-B kinase subunit epsilon
- Insulin receptor
- Insulin receptor-related protein
- Insulin-like growth factor I receptor
- Interferon-induced, double-stranded RNA-activated protein kinase
- Interleukin-1 receptor-associated kinase 1
- Interleukin-1 receptor-associated kinase 3
- Interleukin-1 receptor-associated kinase 4
- LIM domain kinase 1
- LIM domain kinase 2
- Leucine-rich repeat serine/threonine-protein kinase 2 (LRRK2)
- Leukocyte tyrosine kinase receptor
- MAP kinase p38
- MAP kinase-activated protein kinase 2
- MAP kinase-activated protein kinase 5
- MAP kinase-interacting serine/threonine-protein kinase 1
- MAP kinase-interacting serine/threonine-protein kinase 2
- MAP/microtubule affinity-regulating kinase 2
- MAP/microtubule affinity-regulating kinase 4
- MAST1/MAST2
- Macrophage colony-stimulating factor 1 receptor
- Macrophage-stimulating protein receptor
- Mast/stem cell growth factor receptor Kit
- Maternal embryonic leucine zipper kinase (MELK)
- Misshapen-like kinase 1
- Mitogen-activated protein kinase 1
- Mitogen-activated protein kinase 10
- Mitogen-activated protein kinase 13 (MAPK13)
- Mitogen-activated protein kinase 14
- Mitogen-activated protein kinase 15
- Mitogen-activated protein kinase 2
- Mitogen-activated protein kinase 3
- Mitogen-activated protein kinase 4
- Mitogen-activated protein kinase 6
- Mitogen-activated protein kinase 9
- Mitogen-activated protein kinase kinase kinase 1
- Mitogen-activated protein kinase kinase kinase 10
- Mitogen-activated protein kinase kinase kinase 11
- Mitogen-activated protein kinase kinase kinase 12
- Mitogen-activated protein kinase kinase kinase 13
- Mitogen-activated protein kinase kinase kinase 15
- Mitogen-activated protein kinase kinase kinase 2
- Mitogen-activated protein kinase kinase kinase 3
- Mitogen-activated protein kinase kinase kinase 4
- Mitogen-activated protein kinase kinase kinase 6
- Mitogen-activated protein kinase kinase kinase 9 (MLK1)
- Mitogen-activated protein kinase kinase kinase kinase 1
- Mitogen-activated protein kinase kinase kinase kinase 3
- Mitogen-activated protein kinase kinase kinase kinase 4
- Mitogen-activated protein kinase kinase kinase kinase 5
- Mixed lineage kinase 7
- Multidrug resistance-associated protein 2 (MRP2)
- Muscle, skeletal receptor tyrosine protein kinase
- Myosin IIIA
- Myosin light chain kinase
- Myosin light chain kinase family member 4
- Myosin light chain kinase, smooth muscle
- Myosin-IIIB
- Myotonin-protein kinase
- NT-3 growth factor receptor
- NUAK family SNF1-like kinase 1
- NUAK family SNF1-like kinase 2
- Non-receptor tyrosine-protein kinase TNK1
- Non-receptor tyrosine-protein kinase TYK2
- P-glycoprotein 1
- PAK1
- PITSLRE serine/threonine-protein kinase CDC2L1
- PRP4 kinase (PRP4)
- PTK2B protein tyrosine kinase 2 beta (PTK2B)
- Peptidyl-prolyl cis-trans isomerase FKBP1B/Serine/threonine-protein kinase mTOR
- Peripheral plasma membrane protein CASK
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform/gamma isoform
- Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
- Phosphatidylinositol 4-kinase beta
- Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta
- Phosphatidylinositol-4-phosphate 3-kinase C2 domain-containing subunit gamma
- Phosphatidylinositol-4-phosphate 5-kinase type-1 alpha
- Phosphatidylinositol-4-phosphate 5-kinase type-1 gamma
- Phosphatidylinositol-5-phosphate 4-kinase type-2 beta
- Phosphatidylinositol-5-phosphate 4-kinase type-2 gamma
- Phosphorylase kinase
- Platelet-derived growth factor receptor
- Platelet-derived growth factor receptor beta
- Protein kinase C delta type
- Protein kinase C iota (PKCι)
- Protein kinase C theta type
- Protein kinase C, epsilon
- Protein kinase C, eta
- Protein kinase N1
- Protein kinase N2
- Proto-oncogene tyrosine-protein kinase ROS
- Proto-oncogene tyrosine-protein kinase Src
- Proto-oncogene tyrosine-protein kinase receptor Ret
- Putative uncharacterized serine/threonine-protein kinase SgK110
- RAC-alpha serine/threonine-protein kinase AKT1
- RAF proto-oncogene serine/threonine-protein kinase
- RAF serine/threonine protein kinase
- RET Mutant (M918T)
- Receptor tyrosine-protein kinase erbB-2
- Receptor tyrosine-protein kinase erbB-4
- Receptor-interacting protein 1 (RIPK1)
- Receptor-interacting serine/threonine-protein kinase 4
- Rho-associated protein kinase 1
- Rho-associated protein kinase 2
- Rhodopsin kinase
- Ribosomal protein S6 kinase (P70S6K)
- Ribosomal protein S6 kinase alpha 1
- Ribosomal protein S6 kinase alpha 2
- Ribosomal protein S6 kinase alpha 4
- Ribosomal protein S6 kinase alpha 5
- Ribosomal protein S6 kinase alpha 6
- Ribosomal protein S6 kinase alpha-3
- SNF-related serine/threonine-protein kinase
- SPS1/STE20-related protein kinase YSK4
- SRC
- STE20/SPS1-related proline-alanine-rich protein kinase
- Salt-inducible kinase 2 (SIK2)
- Serine/threonine protein kinase NLK
- Serine/threonine-protein kinase 10
- Serine/threonine-protein kinase 11
- Serine/threonine-protein kinase 17A
- Serine/threonine-protein kinase 17B (STK17B)
- Serine/threonine-protein kinase 2
- Serine/threonine-protein kinase 24
- Serine/threonine-protein kinase 25
- Serine/threonine-protein kinase 32A
- Serine/threonine-protein kinase 32B
- Serine/threonine-protein kinase 32C
- Serine/threonine-protein kinase 33
- Serine/threonine-protein kinase 35
- Serine/threonine-protein kinase 36
- Serine/threonine-protein kinase 38
- Serine/threonine-protein kinase 38-like
- Serine/threonine-protein kinase 4 (STK4)
- Serine/threonine-protein kinase AKT
- Serine/threonine-protein kinase AKT2
- Serine/threonine-protein kinase Aurora-C
- Serine/threonine-protein kinase CHK2
- Serine/threonine-protein kinase Chk1
- Serine/threonine-protein kinase D1
- Serine/threonine-protein kinase D2
- Serine/threonine-protein kinase D3
- Serine/threonine-protein kinase DCLK1
- Serine/threonine-protein kinase DCLK2
- Serine/threonine-protein kinase DCLK3
- Serine/threonine-protein kinase GAK
- Serine/threonine-protein kinase ICK
- Serine/threonine-protein kinase LATS1
- Serine/threonine-protein kinase LATS2
- Serine/threonine-protein kinase MAK
- Serine/threonine-protein kinase MARK1
- Serine/threonine-protein kinase MRCK alpha
- Serine/threonine-protein kinase MRCK beta
- Serine/threonine-protein kinase MRCK gamma
- Serine/threonine-protein kinase MST2
- Serine/threonine-protein kinase MST4
- Serine/threonine-protein kinase NEK6
- Serine/threonine-protein kinase NEK7
- Serine/threonine-protein kinase NEK9
- Serine/threonine-protein kinase NIM1
- Serine/threonine-protein kinase Nek1
- Serine/threonine-protein kinase Nek11
- Serine/threonine-protein kinase Nek2
- Serine/threonine-protein kinase Nek3
- Serine/threonine-protein kinase Nek4
- Serine/threonine-protein kinase Nek5
- Serine/threonine-protein kinase OSR1
- Serine/threonine-protein kinase PAK 4
- Serine/threonine-protein kinase PAK6
- Serine/threonine-protein kinase PAK7
- Serine/threonine-protein kinase PCTAIRE-1
- Serine/threonine-protein kinase PCTAIRE-2
- Serine/threonine-protein kinase PCTAIRE-3
- Serine/threonine-protein kinase PFTAIRE-1
- Serine/threonine-protein kinase PIM
- Serine/threonine-protein kinase PLK1
- Serine/threonine-protein kinase PLK2
- Serine/threonine-protein kinase PLK3
- Serine/threonine-protein kinase PLK4
- Serine/threonine-protein kinase PRKX
- Serine/threonine-protein kinase RIO1
- Serine/threonine-protein kinase RIO2
- Serine/threonine-protein kinase RIO3
- Serine/threonine-protein kinase RIPK2
- Serine/threonine-protein kinase SBK1
- Serine/threonine-protein kinase SIK1
- Serine/threonine-protein kinase SIK3
- Serine/threonine-protein kinase SRPK1
- Serine/threonine-protein kinase SRPK2
- Serine/threonine-protein kinase SRPK3
- Serine/threonine-protein kinase Sgk3
- Serine/threonine-protein kinase TAO1
- Serine/threonine-protein kinase TAO2
- Serine/threonine-protein kinase TAO3
- Serine/threonine-protein kinase TBK1
- Serine/threonine-protein kinase ULK1
- Serine/threonine-protein kinase ULK2
- Serine/threonine-protein kinase ULK3
- Serine/threonine-protein kinase VRK2
- Serine/threonine-protein kinase WEE1
- Serine/threonine-protein kinase c-TAK1
- Serine/threonine-protein kinase pim-2
- Serine/threonine-protein kinase pim-3
- Serine/threonine-protein kinase pknB
- Serine/threonine-protein kinase receptor R3
- Serine/threonine-protein kinase tousled-like 1
- Serine/threonine-protein kinase tousled-like 2
- Serine/threonine-protein kinase/endoribonuclease IRE1 Alpha
- Solute carrier organic anion transporter family member 1B1 (OATP1B1)
- Solute carrier organic anion transporter family member 1B3 (OATP1B3)
- Solute carrier organic anion transporter family member 2B1
- Src Mutant (S345C)
- Src Mutant (S345C/T338M)
- TAK1/TAB1
- TGF-beta receptor type I
- TGF-beta receptor type II
- TNK1
- TNNI3K
- TRAF2 and NCK-interacting protein kinase (TNIK)
- Testis-specific serine/threonine-protein kinase 1
- Transient receptor potential cation channel subfamily M member 6
- Tubulin alpha-1 chain
- Tyrosine Kinase EPHA3
- Tyrosine Kinase FLT3 Mutant (N841I)
- Tyrosine kinase non-receptor protein 2
- Tyrosine- and threonine-specific cdc2-inhibitory kinase
- Tyrosine-protein kinase ABL1
- Tyrosine-protein kinase ABL2
- Tyrosine-protein kinase BMX
- Tyrosine-protein kinase BRK
- Tyrosine-protein kinase BTK
- Tyrosine-protein kinase Blk
- Tyrosine-protein kinase CSK
- Tyrosine-protein kinase CTK
- Tyrosine-protein kinase FER
- Tyrosine-protein kinase Fes/Fps
- Tyrosine-protein kinase ITK/TSK
- Tyrosine-protein kinase JAK1
- Tyrosine-protein kinase JAK2
- Tyrosine-protein kinase JAK3
- Tyrosine-protein kinase Lck
- Tyrosine-protein kinase Lyn
- Tyrosine-protein kinase Mer
- Tyrosine-protein kinase STK16 (STK16)
- Tyrosine-protein kinase SYK
- Tyrosine-protein kinase TEC
- Tyrosine-protein kinase TXK (TXK)
- Tyrosine-protein kinase Yes
- Tyrosine-protein kinase ZAP-70
- Tyrosine-protein kinase receptor FLT3
- Tyrosine-protein kinase receptor TYRO3
- Tyrosine-protein kinase receptor Tie-1
- Tyrosine-protein kinase receptor UFO
- ULK3 kinase
- Uncharacterized aarF domain-containing protein kinase 4
- Vascular endothelial growth factor receptor 1
- Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)
- Wee1-like protein kinase 2
- c-Jun N-terminal kinase, JNK
- cAMP-dependent protein kinase (PKA)
- cGMP-dependent protein kinase
- cGMP-dependent protein kinase 2
- myosin light chain kinase 2
- p21-Activated kinase 2 (PAK2)
- p21-Activated kinase 3 (PAK3)
- p38 delta/gamma
| 22 | 133 | 858 | 0 | 0 | 0 | 0 | 0 | - CHEMBL553
- ERLOTINIB HYDROCHLORIDE
- Erlotinib
- Erotinib
- N-(3-Ethynylphenyl)-6,7-bis(2-methoxyethoxy)-4-quinazolinamine Monohydrochloride
- N-(3-ethynylphenyl)-6,7-bis(2-methoxyethoxy)quinazolin-4-amine
- OSI-774
- Tarceva
- US10189853, erlotinib
- US9409845, Table 1, Compound 22: erlotinib
- US9730934, Erlotinib
- cid_176870
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