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Compound Name:

Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically

Compound Name (alphabetical)	Binding Targets	Enz. Inhib. Data							ITC Data	Alternate Compound Names
		Ki	IC50	Kd	EC50	Koff	Kon	Other
BDBM26266	GABA A Alpha2Beta1Gamma2 GABA A Alpha4Beta2Gamma2 GABA A receptor alpha-1/beta-1/gamma-2 GABA A receptor alpha-2/beta-2/gamma-2 GABA A receptor alpha-3/beta-2/gamma-2 GABA A receptor alpha-5/beta-3/gamma-2 GABA A receptor alpha-6/beta-2/gamma-2 GABA receptor alpha-1/beta-2/gamma-2 subunit GABA receptor alpha-1/beta-3/gamma-2 subunit GABA receptor alpha-2/beta-2/gamma-2 subunit GABA receptor alpha-2/beta-3/gamma-2 subunit GABA receptor alpha-3/beta-2/gamma-2 subunit GABA receptor alpha-3/beta-3/gamma-2 subunit GABA receptor alpha-5/beta-3/gamma-2 subunit GABA receptor alpha-6/beta-2/gamma-2 subunit GABA receptor alpha-6/beta-3/gamma-2 subunit GABA(A) receptor subunit alpha-2 GABAA Receptor Mutant, alpha-1 (A160C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (F99C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (G157C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (G200C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (S204C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (S205C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (T162C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (T206C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (V202C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1 (V211C), beta-2, gamma-2 GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (A79C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (Chimera) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (D56C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (L140C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (M130C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R132C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R144C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R185C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (R194C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T126C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T142C) GABAA Receptor Mutant, alpha-1, beta-2, gamma-2 (T81C) GABAA Receptor, alpha-1, beta-2, gamma-2 GABAA Receptor, alpha-2, beta-2, gamma-2 GABAA Receptor, alpha-3, beta-2, gamma-2 GABAA Receptor, alpha-4, beta-2, gamma-2 GABAA Receptor, alpha-5, beta-2, gamma-2 GABAA Receptor, alpha-6, beta-2, gamma-2 Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1) Gamma-aminobutyric acid receptor subunit alpha-1/ beta-1 Gamma-aminobutyric acid receptor subunit alpha-3 Gamma-aminobutyric acid receptor subunit alpha-5 (GABA(A)) Gamma-aminobutyric acid type B receptor subunit 1 Peripheral-Type Benzodiazepine Receptor	128	4	0	7	0	0	0	0	Ambien CHEMBL911 Dalparan N,N-dimethyl-2-[6-methyl-2-(4-methylphenyl)imidazo[1,2-a]pyridin-3-yl]acetamide ZPM Zolpidem Zolpidem tartrate
BDBM26948	15-Lipoxygenase (LoxA) 5-HT3A Serotonin Receptor 5-Hydroxytryptamine receptor 6 (5-HT6) 5-hydroxytryptamine receptor 1A (5-HT1A) 5-hydroxytryptamine receptor 1B 5-hydroxytryptamine receptor 1D 5-hydroxytryptamine receptor 2A Alpha-1A adrenergic receptor Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor Alpha-2C adrenergic receptor Beta-1 adrenergic receptor Beta-2 adrenergic receptor and beta-3 adrenergic receptor CCKBR Calcium channel Cholecystokinin B Cholinergic, muscarinic Cysteinyl leukotriene receptor 1 D(2) dopamine receptor D(3) dopamine receptor DNA damage-inducible transcript 3 protein DOPAMINE DRD1 DRD2 Delta-type opioid receptor Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor Dopamine Transporter (DAT) Dopamine receptor Dopamine receptors; D2 & D4 Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1) Glycine receptor subunit alpha-1 HTR2C Histamine H1 receptor Kappa-type opioid receptor Muscarinic acetylcholine receptor M2 NT Nociceptin receptor Nociceptin/mu opioid receptor Norepinephrine transporter Potassium voltage-gated channel subfamily H member 2 Prostanoid TP receptor Serotonin (5-HT) receptor Serotonin 1B/1D receptor Serotonin receptor (2b and 2c) Sigma non-opioid intracellular receptor 1 Sodium-dependent serotonin transporter Substance P Twik-RElated Potassium (K+) channel 1 (TREK1) Voltage-gated sodium channel subunit alpha Nav1.8 XBP1 adrenergic Alpha2	56	5	0	2	0	0	0	0	8-[4,4-bis(4-fluorophenyl)butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one CHEMBL46516 FLUSPIRILENE NCGC00015424 cid_3396 spiropiperidine analogue, 1
BDBM50021626	40S ribosomal protein S27 ALK tyrosine kinase receptor Activator of S phase kinase DBF4/Cell division cycle 7-related protein kinase Aurora kinase A Aurora kinase B Ephrin receptor Epidermal growth factor receptor Eukaryotic elongation factor 2 kinase Fibroblast growth factor receptor 1 Focal adhesion kinase 1 Focal adhesion kinase 1/vascular endothelial growth factor receptor 3 Glycogen synthase kinase-3 beta Hepatocyte growth factor receptor High affinity immunoglobulin gamma Fc receptor I High affinity nerve growth factor receptor Inhibitor of NF-kappa-B kinase (IKK) Insulin receptor MAP kinase-activated protein kinase 2 MAP kinase-interacting serine/threonine-protein kinase 2 Mast/stem cell growth factor receptor Kit Maternal embryonic leucine zipper kinase (MELK) Mitogen-activated protein kinase 1 Mitogen-activated protein kinase 14 Mitotic checkpoint serine/threonine-protein kinase BUB1 Non-receptor tyrosine-protein kinase TYK2 PKC alpha and beta-2 Pancreatic endoplasmic reticulum kinase (PERK) Proto-oncogene tyrosine-protein kinase ROS Proto-oncogene tyrosine-protein kinase receptor Ret Pyruvate dehydrogenase kinase isoenzyme 1 (PDK1) RAC-alpha serine/threonine-protein kinase AKT1 Serine/threonine-protein kinase Chk1 Serine/threonine-protein kinase MST4 Serine/threonine-protein kinase NEK6 Serine/threonine-protein kinase NIM1 Serine/threonine-protein kinase PAK 4 Serine/threonine-protein kinase PIM Serine/threonine-protein kinase PLK1 Serine/threonine-protein kinase haspin Tyrosine kinase non-receptor protein 2 Tyrosine-protein kinase ABL1 Tyrosine-protein kinase BRK Tyrosine-protein kinase JAK1 Tyrosine-protein kinase JAK2 Tyrosine-protein kinase JAK3 Tyrosine-protein kinase Lck Tyrosine-protein kinase Lyn Tyrosine-protein kinase SYK Tyrosine-protein kinase ZAP-70 Tyrosine-protein kinase receptor FLT3 Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2)	0	52	0	0	0	0	0	0	CHEMBL3298400
BDBM50212239	5-Hydroxytryptamine receptor 6 (5-HT6) 5-Hydroxytryptamine receptor 7 (5-HT7) 5-hydroxytryptamine receptor 1A (5-HT1A) 5-hydroxytryptamine receptor 1B 5-hydroxytryptamine receptor 2A 5-hydroxytryptamine receptor 2C 5-hydroxytryptamine receptor 3A Adenosine receptor A1 Adenosine receptor A2 Adenosine receptor A3 Adrenergic alpha1B Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor C-C chemokine receptor type 1 Cannabinoid receptor 1 Cannabinoid receptor 2 Cholecystokinin receptor D(1A) dopamine receptor D(2) dopamine receptor D(3) dopamine receptor Delta-type opioid receptor Dopamine D5 receptor Endothelin-1 receptor Histamine H1 receptor Histamine H2 Receptor Interleukin-8 receptors, CXCR2 KCNQ (Kv7) potassium channel Kappa-type opioid receptor Mu-type opioid receptor Muscarinic acetylcholine receptor M1 Muscarinic acetylcholine receptor M1/M5 chimeric protein Muscarinic acetylcholine receptor M2 Muscarinic acetylcholine receptor M3 Muscarinic acetylcholine receptor M4 Nociceptin receptor P2X purinoceptor 2 P2X purinoceptor 3 Potassium voltage-gated channel subfamily H member 2 Purinergic receptor P2Y2 Serotonin (5-HT) receptor Sigma non-opioid intracellular receptor 1 Sodium channel protein type 10 subunit alpha Sodium channel protein type 5 subunit alpha Sodium channel protein type 9 subunit alpha Sodium channel protein type X alpha subunit Transient receptor potential cation channel subfamily V member 1 Translocator protein Voltage-gated calcium channel subunit alpha Cav2.2 Voltage-gated sodium channel subunit alpha Nav1.2 (Nav1.2) Voltage-gated sodium channel subunit alpha Nav1.3 (Nav1.3) Voltage-gated sodium channel subunit alpha Nav1.8	0	75	0	0	0	0	0	0	5-(4-chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide A-803467 CHEMBL250699