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Compounds Sorted by Binding Targets per Compound

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Compounds Sorted Alphabetically

Compound Name (alphabetical)	Binding Targets	Enz. Inhib. Data							ITC Data	Alternate Compound Names
		Ki	IC50	Kd	EC50	Koff	Kon	Other
BDBM50001888	5-HT3A Serotonin Receptor 5-Hydroxytryptamine receptor 6 (5-HT6) 5-Hydroxytryptamine receptor 7 (5-HT7) 5-hydroxytryptamine receptor 1A (5-HT1A) 5-hydroxytryptamine receptor 2A 5-hydroxytryptamine receptor 2C 5-hydroxytryptamine receptor 7 (5HT7) ADRA1A ADRA2C ADRB2 Adenylate cyclase Adrenergic Alpha Adrenergic receptor alpha Adrenergic receptor alpha-2 Aldehyde oxidase Alpha-1 Adrenergic Receptor/ adrenergic receptor/ adrenergic receptor Alpha-1A adrenergic receptor Alpha-2A adrenergic receptor Alpha-2B adrenergic receptor Alpha-2C adrenergic receptor Bile salt export pump Bile salt export pump (BSEP) CHRM5 Calmodulin Cruzipain Cytochrome P450 1A Cytochrome P450 2C19 Cytochrome P450 2C9 Cytochrome P450 2D6 (2D6) Cytochrome P450 2J2 Cytochrome P450 3A D(1A) dopamine receptor D(2) dopamine receptor D(3) dopamine receptor DOPAMINE DRD1 DRD2 Dopamine D1 receptor Dopamine D2 receptor Dopamine D2 receptor and Serotonin 2a receptor (D2 and 5HT2a) Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor Dopamine D5 receptor Dopamine receptor Dopamine receptors; D2 & D4 HTR2B HTR2C HTR6 Histamine H1 receptor Histamine H4 receptor Histamine receptor (H3) Muscarinic acetylcholine receptor Muscarinic acetylcholine receptor M1 Muscarinic acetylcholine receptor M2 Muscarinic acetylcholine receptor M3 Muscarinic acetylcholine receptor M4 NADPH oxidase 1 P-glycoprotein 1 Pleiotropic ABC efflux transporter of multiple drugs Potassium voltage-gated channel subfamily H member 2 Prion protein Proteasome subunit alpha type-6 Serotonin (5-HT) receptor Serotonin 1 (5-HT1) receptor Serotonin 2 (5-HT2) receptor Serotonin receptor (2b and 2c) Serotonin receptor 2a and 2c (5HT2A and 5HT2C) Serum albumin Sigma non-opioid intracellular receptor 1 Sodium channel protein type 7 subunit alpha Sodium channel protein type I I alpha subunit Trypanothione reductase Twik-RElated Potassium (K+) channel 1 (TREK1) adrenergic Alpha2	218	66	4	3	0	0	0	0	(chloropromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine (chlorpromazine)[3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine 1-(2-Allyl-phenoxy)-3-isopropylamino-propan-2-ol 1N,1N-dimethyl-3-(2-chloro-10H-10-phenothiazinyl)-1-propanamine 3-(2-chloro-10H-phenothiazin-10-yl)-N,N-dimethylpropan-1-amine CHEMBL71 CHLORPROMAZINE CHLORPROMAZINE HIBENZATE CHLORPROMAZINE HYDROCHLORIDE CHLORPROMAZINE PHENOLPHTHALINATE CHLORPROMAZINE TANNATE Chlorpromazine;[3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine PROMAPAR SONAZINE THORAZINE [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine (chlor-promazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine( Chlorpromazine) [3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-amine(clorpromazine) chloropromazine
BDBM50235816	ALK tyrosine kinase receptor Activin receptor type-1 Aurora kinase A Aurora kinase B Axin-1/Glycogen synthase kinase-3 beta CAMK2A CDK7/Cyclin H/MNAT1 CaM kinase I delta CaM-kinase kinase beta Casein kinase I isoform alpha Cyclin-dependent kinase 2 Cyclin-dependent kinase 8 Cyclin-dependent kinase 9 Death-associated protein kinase 3 Dual specificity mitogen-activated protein kinase kinase 1/Mitogen-activated protein kinase 1/RAF proto-oncogene serine/threonine-protein kinase Dual specificity mitogen-activated protein kinase kinase 3 Dual specificity mitogen-activated protein kinase kinase; MEK1/2 Dual specificity protein kinase CLK2 Dual specificity tyrosine-phosphorylation-regulated kinase 1B Dual-specificity tyrosine-phosphorylation regulated kinase 1A Epidermal growth factor receptor Epithelial discoidin domain-containing receptor 1 Fibroblast growth factor receptor 1 Focal adhesion kinase 1 G protein-coupled receptor kinase 5 Glycogen synthase kinase-3 Hepatocyte growth factor receptor Hepatocyte growth factor-like protein High affinity nerve growth factor receptor Inhibitor of nuclear factor kappa-B kinase subunit epsilon Insulin receptor Insulin-like growth factor I receptor JNK2/JNK3 Leukocyte tyrosine kinase receptor Macrophage colony-stimulating factor 1 receptor Mitogen-activated protein kinase 2 Mitogen-activated protein kinase kinase kinase 10 Mitogen-activated protein kinase kinase kinase kinase 4 Neurotrophic tyrosine kinase receptor Platelet-derived growth factor receptor Platelet-derived growth factor receptor beta Protein kinase C iota type/zeta type Protein kinase C theta type Protein kinase C, PKC; classical/novel Proto-oncogene tyrosine-protein kinase Src Proto-oncogene tyrosine-protein kinase receptor Ret RAC-alpha serine/threonine-protein kinase AKT1 RAF serine/threonine protein kinase Rho-associated protein kinase 1 Rho-associated protein kinase 2 Ribosomal protein S6 kinase alpha-1/alpha-3 SRC Serine/threonine-protein kinase 16 Serine/threonine-protein kinase NEK2 Serine/threonine-protein kinase PAK 4 Serine/threonine-protein kinase PIM Serine/threonine-protein kinase Sgk1 Serine/threonine-protein kinase TAO2 Serine/threonine-protein kinase TBK1 Serine/threonine-protein kinase WEE1 Serine/threonine-protein kinase pim-2 Tyrosine kinase non-receptor protein 2 Tyrosine-protein kinase ABL1 Tyrosine-protein kinase BTK Tyrosine-protein kinase JAK2 Tyrosine-protein kinase JAK3 Tyrosine-protein kinase Lck Tyrosine-protein kinase SYK Tyrosine-protein kinase receptor TYRO3 Vascular endothelial growth factor receptor 1 Vascular endothelial growth factor receptor 2 and tyrosine-protein kinase TIE-2 (KDR and TIE2) c-Jun N-terminal kinase, JNK cGMP-dependent protein kinase 1 beta	0	75	0	1	0	0	0	0	CHEMBL4069365
BDBM82071	5-HT3A Serotonin Receptor 5-Hydroxytryptamine receptor 6 (5-HT6) 5-Hydroxytryptamine receptor 7 (5-HT7) 5-hydroxytryptamine receptor 1A (5-HT1A) 5-hydroxytryptamine receptor 1B 5-hydroxytryptamine receptor 1D 5-hydroxytryptamine receptor 2A 5-hydroxytryptamine receptor 2C ADENOSINE A2 ADRA2B ADRB2 Adenosine receptor A1 Adenosine transporter Adenylate cyclase Forskolin Adrenergic receptor beta Alpha adrenergic receptor 1A and 1B Alpha-1A adrenergic receptor Alpha-2A adrenergic receptor Bile salt export pump CHRM5 Calcium channel Cholecystokinin receptor D(2) dopamine receptor D(3) dopamine receptor DOPAMINE Dopamine D2 receptor/Serotonin 2 (5-HT2) receptor Dopamine Transporter (DAT) Ecto-5'-nucleotidase (e5'NT) GABA A GRIA3 Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1) Glutamate kainate Glycine, non-strychnine HTR4 Histamine H1 receptor Histamine H2 receptor Inositol Triphosphate Ionotropic glutamate receptor NMDA 1/2D Kappa-type opioid receptor Monoamine Oxidase Type B (MAO-B) Monoamine oxidase Monoamine transporters; Norepininephrine & dopamine Monoamine transporters; serotonin & dopamine Muscarinic acetylcholine receptor M1 Muscarinic acetylcholine receptor M2 Muscarinic acetylcholine receptor M3 Muscarinic acetylcholine receptor M4 Neurokinin 1 receptor Neurokinin 3 receptor Neuropeptide Y receptor type 1 Nicotinic Alpha-Bungarotoxin Nitric-oxide synthase, brain Nociceptin/mu opioid receptor Norepinephrine Monoamine transporters Norepinephrine transporter Opioid receptors; mu & delta Potassium Channel (Ca2+ dependent) Protein kinase C Renal Outer Medullary Potassium (ROMK) SOMATOSTATIN Serotonin (5-HT) receptor Serotonin receptor (2b and 2c) Serotonin receptor 2a and 2c (5HT2A and 5HT2C) Serum albumin Sigma non-opioid intracellular receptor 1 Sodium (Site 1) Sodium (Site 2) Sodium-dependent noradrenaline transporter Sodium-dependent serotonin transporter TACR2 Transporter Voltage-dependent N-type calcium channel subunit alpha-1B adrenergic Alpha2	161	42	4	0	0	0	0	0	CAS_93413-69-5 CAS_99300-78-4 NSC_62923 VENLAFAXINE Venlafaxine hydrochloride WY-45030 WY-45655
BDBM84745	5-Hydroxytryptamine receptor 6 (5-HT6) 5-Hydroxytryptamine receptor 7 (5-HT7) 5-hydroxytryptamine receptor 1A (5-HT1A) 5-hydroxytryptamine receptor 1B 5-hydroxytryptamine receptor 1D 5-hydroxytryptamine receptor 2A 5-hydroxytryptamine receptor 2C ADENOSINE A2 ADRA2B ADRB2 Adenosine receptor A1 Adenosine transporter Adenylate cyclase Forskolin Adrenergic receptor beta Alpha adrenergic receptor 1A and 1B Alpha-1A adrenergic receptor Alpha-2A adrenergic receptor Calcium channel Calcium channel (Type L) Cholecystokinin receptor Cytochrome P450 1A Cytochrome P450 2C19 Cytochrome P450 2C9 Cytochrome P450 2D6 (2D6) Cytochrome P450 3A D(2) dopamine receptor DOPAMINE Dopamine Transporter (DAT) Ecto-5'-nucleotidase (e5'NT) GABA A GRIA3 Gamma-aminobutyric acid receptor subunit alpha-1 (GABA(A) alpha-1) Glutamate kainate Glycine, non-strychnine HTR4 Histamine H1 receptor Histamine H2 receptor Histamine H3 receptor Histamine receptor (H3) Inositol Triphosphate Ionotropic glutamate receptor NMDA 1/2D Kappa-type opioid receptor Monoamine Oxidase Type B (MAO-B) Monoamine oxidase Monoamine transporters; serotonin & dopamine Muscarinic acetylcholine receptor M1 Muscarinic acetylcholine receptor M2 Neurokinin 1 receptor Neurokinin 3 receptor Neuropeptide Y receptor type 1 Nicotinic Alpha-Bungarotoxin Nitric-oxide synthase, brain Nociceptin/mu opioid receptor Norepinephrine transporter Opioid receptors; mu & delta Potassium Channel (Ca2+ dependent) Potassium voltage-gated channel subfamily H member 2 Protein kinase C Renal Outer Medullary Potassium (ROMK) SOMATOSTATIN Serotonin (5-HT) receptor Serotonin receptor (2b and 2c) Sigma non-opioid intracellular receptor 1 Sodium (Site 1) Sodium (Site 2) Sodium channel protein type 5 subunit alpha Sodium-dependent noradrenaline transporter Sodium-dependent serotonin transporter TACR2 Transporter Voltage-dependent N-type calcium channel subunit alpha-1B Voltage-gated potassium channel beta subunit Mink/subunit Kv7.1 Voltage-gated potassium channel subunit Kv4.3	100	52	0	0	0	0	0	0	CAS_136434-34-9 DULOXETINE LY-248686 LY248686