Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucagon receptor (Homo sapiens (Human)) | BDBM50068641 (2-(5-tert-Butyl-1H-benzoimidazol-2-ylsulfanyl)-1-(...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 5.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068631 (3-{2-[2-(3-Chloro-4-hydroxy-phenyl)-2-oxo-ethylsul...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.20E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068620 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068626 (3-{2-[2-(3,4-Dihydroxy-phenyl)-2-oxo-ethylsulfanyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068614 (2-(5-Benzyloxy-1H-benzoimidazol-2-ylsulfanyl)-1-(3...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068636 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Compound was evaluated for its binding affinity towards cloned human Glucagon receptor in BHK cells | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068627 (2-(5,6-Dichloro-1H-benzoimidazol-2-ylsulfanyl)-1-(...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068616 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(4-hydroxy-3-m...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM45955 (1-(3,4-dihydroxyphenyl)-2-[(6-methoxy-1H-benzimida...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.20E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM32012 (1-(3,4-Dihydroxy-phenyl)-2-(5-phenyl-4H-[1,2,4]tri...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068633 (1-(3,4-Dihydroxy-phenyl)-2-(5-nitro-1H-benzoimidaz...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | 5.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068630 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(4-hydroxy-phe...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >6.00E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068618 (2-(Benzothiazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phe...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | 7.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068617 (3-{2-[2-(3,4-Dihydroxy-phenyl)-2-oxo-ethylsulfanyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 9.50E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068634 (1-(3,4-Dihydroxy-phenyl)-2-(quinolin-2-ylsulfanyl)...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem | Article PubMed | 1.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068637 (1-(3,4-Dihydroxy-phenyl)-2-(4,5-diphenyl-1H-imidaz...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068643 (5-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-2-hyd...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068635 (2-(Benzooxazol-2-ylsulfanyl)-1-(3,4-dihydroxy-phen...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.50E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068628 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-hydroxy-phe...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068621 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dichloro-...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068619 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068642 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-phenyl-ethanon...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068615 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dimethoxy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068640 (1-(3,4-Dihydroxy-phenyl)-2-(1-methyl-1H-benzoimida...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068639 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068613 (4-[2-(1H-Benzoimidazol-2-ylsulfanyl)-1-hydroxy-eth...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068632 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50408685 (CHEMBL2112026) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068622 (4-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3,4-dihydroxy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068623 (1-(3,4-Dihydroxy-phenyl)-2-(1H-imidazol-2-ylsulfan...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068625 (3-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzo...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068624 (2-(1H-Benzoimidazol-2-ylsulfanyl)-1-(3-chloro-4-hy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50068629 (4-[2-(1H-Benzoimidazol-2-ylsulfanyl)-acetyl]-benzo...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | >5.00E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity towards cloned human glucagon receptor in BHK cells. | J Med Chem 41: 5150-7 (1999) Article DOI: 10.1021/jm9810304 BindingDB Entry DOI: 10.7270/Q24F1PV6 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Rattus norvegicus) | BDBM50122102 (3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity of the compound towards rat glucagon receptor | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Rattus norvegicus) | BDBM50110054 (3-Cyano-4-hydroxy-benzoic acid [1-[4-(4-isopropyl-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
Pfizer Global Research and Development Curated by ChEMBL | Assay Description Compound was evaluated in vitro for its inhibitory activity against rat glucagon receptor using [127I]-labeled glucagon | Bioorg Med Chem Lett 12: 663-6 (2002) BindingDB Entry DOI: 10.7270/Q2J67G77 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122102 (3-Cyano-4-hydroxy-benzoic acid [1-(2,3,5,6-tetrame...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | Purchase CHEMBL MCE PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 2.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122159 (CHEMBL152477 | Cyclopentanecarboxylic acid {4-[(3-...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 2.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122153 (CHEMBL156724 | Cyclopentanecarboxylic acid {4-[(3-...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 3.40 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50244455 ((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3,5-dichl...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity to human cloned GluR expressed in BHK cells | J Med Chem 51: 5387-96 (2008) Article DOI: 10.1021/jm7015599 BindingDB Entry DOI: 10.7270/Q2X34X9R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50245098 ((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3,5-dichloroph...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 4 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity to human cloned GluR expressed in BHK cells | J Med Chem 51: 5387-96 (2008) Article DOI: 10.1021/jm7015599 BindingDB Entry DOI: 10.7270/Q2X34X9R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50110074 (3-Chloro-4-hydroxy-benzoic acid [1-[4-(4-isopropyl...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122116 (3-Chloro-4-hydroxy-benzoic acid (4-{2-[4-(4-chloro...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | PubMed | n/a | n/a | 4.60 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122160 (3-Cyano-4-hydroxy-benzoic acid {4-[4-(4-chloro-ben...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 4.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50245102 ((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(3-methane...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 5 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity to human cloned GluR expressed in BHK cells | J Med Chem 51: 5387-96 (2008) Article DOI: 10.1021/jm7015599 BindingDB Entry DOI: 10.7270/Q2X34X9R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122135 (3-Chloro-4-hydroxy-benzoic acid [1-(2,3,5,6-tetram...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122142 (3-Chloro-4-hydroxy-benzoic acid [1-(2,4,6-trimethy...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.80 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122152 (4-[(3-Chloro-4-hydroxy-benzoyl)-hydrazonomethyl]-n...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 5.90 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50245099 ((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(2,2,4,4-t...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity to human cloned GluR expressed in BHK cells | J Med Chem 51: 5387-96 (2008) Article DOI: 10.1021/jm7015599 BindingDB Entry DOI: 10.7270/Q2X34X9R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50245060 ((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(4-trifluoromet...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 6 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description Binding affinity to human cloned GluR expressed in BHK cells | J Med Chem 51: 5387-96 (2008) Article DOI: 10.1021/jm7015599 BindingDB Entry DOI: 10.7270/Q2X34X9R | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucagon receptor (Homo sapiens (Human)) | BDBM50122158 (3-Cyano-4-hydroxy-benzoic acid (4-{2-[4-(4-bromo-p...) | PDB MMDB UniProtKB/SwissProt B.MOAD antibodypedia GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Patents Similars | PubMed | n/a | n/a | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a |
Novo Nordisk A/S Curated by ChEMBL | Assay Description In vitro binding affinity for recombinant human glucagon receptor (hGGR) in BHK cells | J Med Chem 45: 5755-75 (2002) BindingDB Entry DOI: 10.7270/Q26W99FD | |||||||||||
More data for this Ligand-Target Pair |
Displayed 1 to 50 (of 392 total ) | Next | Last >> |