Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92766 (PDF inhibitor, compound 8) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 53.7 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (docked) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92761 (PDF inhibitor, compound 3) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 117 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92764 (PDF inhibitor, compound 6) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 213 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (docked) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92760 (PDF inhibitor, compound 2) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | MMDB PC cid PC sid PDB UniChem Similars | PDB Article PubMed | 334 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92765 (PDF inhibitor, compound 7) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem Similars | Article PubMed | 650 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (docked) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92759 (PDF inhibitor, compound 1) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 6.31E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92762 (PDF inhibitor, compound 4) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | KEGG PC cid PC sid UniChem | Article PubMed | 2.59E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae (strain ATCC BAA-255 / R6...) | BDBM92763 (PDF inhibitor, compound 5) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | PC cid PC sid UniChem | Article PubMed | 3.17E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline | Assay Description Binding assay using PDF inhibitors. | Biochemistry 50: 6642-54 (2011) Article DOI: 10.1021/bi200655g BindingDB Entry DOI: 10.7270/Q2MS3RBV | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383996 (CHEMBL2032134) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.100 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383999 (CHEMBL2032137) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.120 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383966 (CHEMBL2032148) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.150 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383998 (CHEMBL2032136) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50384000 (CHEMBL2032138) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.190 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383997 (CHEMBL2032135) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.200 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383994 (CHEMBL2032132) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.220 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383987 (CHEMBL2032125) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.260 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383982 (CHEMBL2032119) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL MMDB PC cid PC sid PDB UniChem | PDB Article PubMed | n/a | n/a | 0.280 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | 3D Structure (crystal) | ||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383995 (CHEMBL2032133) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383988 (CHEMBL2032126) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.300 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383993 (CHEMBL2032131) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.310 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383968 (CHEMBL2032140) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.350 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50384003 (CHEMBL2032142) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.350 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50384002 (CHEMBL2032141) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.370 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383972 (CHEMBL2032146) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.380 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383969 (CHEMBL2032143) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.410 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383980 (CHEMBL2032117) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.430 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383992 (CHEMBL2032130) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.440 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383965 (CHEMBL2032129) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.460 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383967 (CHEMBL2032122) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.480 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383981 (CHEMBL2032118) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.5 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383986 (CHEMBL2032124) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.510 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383996 (CHEMBL2032134) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.520 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383985 (CHEMBL2032123) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.520 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383984 (CHEMBL2032121) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.540 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383989 (CHEMBL2032127) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.660 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383978 (CHEMBL2032115) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.700 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383973 (CHEMBL2032147) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.720 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383971 (CHEMBL2032145) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.770 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383976 (CHEMBL2032113) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.800 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383999 (CHEMBL2032137) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.860 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383995 (CHEMBL2032133) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.900 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383991 (CHEMBL2029376) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.910 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383997 (CHEMBL2032135) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 0.930 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383964 (CHEMBL2032111) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50384000 (CHEMBL2032138) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383970 (CHEMBL2032144) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL KEGG PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.10 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383979 (CHEMBL2032116) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383994 (CHEMBL2032132) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.20 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Staphylococcus aureus) | BDBM50383966 (CHEMBL2032148) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD DrugBank GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Staphylococcus aureus PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled assay | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Peptide deformylase (Streptococcus pneumoniae serotype 4 (strain ATCC B...) | BDBM50383977 (CHEMBL2032114) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 1.30 | n/a | n/a | n/a | n/a | n/a | n/a |
GlaxoSmithKline Curated by ChEMBL | Assay Description Inhibition of Streptococcus pneumoniae PDF assessed as formate release from fMAS peptide substrate after 20 mins by formate dehydrogenase coupled ass... | Bioorg Med Chem Lett 22: 4028-32 (2012) Article DOI: 10.1016/j.bmcl.2012.04.086 BindingDB Entry DOI: 10.7270/Q2K64K3V | |||||||||||
More data for this Ligand-Target Pair |
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