Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333520![]() (2-(1,4'-bipiperidin-1'-yl)-5-(6-methoxypyridin-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333511![]() (1-(3-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333521![]() (2-(1,4'-bipiperidin-1'-yl)-5-(6-methylpyridin-2-yl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 6.10 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333534![]() (1-(2-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 8.40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333515![]() (3-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333514![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3-chloro-5-methoxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 12 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333513![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3,5-dimethoxyphenyl)...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 15 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333516![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3-fluoro-5-methoxyph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 16 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333518![]() (5-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333524![]() (2-(1,4'-bipiperidin-1'-yl)-5-(2-methoxythiazol-5-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 28 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333519![]() (2-(1,4'-bipiperidin-1'-yl)-5-(pyridin-2-yl)-1,3,4-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 30 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333506![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3-methoxyphenyl)-1,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 31.9 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333533![]() (2-(1,4'-bipiperidin-1'-yl)-5-o-tolyl-1,3,4-thiadia...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333531![]() (2-(1,4'-bipiperidin-1'-yl)-5-(2-fluorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 36 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333535![]() (4-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 36.4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333536![]() (2-(1,4'-bipiperidin-1'-yl)-5-(4-fluorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 39 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333530![]() (2-(1,4'-bipiperidin-1'-yl)-5-(2-methoxyphenyl)-1,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333525![]() (2-(1,4'-bipiperidin-1'-yl)-5-(4-methoxyphenyl)-1,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 40.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333507![]() (3-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 42.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333504![]() (1-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 48.6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333509![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3-chlorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 49 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333517![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3,5-difluorophenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333510![]() (2-(1,4'-bipiperidin-1'-yl)-5-m-tolyl-1,3,4-thiadia...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333508![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3-fluorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 62 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333539![]() (1-(4-(5-(1,4'-bipiperidin-1'-yl)-1,3,4-thiadiazol-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 65 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333532![]() (2-(1,4'-bipiperidin-1'-yl)-5-(2-chlorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 69 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333512![]() (2-(1,4'-bipiperidin-1'-yl)-5-(3,5-dichlorophenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 72 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333505![]() (2-(1,4'-bipiperidin-1'-yl)-5-phenyl-1,3,4-thiadiaz...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 80.1 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333522![]() (2-(1,4'-bipiperidin-1'-yl)-5-(pyrimidin-2-yl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem | Article PubMed | 103 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333537![]() (2-(1,4'-bipiperidin-1'-yl)-5-(4-chlorophenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 161 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333526![]() (2-(4-ethylpiperazin-1-yl)-5-(4-methoxyphenyl)-1,3,...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 162 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333538![]() (2-(1,4'-bipiperidin-1'-yl)-5-p-tolyl-1,3,4-thiadia...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 163 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333527![]() (2-(4-cyclopentylpiperazin-1-yl)-5-(4-methoxyphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 182 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333523![]() (2-(1,4'-bipiperidin-1'-yl)-5-(1H-pyrazol-4-yl)-1,3...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents | Article PubMed | 192 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333529![]() (2-(4-methoxyphenyl)-5-(4-(pyrrolidin-1-yl)piperidi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 601 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Homo sapiens (Human)) | BDBM50333528![]() (2-(hexahydropyrrolo[1,2-a]pyrazin-2(1H)-yl)-5-(4-m...) | PDB Reactome pathway KEGG UniProtKB/SwissProt DrugBank antibodypedia GoogleScholar AffyNet ![]() | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 653 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Merck Research Laboratories Curated by ChEMBL | Assay Description Displacement of [3H]-N-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in HEK cells after 30 mins by scintillation count... | Bioorg Med Chem Lett 21: 861-4 (2011) Article DOI: 10.1016/j.bmcl.2010.11.065 BindingDB Entry DOI: 10.7270/Q20V8D24 | |||||||||||
More data for this Ligand-Target Pair |